Inventor
SCHWARK JAN-ROBERT
DE48 patents
⚠️ This page may combine multiple inventors who share the name “SCHWARK JAN-ROBERT”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
HOECHST AG
39 patentsUS5852046ADec 22, 1998
Benzo-fused heterocyclic compounds having a 5-membered ring processes for their preparation their use as medicaments their use as diagnostic agents and medicaments containing them
HOECHST AG82 citations96
US5866610AFeb 2, 1999
Substituted benzoylguanidines, process for their preparation, their use as a pharmaceutical as inhibitors of the cellular NA+/H+ exchange or as a diagnostic, and pharmaceutical containing them
HOECHST AG55 citations93
US5708034AJan 13, 1998
Substituted sulfonimidamides, processes for their preparation, their use as a medicament or diagnostic, and medicament comprising them
HOECHST AG42 citations93
US5698581ADec 16, 1997
Substituted N-heteroaroylguanidines, a process for their preparation, their use as a medicament or diagnostic agent, and a medicament containing them
HOECHST AG38 citations93
US5571842ANov 5, 1996
Perfluoroalkyl-substituted, benzoylguanidines, a process for their preparation, their use as a medicament or diagnostic agent, and a medicament containing them
HOECHST AG36 citations93
US5547953AAug 20, 1996
Substituted 1-oxo-1,2-dihydroisoquinolinoylguanidines and 1,1-dioxo-2H-1,2-benzothiazinoylguanidines, a process for their preparation, their use as medicaments or diagnostic agents, and medicaments containing them
HOECHST AG24 citations93
US6335451B1Jan 1, 2002
Five-membered heterocycles having biphenylsulfonyl substitution, with sulfonylcyanamide side chain, compositions containing them, and methods of using them
HOECHST AG26 citations92
US6005010ADec 21, 1999
Phenyl-substituted alkenylcarboxylic acid guanidides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
HOECHST AG45 citations92
US6057322AMay 2, 2000
Basically-substituted benzoylguanidines, a process for preparing them, their use as a medicament or diagnostic agent, and a medicament containing them
HOECHST AG19 citations84
US6087304AJul 11, 2000
Substituted 2-naphthoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
HOECHST AG11 citations74
US6025349AFeb 15, 2000
Phenyl.-substituted alkenylcarboguanidides carrying perfluoroalkyl groups, a process for their preparation, their use as a medicament or diagnostic agent, and also a medicament containing them
HOECHST AG14 citations74
US5965744AOct 12, 1999
Ortho-substituted benzoylguanidines, including composition and methods of using them
HOECHST AG10 citations74
US5883133AMar 16, 1999
Substituted cinnamic acid guanidides, a process for their preparation, their use as medicaments or diagnostic agents and medicaments comprising them
HOECHST AG16 citations74
US5747541AMay 5, 1998
Substituted benzoylguanidines, a process for their preparation, their use as medicament of diagnostic agent, and medicament comprising them
HOECHST AG15 citations74
US5719169AFeb 17, 1998
Substituted benzoylguanidines, their use as a medicament or diagnostic, and medicament containing them
HOECHST AG14 citations74
US5679712AOct 21, 1997
Substituted benzoylguanidines, process for their preparation, their use as a pharmaceutical or diagnostic, and pharmaceutical containing them
HOECHST AG15 citations74
US5641792AJun 24, 1997
Benzoylguanidines substituted by heterocyclic N-oxide, process for their preparation and pharmaceutical compositions containing them
HOECHST AG8 citations74
US5631293AMay 20, 1997
Preparation of amino acid-substituted benzoylguanidines as diagnostic agents
HOECHST AG12 citations74
US5567734AOct 22, 1996
Phenyl-substituted alkylcarboguanidides carrying perfluoroalkyl groups, a process for their preparation, their use as a medicament or a diagnostic agent, and a medicament containing them
HOECHST AG14 citations74
US5559153ASep 24, 1996
Urea-substituted benzoylguanidines, process for their preparation, their use as pharmaceutical or diagnostic, and pharmaceutical containing them
HOECHST AG8 citations74
US5900436AMay 4, 1999
Substituted indanylidineacetylguanidines, processes for their preparation, their use as medicaments or diagnostics and medicaments containing them
HOECHST AG12 citations69
US6632840B1Oct 14, 2003
