Inventor
GILLESPIE PAUL
US39 patents
⚠️ This page may combine multiple inventors who share the name “GILLESPIE PAUL”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
HOFFMANN LA ROCHE
22 patentsUS6803384B2Oct 12, 2004
Diaminopropionic acid derivatives
HOFFMANN LA ROCHE73 citations97
US7217728B2May 15, 2007
Diaminopropionic acid derivatives
HOFFMANN LA ROCHE40 citations96
US6331640B1Dec 18, 2001
Diaminopropionic acid derivatives
HOFFMANN LA ROCHE80 citations96
US6515124B2Feb 4, 2003
Dehydroamino acids
HOFFMANN LA ROCHE53 citations92
US7094896B2Aug 22, 2006
Diaminothiazoles having antiproliferative activity
HOFFMANN LA ROCHE17 citations90
US9296711B2Mar 29, 2016
Substituted isoxazole amide compounds as inhibitors of stearoyl-CoA desaturase 1 (SCD1)
HOFFMANN LA ROCHE9 citations84
US7504513B2Mar 17, 2009
Thiazolyl-benzimidazoles
HOFFMANN LA ROCHE13 citations83
US7728029B2Jun 1, 2010
Adamantyl-pyrazole carboxamides as inhibitors of 11β-hdroxysteroid dehydrogenase
HOFFMANN LA ROCHE8 citations82
US9290465B2Mar 22, 2016
Substituted isoxazole amine compounds as inhibitors of SCD1
HOFFMANN LA ROCHE9 citations80
US7138529B2Nov 21, 2006
Substituted 3-cyanothiophene acetamides as glucagon receptor antagonists
HOFFMANN LA ROCHE7 citations73
US7355049B2Apr 8, 2008
Biaryloxymethylarenecarboxylic acids as glycogen synthase activator
HOFFMANN LA ROCHE8 citations71
US6756374B2Jun 29, 2004
Diaminothiazoles having antiproliferative activity
HOFFMANN LA ROCHE6 citations71
US7652013B2Jan 26, 2010
Inhibitors of stearoyl-CoA desaturase
HOFFMANN LA ROCHE2 citations63
US7524870B2Apr 28, 2009
Biaryloxymethylarenecarboxylic acids as glycogen synthase activators
HOFFMANN LA ROCHE4 citations63
US7345058B2Mar 18, 2008
Pyrazoles
HOFFMANN LA ROCHE2 citations63
US7645773B2Jan 12, 2010
Thiazoles as inhibitors of 11β-hydroxysteroid dehydrogenase
HOFFMANN LA ROCHE6 citations62
US7491741B2Feb 17, 2009
Diaminopropionic acid derivatives
HOFFMANN LA ROCHE1 citations62
US7842825B2Nov 30, 2010
Biaryloxymethylarenecarboxylic acids as glycogen synthase activator
HOFFMANN LA ROCHE1 citations60
US7790711B2Sep 7, 2010
Inhibitors of 11β-Hydroxysteroid Dehydrogenase
HOFFMANN LA ROCHE0 citations51
US7105670B2Sep 12, 2006
Intermediates useful in the preparation of diaminothiazoles
HOFFMANN LA ROCHE0 citations50
US7700632B2Apr 20, 2010
Biaryloxymethylarenecarboxylic acids as glycogen synthase activator
HOFFMANN LA ROCHE0 citations49
US7622492B2Nov 24, 2009
Pyrazolones as inhibitors of 11β-hydroxysteroid dehydrogenase
HOFFMANN LA ROCHE0 citations38
CHEN LI
5 patentsUS8268870B2Sep 18, 2012
Aminotetrahydroindazoloacetic acids
CHEN LI2 citations62
US8124641B2Feb 28, 2012
Aminotetrahydroindazoloacetic acids
CHEN LI2 citations62
US8420675B2Apr 16, 2013
Aminotetrahydroindazoloacetic acids
CHEN LI0 citations51
US8138208B2Mar 20, 2012
Aminotetrahydroindazoloacetic acids
CHEN LI0 citations51
US8642629B2Feb 4, 2014
Naphthylacetic acids
CHEN LI0 citations41