Inventor
ALCACIO TIM EDWARD
US10 patents
Patents
10 patentsUS9051303B2Jun 9, 2015
Solid forms of (R)-1(2,2-difluorobenzo[D][1,3]dioxol-5-YL)-N-(1-(2,3-dihydroxypropyl-6-fluoro-2-(1-hydroxy-2-methylpropan-2-YL)-1H-indol-5-YL)-cyclopropanecarboxamide
VERTEX PHARMA59 citations97
US8802868B2Aug 12, 2014
Solid forms of (R)-1(2,2-difluorobenzo[D][1,3]dioxo1-5-yl)-N-(1-(2,3-dihydroxypropyl-6-fluoro-2-(1-hydroxy-2-methylpropan2-yl)-1H-Indol-5-yl)-Cyclopropanecarboxamide
VERTEX PHARMA68 citations97
US10906891B2Feb 2, 2021
Solid forms of (R)-1(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-N-(1-(2,3-dihydroxypropyl)-6-fluoro-2-(1-hydroxy-2-methylpropan-2-yl)-1H-indol-5-yl)cyclopropanecarboxamide
VERTEX PHARMA13 citations94
US10081621B2Sep 25, 2018
Solid forms of (R)-1(2,2-difluorobenzo[D][1,3]dioxol-5-yl)-N-(1-(2,3-dihydroxypropyl)-6-fluoro-2-(1-hydroxy-2-methylpropan-2-yl)-1H-indol-5-yl)cyclopropanecarboxamide
VERTEX PHARMA29 citations94
US10787472B2Sep 29, 2020
Prodrugs of pyridone amides useful as modulators of sodium channels
VERTEX PHARMA12 citations93
US10253054B2Apr 9, 2019
Prodrugs of pyridone amides useful as modulators of sodium channels
VERTEX PHARMA17 citations93
US9828397B2Nov 28, 2017
Prodrugs of pyridone amides useful as modulators of sodium channels
VERTEX PHARMA23 citations93
US9464102B2Oct 11, 2016
Prodrugs of pyridone amides useful as modulators of sodium channels
VERTEX PHARMA23 citations92
US11578062B2Feb 14, 2023
Solid forms of (R)-1(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-N-(1-(2,3-dihydroxypropyl)-6-fluoro-2-(1-hydroxy-2-methylpropan-2-yl)-1H-indol-5-yl)cyclopropanecarboxamide
VERTEX PHARMA4 citations85
US11773119B2Oct 3, 2023
Prodrugs of pyridone amides useful as modulators of sodium channels
VERTEX PHARMA2 citations72