Inventor
COATES DAVID ANDREW
US31 patents
⚠️ This page may combine multiple inventors who share the name “COATES DAVID ANDREW”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
LILLY CO ELI
24 patentsUS10287270B2May 14, 2019
Amino pyrimidine SSAO inhibitors
LILLY CO ELI5 citations82
US8962654B2Feb 24, 2015
3,4-dihydroisoquinolin-2(1H)-yl compounds
LILLY CO ELI9 citations80
US11834435B2Dec 5, 2023
SSTR4 agonist salts
LILLY CO ELI3 citations72
US10793552B2Oct 6, 2020
Amino pyrimidine ssao inhibitors
LILLY CO ELI1 citations71
US10464928B2Nov 5, 2019
Amino pyrimidine SSAO inhibitors
LILLY CO ELI2 citations71
US11124500B2Sep 21, 2021
Disubstituted pyrazole compounds
LILLY CO ELI2 citations70
US9637495B2May 2, 2017
CGRP receptor antagonists
LILLY CO ELI2 citations70
US10968214B2Apr 6, 2021
KRas G12C inhibitors
LILLY CO ELI2 citations68
US9828390B2Nov 28, 2017
Tetrahydropyrrolo[3,4-D][1,3]thiazine-derivative as BACE inhibitor
LILLY CO ELI2 citations68
US9708297B2Jul 18, 2017
CGRP receptor antagonists
LILLY CO ELI2 citations68
US12486249B2Dec 2, 2025
SSTR4 agonist salts
LILLY CO ELI0 citations61
US11066386B2Jul 20, 2021
CGRP receptor antagonists
LILLY CO ELI0 citations60
US11999722B2Jun 4, 2024
Disubstituted pyrazole compounds
LILLY CO ELI0 citations59
US12071423B2Aug 27, 2024
Processes and intermediate for the large-scale preparation of 2,4,6-trifluoro-N-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide hemisuccinate, and preparation of 2,4,6-trifluoro-N-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide acetate
LILLY CO ELI1 citations57
US11827618B2Nov 28, 2023
Processes and intermediate for the large-scale preparation of 2,4,6-trifluoro-n-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide hemisuccinate, and preparation of 2,4,6-trifluoro-n-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide acetate
LILLY CO ELI0 citations57
US10611751B2Apr 7, 2020
Dopamine D1 receptor positive allosteric modulators
LILLY CO ELI1 citations57
US11655242B2May 23, 2023
Glucagon-like peptide1 receptor agonists
LILLY CO ELI1 citations56
US12252491B2Mar 18, 2025
IL-17A inhibitors
LILLY CO ELI0 citations53
US11746115B2Sep 5, 2023
Solid forms of 7-[[(1S)-1-[4-[(1S)-2-cyclopropyl-1-(4-prop-2-enoylpiperazin-1-yl)ethyl]phenyl]ethyl]amino]-1-ethyl-4H-pyrimido[4,5-d][1,3]oxazin-2-one
LILLY CO ELI0 citations53
US10323019B2Jun 18, 2019
Pyrazolylaminobenzimidazole derivatives as JAK inhibitors
LILLY CO ELI0 citations51
US10080758B2Sep 25, 2018
Tosylate salt of N-[3-[(4aR,7aS)-2-amino-6-(5-fluoropyrimidin-2-yl)-4,4a,5,7-tetrahydropyrrolo[3,4-d][1,3]thiazin-7a-yl]-4-fluoro-phenyl]-5-methoxy-pyrazine-2-carboxamide
LILLY CO ELI0 citations47
US10934280B2Mar 2, 2021
Condensed thiophene derivatives useful as NaPi-IIb inhibitors
LILLY CO ELI0 citations44
US9920056B2Mar 20, 2018
2-oxo-1,3,8-triazaspiro[4.5]decan-3-yl] carboxylic acid derivatives
LILLY CO ELI0 citations44
US10787460B2Sep 29, 2020
(E)-1-(4-(dimethylamino)but-2-enoyl)pyrrolidin-3-yl 4-((3-isopropyl-5-methylpyrazolo[1,5-a]pyrimidin-7-yl)amino)piperidine-1-carboxylate for inhibiting CDK7
LILLY CO ELI0 citations42
WARNER LAMBERT CO
2 patentsUS6605729B1Aug 12, 2003
Crystalline forms of [R-(R*,R*)]-2-(4-fluorophenyl)-β,δ-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid calcium salt (2:1)
WARNER LAMBERT CO104 citations94
US7144915B2Dec 5, 2006
Crystalline forms of [R-(R*,R*)]-2-(4-fluorophenyl)-β,δ-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid calcium salt (2:1)
WARNER LAMBERT CO9 citations70