Inventor
DESIMONE ROBERT W
US29 patents
⚠️ This page may combine multiple inventors who share the name “DESIMONE ROBERT W”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
NEUROGEN CORP
20 patentsUS6723730B2Apr 20, 2004
Capsaicin receptor ligands
NEUROGEN CORP105 citations96
US6271241B1Aug 7, 2001
Cycloalkyl and aryl fused aminoalkyl-imidazole derivatives: modulators and GLP-1 receptors
NEUROGEN CORP65 citations96
US6143760ANov 7, 2000
Substituted 4-oxo-napthyridine-3-carboxamides: GABA brain receptor ligands
NEUROGEN CORP47 citations96
US6646124B2Nov 11, 2003
Substituted 4-oxo-napthyridine-3-carboxamides: GABA brain receptor ligands
NEUROGEN CORP24 citations92
US6399604B1Jun 4, 2002
Substituted 4-OXO-napthyridine-3-carboxamides; GABA brain receptor ligands
NEUROGEN CORP33 citations92
US6380210B1Apr 30, 2002
Heteroaryl fused aminoalkyl-imidazole derivatives: selective modulators of GABAa receptors
NEUROGEN CORP37 citations92
US6127395AOct 3, 2000
Substituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligands
NEUROGEN CORP18 citations92
US5637724AJun 10, 1997
Substituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligands
NEUROGEN CORP21 citations92
US6194427B1Feb 27, 2001
Substituted cycloalkyl-4-Oxonicotinic carboxamides; gaba brain receptor ligands
NEUROGEN CORP19 citations91
US7160879B2Jan 9, 2007
Melanin concentrating hormone receptor ligands: substituted 2-(4-benzyl-piperazin-1-ylmethyl)- and 2-(4-benzyl-diazepan-1-ylmethyl)-1H-benzoimidazole analogues
NEUROGEN CORP26 citations90
US5936095AAug 10, 1999
Substituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligands
NEUROGEN CORP15 citations82
US5849927ADec 15, 1998
Substituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligands
NEUROGEN CORP16 citations82
US5637725AJun 10, 1997
Substituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligands
NEUROGEN CORP16 citations82
US6448259B1Sep 10, 2002
Substituted cycloalkyl-4-oxonicotinic carboxamides; GABA brain receptor ligands
NEUROGEN CORP13 citations72
US6358949B1Mar 19, 2002
Aryl and hetroaryl fused aminoalkyl-imidazole derivatives: selective modulators of bradykinin B2 receptors
NEUROGEN CORP10 citations72
US6156898ADec 5, 2000
Substituted 1,4-dihydro-4-oxonicotinic carboxamides; GABA brain receptor ligands
NEUROGEN CORP13 citations70
US6972293B2Dec 6, 2005
Heteroaryl fused aminoalkyl-imidazole derivatives: selective modulators of GABAa receptors
NEUROGEN CORP3 citations62
US6627624B1Sep 30, 2003
Aryl fused aminoalkyl-imidazole derivatives: selective modulators of GABAa receptors
NEUROGEN CORP4 citations62
US6906075B2Jun 14, 2005
Melanin concentrating hormone receptor ligands: substituted benzoimidazole analogues
NEUROGEN CORP3 citations60
US7241765B2Jul 10, 2007
Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
NEUROGEN CORP0 citations50
CGI PHARMACEUTICALS INC
8 patentsUS7393848B2Jul 1, 2008
Certain heterocyclic substituted imidazo[1,2-A]pyrazin-8-ylamines and methods of inhibition of Bruton's tyrosine kinase by such compounds
CGI PHARMACEUTICALS INC67 citations98
US7160885B2Jan 9, 2007
Certain 6, 8-(heteroaryl or aryl) disubstituted imidazo[1,2-a]pyrazines as modulators of Hsp90 complex activity
CGI PHARMACEUTICALS INC77 citations97
US7405295B2Jul 29, 2008
Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of Bruton's tyrosine kinase by such compounds
CGI PHARMACEUTICALS INC98 citations95
US7312341B2Dec 25, 2007
6-aryl-imidazo[1,2-a] pyrazin-8-ylamines, method of making, and method of use thereof
CGI PHARMACEUTICALS INC50 citations92
US7189723B2Mar 13, 2007
Certain 8-heteroaryl-6-phenyl-imidazo[1,2-a]pyrazines as modulators of kinase activity
CGI PHARMACEUTICALS INC48 citations92
US7259164B2Aug 21, 2007
Certain substituted imidazo[1,2-a]pyrazines, as modulators of kinase activity
CGI PHARMACEUTICALS INC46 citations90
US7015227B2Mar 21, 2006
Certain amino-substituted monocycles as kinase modulators
CGI PHARMACEUTICALS INC21 citations84
US7625931B2Dec 1, 2009
Certain substituted diphenyl ureas, as modulators of kinase activity
CGI PHARMACEUTICALS INC0 citations39