Inventor
DIELS GASTON S M
BE17 patents
Patents
17 patentsUS5258380ANov 2, 1993
(4-piperidinylmethyl and -hetero)purines
JANSSEN PHARMACEUTICA NV122 citations98
US5041448AAug 20, 1991
(4-piperidinylmethyl and -hetero) purines
JANSSEN PHARMACEUTICA NV128 citations98
US4695575ASep 22, 1987
4-[(bicycle heterocyclyl)-methyl and -hetero]-piperidines
JANSSEN PHARMACEUTICA NV113 citations96
US5360807ANov 1, 1994
Substituted thiazolyl and substituted pyridinyl derivatives
JANSSEN PHARMACEUTICA NV22 citations92
US5468743ANov 21, 1995
Imidazo[2,1-b]benzazepine derivatives, compositions and method of use
JANSSEN PHARMACEUTICA NV32 citations91
US4988689AJan 29, 1991
((Pharmacologically active bicyclic heterocyclic)methyl and -heteroatom) substituted hexahydro-1H-azepines and pyrrolidines
JANSSEN PHARMACEUTICA NV31 citations90
US5086056AFeb 4, 1992
2-(heterocyclylalkyl)imidazopyridines
JANSSEN PHARMACEUTICA NV16 citations81
US4946843AAug 7, 1990
2-(heterocyclylalkyl)imidazopyridines
JANSSEN PHARMACEUTICA NV22 citations81
US4943580AJul 24, 1990
Anti-histaminic benzimidazole, imidazopyridine and purine derivatives
JANSSEN PHARMACEUTICA NV8 citations73
US4839374AJun 13, 1989
4-((Bicyclic heterocyclyl)-methyl and -hetero)-piperidines
JANSSEN PHARMACEUTICA NV11 citations73
US5629308AMay 13, 1997
Imidazo [1,2-A] (pyrrolo, thieno or furano) [2,3-D] azepine derivatives
JANSSEN PHARMACEUTICA NV7 citations72
US5272150ADec 21, 1993
Hydroxyalkylfuranyl derivatives
JANSSEN PHARMACEUTICA NV14 citations72
US5151424ASep 29, 1992
Pharmacologically active (Bicyclic heterocyclyl)methyl and -hetero) substituted hexahydro-1H-azepines and pyrrolidines
JANSSEN PHARMACEUTICA NV11 citations71
US5011842AApr 30, 1991
2-(heterocyclylalkyl)imidazopyridines for treating allergic diseases
JANSSEN PHARMACEUTICA NV4 citations62
US4897401AJan 30, 1990
N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives useful in treating allergic diseases
JANSSEN PHARMACEUTICA NV5 citations62
US5461050AOct 24, 1995
Imidazo[1,2-a](pyrrolo, thieno or furano) [3,2a-d]azepine derivatives, compositions and methods of use
JANSSEN PHARMACEUTICA NV6 citations61
US5071846ADec 10, 1991
Anti-hystaminic [(bicyclic heterocyclyl) methyl and --hetero] substituted hexahydro-1H-azepines and pyrrolidines
JANSSEN PHARMACEUTICA NV3 citations60