Monoacyl-substituted guanidines, a process for their preparation, their use as a medicament or diagnostic aid, and pharmaceutical compositions containing them
HOECHST AG2 citations63
US6504057B2Jan 7, 2003
Fluorophenyl-substituted alkenylcarboxylic acid guanidides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
HOECHST AG5 citations63
US6093729AJul 25, 2000
Substituted bicyclic heteroaroylguanidines, a process for their preparation, their use as a medicament or a diagnostic agent, and a medicament containing them
HOECHST AG3 citations63
US6011063AJan 4, 2000
Ortho-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament comprising them
HOECHST AG2 citations63
US6001881ADec 14, 1999
Ortho-substituted benzoylguanidines, a process for their preparation, their use as a medicament or diagnostic agent, and a medicament comprising them
HOECHST AG5 citations63
US5856344AJan 5, 1999
Sulfonylamino-substituted benzoylguanidines, a process for their preparation, their use as a medicament or diagnostic aid, and medicament containing them
HOECHST AG4 citations63
US5849775ADec 15, 1998
Substituted benzoylguanidines process for their preparation, their use as a medicament or diagnostic, and pharmaceutical containing them
HOECHST AG2 citations63
US5756535AMay 26, 1998
Substituted thiophenylalkenylcarboxylic acid guanidines, processes for their preparation, their use as a medicament or diagnositc, and a medicament containing them
HOECHST AG4 citations63
US5753710AMay 19, 1998
Substituted benzyloxycarbonylguanidines, a process for their preparation, their use as a medicament or diagnostic, and a medicament containing them
HOECHST AG3 citations63
US6486189B2Nov 26, 2002
Five-membered heterocycles having biphenylsulfonyl substitution, process for their preparation, their use as a medicament or diagnostic, and medicament comprising them
HOECHST AG2 citations62
US6436999B1Aug 20, 2002
Diacyl-substituted guanidines, a process for their preparation, their use as medicine or diagnostic aid, and medicine containing them
HOECHST AG0 citations52
US6075054AJun 13, 2000
Ortho-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament comprising them
HOECHST AG0 citations52
US6022899AFeb 8, 2000
Substituted benzyloxy-carbonylguanidines, a process for their preparation, their use as a medicament or diagnostic, and a medicament containing them
HOECHST AG1 citations52
US5998481ADec 7, 1999
Fluoroalkyl/alkenyl-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
HOECHST AG0 citations52
US5869531AFeb 9, 1999
Fluoroalkyl substituted benzoylguanidines
HOECHST AG0 citations52
US5856574AJan 5, 1999
Ortho-subsituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
HOECHST AG1 citations52
US6153651ANov 28, 2000
Ortho-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament comprising them
HOECHST AG0 citations42
US5731350AMar 24, 1998
Substituted benzenedicarboxylic acid diguanides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
HOECHST AG0 citations42
AVENTIS PHARMA GMBH
8 patentsUS6825231B2Nov 30, 2004
Substituted norbornylamino derivatives, processes for their preparation, their use as medicaments or diagnostics, and a medicament comprising them
AVENTIS PHARMA GMBH8 citations74
US6156800ADec 5, 2000
4-fluoroalkyl-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
AVENTIS PHARMA GMBH9 citations74
US6166002ADec 26, 2000
Substituted phenylalkenoylguanidines, process for their preparation, and their use in medicaments and in diagnostics
AVENTIS PHARMA GMBH14 citations71
US6372917B1Apr 16, 2002
Biphenylsulfonyl-substituted imidazole derivatives, their preparation process, their use as a drug or diagnostic agent and drug containing them
AVENTIS PHARMA GMBH6 citations63
US6369236B1Apr 9, 2002
Imidazole derivatives with biphenylsulfonyl substitution method for preparing them and their use as a drug or diagnostic agent
AVENTIS PHARMA GMBH5 citations63
US6573288B1Jun 3, 2003
Substituted sulphonyl cyanamides, method for producing same and their use as medicament
AVENTIS PHARMA GMBH5 citations62
US6369069B1Apr 9, 2002
Biphenylsulfonyl cyanamides, method for the production thereof and their utilization as a medicament
AVENTIS PHARMA GMBH3 citations62
US6262123B1Jul 17, 2001
Ortho-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament comprising them
AVENTIS PHARMA GMBH0 citations42