Inventor
KRUSE CORNELIS G
NL53 patents
⚠️ This page may combine multiple inventors who share the name “KRUSE CORNELIS G”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
SOLVAY PHARM BV
21 patentsUS6476060B2Nov 5, 2002
4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity
SOLVAY PHARM BV78 citations94
US6974810B2Dec 13, 2005
4,5-Dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity
SOLVAY PHARM BV31 citations91
US7319110B2Jan 15, 2008
1H-1,2,4-triazole-3-carboxamide derivatives having cannabinoid-CB1 receptor agonistic, partial agonistic, inverse agonistic or antagonistic activity
SOLVAY PHARM BV14 citations83
US7528162B2May 5, 2009
4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity
SOLVAY PHARM BV20 citations82
US6828325B2Dec 7, 2004
Phenylpiperazines
SOLVAY PHARM BV13 citations82
US7728018B2Jun 1, 2010
Sulfonylpyrazole and sulfonylpyrazoline carboxamidine derivatives as 5-HT6 antagonists
SOLVAY PHARM BV11 citations81
US7524867B2Apr 28, 2009
Tetrasubstituted imidazole derivatives as cannabinoid CB1 receptor modulators with a high CB1/CB2 receptor subtype selectivity
SOLVAY PHARM BV10 citations79
US7109216B2Sep 19, 2006
1H-imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity
SOLVAY PHARM BV14 citations79
US6911448B2Jun 28, 2005
Piperazine and piperidine compounds
SOLVAY PHARM BV5 citations71
US7964728B2Jun 21, 2011
Azaindole derivatives with a combination of partial nicotinic acetyl-choline receptor agonism and dopamine reuptake inhibition
SOLVAY PHARM BV2 citations61
US7786144B2Aug 31, 2010
Sulphur containing pyrazole derivatives as selective cannabinoid CB1 receptor antagonists
SOLVAY PHARM BV2 citations61
US7608718B2Oct 27, 2009
4,5-dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity
SOLVAY PHARM BV2 citations61
US7186741B2Mar 6, 2007
Neurotensin active 2,3,diaryl-pyrazolidine derivatives
SOLVAY PHARM BV6 citations58
US7067513B1Jun 27, 2006
Phenylpiperazines
SOLVAY PHARM BV3 citations58
US7495108B2Feb 24, 2009
Imidazoline derivatives having CB1-antagonistic activity
SOLVAY PHARM BV0 citations51
US7173044B2Feb 6, 2007
Imidazoline derivatives having CB1-antagonistic activity
SOLVAY PHARM BV0 citations51
US7498348B2Mar 3, 2009
1 H-imidazole derivatives as cannabinoid receptor modulators
SOLVAY PHARM BV0 citations50
US7271189B2Sep 18, 2007
1H-imidazole derivatives as cannabinoid receptor modulators
SOLVAY PHARM BV0 citations50
US7605162B2Oct 20, 2009
Phenylpiperazine
SOLVAY PHARM BV0 citations48
US7371769B2May 13, 2008
Tetrahydropyridin-4-yl indoles with a combination of affinity for dopamine-D2 receptors and serotonin reuptake sites
SOLVAY PHARM BV1 citations48
US7696383B2Apr 13, 2010
N-oxides of venlafaxine and o-desmethylvenlafaxine as prodrugs
SOLVAY PHARM BV0 citations43
DUPHAR INT RES
15 patentsUS5424313AJun 13, 1995
Bibyclic heteroacrylpiperazine derivatives having psychotropic activity, and pharmaceutical compositions containing these derivatives
DUPHAR INT RES62 citations93
US4772604ASep 20, 1988
Phenyl-substituted (N-piperazinyl) methylazoles for treating affections in the central nervous system
DUPHAR INT RES26 citations92
US6214829B1Apr 10, 2001
Piperazine compounds, their preparation, and methods of using them
DUPHAR INT RES34 citations91
US4782061ANov 1, 1988
Method of treating psychotropic conditions employing substituted piperazine compounds
DUPHAR INT RES38 citations91
US6335326B1Jan 1, 2002
Benzisoxazole derivatives having d4-antagonistic activity
DUPHAR INT RES9 citations72
US6391896B1May 21, 2002
3-Tetrahydropyridin-4-yl indoles for treatment of psychotic disorders
DUPHAR INT RES12 citations71
US6090812AJul 18, 2000
Piperazine and piperidine compounds
DUPHAR INT RES13 citations71
US6281216B1Aug 28, 2001
2-aminoquinoline derivatives having d4-agonistic activity
DUPHAR INT RES2 citations60
US5189219AFeb 23, 1993
Method for the preparation of erythro vicinal amino-alcohols
DUPHAR INT RES2 citations60
US6780864B1Aug 24, 2004
Piperazine and piperidine compounds
DUPHAR INT RES3 citations57
US4791132ADec 13, 1988
Phenyl, Pyrrolidin-2-yl substituted pyrroles having antipsychotic properties
DUPHAR INT RES1 citations51
USRE41425EJul 6, 2010
Piperazine and piperidine compounds
DUPHAR INT RES0 citations50
USRE35128EDec 19, 1995
Method for the preparation of erythro vicinyl amino-alcohols
DUPHAR INT RES0 citations49
US5348949ASep 20, 1994
Method of preparing N-oxo-tetrahydro-β-carbolines
DUPHAR INT RES0 citations45
US5106840AApr 21, 1992
Method of preparing n-oxo-tetrahydro-beta-carbolines
DUPHAR INT RES0 citations45
STOIT AXEL
3 patentsUS8252930B2Aug 28, 2012
Azaindole derivatives with a combination of partial nicotinic acetyl-choline receptor agonism and dopamine reuptake inhibition
STOIT AXEL9 citations81
US8586606B2Nov 19, 2013
Heterocyclic compounds with affinity to muscarinic receptors
STOIT AXEL0 citations49
US8084473B2Dec 27, 2011
Heterocyclic compounds with affinity to muscarinic receptors
STOIT AXEL0 citations45
LANGE JOSEPHUS H M
3 patentsUS8138174B2Mar 20, 2012
Compounds with a combination of cannabinoid CB1 antagonism and serotonin reuptake inhibition
LANGE JOSEPHUS H M2 citations61
US8063062B2Nov 22, 2011
Compounds with a combination of cannabinoid-CB1 antagonism and acetylcholinesterase inhibition
LANGE JOSEPHUS H M1 citations47
US8461184B2Jun 11, 2013
Sulphur containing pyrazole derivatives as selective cannabinoid CB1 receptor antagonists
LANGE JOSEPHUS H M0 citations44
SOLVAY PHARMACEUTICALS INC
3 patentsUS7297699B2Nov 20, 2007
Piperazine and piperidine compounds
SOLVAY PHARMACEUTICALS INC0 citations49
US7456182B2Nov 25, 2008
Phenylpiperazines
SOLVAY PHARMACEUTICALS INC0 citations47
US7342032B2Mar 11, 2008
Thiazole derivatives having CB1-antagonistic, agonistic or partial agonistic activity
SOLVAY PHARMACEUTICALS INC1 citations47
VAN LOEVEZIJN ARNOLD
2 patentsFEENSTRA ROELOF W
1 patentTERWEL LOUISE
1 patentABBOTT HEALTHCARE PRODUCTS BV
1 patentShowing the top 50 of 53 patents by PatentIndex Score.