Inventor
MACLEOD ANGUS MURRAY
GB50 patents
⚠️ This page may combine multiple inventors who share the name “MACLEOD ANGUS MURRAY”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
MERCK SHARP & DOHME
43 patentsUS5885999AMar 23, 1999
Serine derivatives and their use as therapeutic agents
MERCK SHARP & DOHME103 citations97
US6136824AOct 24, 2000
1-piperidinyl-propan-2-derivatives and their use as therapeutic agents
MERCK SHARP & DOHME61 citations96
US6200975B1Mar 13, 2001
Substituted 1,2,4-triazolo[3,4-a]phthalazine derivatives as GABA alpha 5 ligands
MERCK SHARP & DOHME42 citations92
US5760018AJun 2, 1998
Gem-disubstituted azacyclic tachykinin antagonists
MERCK SHARP & DOHME59 citations92
US7381725B2Jun 3, 2008
Pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME17 citations84
US7030128B2Apr 18, 2006
Imidazo-pyrimidine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME11 citations84
US6211219B1Apr 3, 2001
Aminocyclohexane derivatives as 5-HT receptor agonists
MERCK SHARP & DOHME18 citations84
US5977116ANov 2, 1999
Piperazine, piperidine and tetrahydropyridine derivatives
MERCK SHARP & DOHME19 citations84
US6559166B1May 6, 2003
Phenylsulphonyl derivatives as 5-HT receptor ligands
MERCK SHARP & DOHME14 citations82
US5693640ADec 2, 1997
Pyridazino-indole derivatives
MERCK SHARP & DOHME7 citations74
US5686463ANov 11, 1997
Oxadiazoles useful in the treatment of senile dementia
MERCK SHARP & DOHME8 citations74
US6900209B2May 31, 2005
Nitrogen substituted 1,2,4-triazolo[3,4-a]phthalazine derivatives for enhancing cognition
MERCK SHARP & DOHME8 citations73
US5981529ANov 9, 1999
Substituted indolylpropyl-piperazine derivatives as 5-HT1D α agonists
MERCK SHARP & DOHME13 citations73
US5849746ADec 15, 1998
Substituted 1,4-piperazine-heteroaryl derivatives as 5-HT1D receptor agonists
MERCK SHARP & DOHME16 citations73
US5811431ASep 22, 1998
Spiro-substituted azacyclic derivatives and their use as therapeutic agents
MERCK SHARP & DOHME8 citations73
US5719149AFeb 17, 1998
Morpholine derivatives and their use as therapeutic agents
MERCK SHARP & DOHME8 citations73
US5661162AAug 26, 1997
4-aminomethyl/thiomethyl/sulfonylmethyl-4-phenylpiperdines as tachykinin receptor antagonists
MERCK SHARP & DOHME17 citations73
US6465462B1Oct 15, 2002
Substituted triazolo pyridazine derivatives as inverse agonists of the GABAAα5 receptor subtype
MERCK SHARP & DOHME9 citations72
US7482457B2Jan 27, 2009
Substituted quinoline-4-carboxylic hydrazides as NK-2/NK-3 receptor ligands
MERCK SHARP & DOHME2 citations63
US6054456AApr 25, 2000
Substituted piperazine derivatives
MERCK SHARP & DOHME5 citations63
US5710161AJan 20, 1998
Triazole derivatives and their use as therapeutic agents
MERCK SHARP & DOHME5 citations63
US5668153ASep 16, 1997
Piperidine derivatives and their use as therapeutic agents
MERCK SHARP & DOHME2 citations63
US5665883ASep 9, 1997
Aralkoxy and aralkylthio substituted azacyclic compounds as tachykinin antagonists
MERCK SHARP & DOHME6 citations63
US7144887B2Dec 5, 2006
Substituted 1,2,3-triazolo[1,5-a]quinazolines for enhancing cognition
MERCK SHARP & DOHME3 citations62
US6355638B1Mar 12, 2002
Pyrazolo[1,5-d][1,2,4] triazines for enhancing cognition
MERCK SHARP & DOHME4 citations62
US6127388AOct 3, 2000
Azetidine, pyrrolidine and piperidine derivatives as 5-HT1D receptor agonists
MERCK SHARP & DOHME6 citations62
US5998416ADec 7, 1999
Piperazine, piperidine and tetrahydropyridine derivatives as 5-HT receptor agonists
MERCK SHARP & DOHME2 citations62
US5663352ASep 2, 1997
4-phenyl-4-phenylpropyl(enyl)-piperidines as tachykinin antagonists
MERCK SHARP & DOHME2 citations62
US6949549B2Sep 27, 2005
Imidazolophthalazine derivatives as ligands for GABAA receptors
MERCK SHARP & DOHME2 citations61
US6054469AApr 25, 2000
Substituted tetrahydropyridine derivatives acting on 5-HT receptors
MERCK SHARP & DOHME3 citations61
US6777430B2Aug 17, 2004
Phenylsulphonyl derivatives as 5-HT receptor ligands
MERCK SHARP & DOHME2 citations60
US5994374ANov 30, 1999
Substituted 1-indolylpropyl-4-benzyl-tetrahydropyridine derivatives
MERCK SHARP & DOHME2 citations60
US6262103B1Jul 17, 2001
Thienycyclohexanone derivatives as ligands of the GABAA α5 receptor subtype
MERCK SHARP & DOHME2 citations58
US6946461B2Sep 20, 2005
Imidazolophthalazine derivatives as ligands for GABAA receptors
MERCK SHARP & DOHME1 citations52
US6448249B1Sep 10, 2002
Substituted 1,2,4-triazolo[3,4-A]phthalazine derivatives as GABAα5 ligands
MERCK SHARP & DOHME1 citations52
US5889008AMar 30, 1999
Substituted 1-indolylpropyl-4-phenethylpiperazadine derivatives
MERCK SHARP & DOHME1 citations51
US5674889AOct 7, 1997
Aromatic compounds, compositions containing them and their use in therapy
MERCK SHARP & DOHME1 citations50
US7468393B2Dec 23, 2008
Diarylsulfones as 5-HT2A antagonists
MERCK SHARP & DOHME1 citations49
US7022724B2Apr 4, 2006
Cognition enhancing derivatives of isoxazole triazoloindane GABA-A α5 receptor subunit ligands
MERCK SHARP & DOHME1 citations48
US6087372AJul 11, 2000
Method of enhancing cognition with 2-(4-methoxyphenyl)-pyrazolo[4,3-c]quinolin-3-one
MERCK SHARP & DOHME0 citations44
US7060710B2Jun 13, 2006
Isoxazole pyrazoloindane derivatives as cognition enhancing GABAA α5 subtype ligands
MERCK SHARP & DOHME0 citations41
US6048878AApr 11, 2000
Substituted piperidine derivatives as selective agonists of 5-HT receptors
MERCK SHARP & DOHME0 citations41
US7271191B2Sep 18, 2007
Pyrazole derivatives as gamma-secretase inhibitors useful in the treatment of Alzheimer's disease
MERCK SHARP & DOHME0 citations40