P

Inventor

BLYTHIN DAVID J

US39 patents

Patents

39 patents
US5795894AAug 18, 1998

Piperazino derivatives as neurokinn antagonists

SCHERING CORP109 citations98
US5968929AOct 19, 1999

Piperazino derivatives as neurokinin antagonists

SCHERING CORP70 citations96
US5869488AFeb 9, 1999

Piperazino derivatives as neurokinin antagonists

SCHERING CORP78 citations96
US5798359AAug 25, 1998

Piperazino derivatives as neurokinin antagonists

SCHERING CORP56 citations95
US5719156AFeb 17, 1998

Piperazino derivatives as neurokinin antagonists

SCHERING CORP55 citations95
US6635630B2Oct 21, 2003

Selective neurokinin antagonists

SCHERING CORP41 citations92
US6436928B1Aug 20, 2002

Selective neurokinin antagonists

SCHERING CORP17 citations92
US5037826AAug 6, 1991

1-substituted naphthyridine and pyridopyrazine derivatives

SCHERING CORP36 citations92
US4680298AJul 14, 1987

Tricyclic anti-allergy and use as anti-inflammatory agents

SCHERING CORP27 citations92
US4897397AJan 30, 1990

Aryl-alkynoic, alkenoic or alkanoic compounds and compositions useful as antiallergy and anti-inflammatory agents

SCHERING CORP33 citations86
US7956189B2Jun 7, 2011

Maleate, tosylate, fumarate and oxalate salts of 5-(1-(S)-amino-2-hydroxyethyl)-N-[(2,4-difluorophenyl)-methy]-2-[8-methoxy-2-(triflouromethy)-5-quinoline]-4-oxazolecarboxamide and preparation process therefore

SCHERING CORP7 citations80
US6051575AApr 18, 2000

Piperazino derivatives as neurokinin antagonists

SCHERING CORP15 citations74
US5981520ANov 9, 1999

Piperazino derivatives as neurokinin antagonists

SCHERING CORP13 citations74
US5892039AApr 6, 1999

Piperazino derivatives as neurokinin antagonists

SCHERING CORP13 citations74
US5011860AApr 30, 1991

Aryl-substituted naphthyridine and pyridopyrazine derivatives and their use in treating hyperproliferative skin diseases

SCHERING CORP8 citations74
US4794116ADec 27, 1988

Anti-allergic esters, acetal ethers, thioethers and nitrogen substituted derivatives of bicyclic compounds

SCHERING CORP5 citations74
US4782067ANov 1, 1988

Anti-allergic composition containing zwitterionic bicyclic compounds

SCHERING CORP12 citations74
US4760073AJul 26, 1988

Aryl-substituted naphthyridine and pyridopyrazine derivatives, useful as anti-allergic agents

SCHERING CORP13 citations74
US4740511AApr 26, 1988

Method of treating hyperproliferative skin disease

SCHERING CORP9 citations74
US4684727AAug 4, 1987

Zwitterionic 1,8-naphthyridine and pyrazino[2,3-b]pyridine containing compounds useful as anti-allergic, anti-inflammatory and cycloprotective agents

SCHERING CORP7 citations74
US4652564AMar 24, 1987

Substituted spiro pyridine derivatives as anti-allergy and antiinflammatory agents

SCHERING CORP15 citations74
US4632923ADec 30, 1986

Substituted hetero spiro pyridine derivatives as anti-allergy and anti-inflammatory agents

SCHERING CORP13 citations74
US4297355AOct 27, 1981

(1H,3H,5H)-(1)-Benzopyrano-(2,3-d)-pyrimidine-4-one-2-thiones and their use as anti-allergy agents

SCHERING CORP7 citations74
US4272535AJun 9, 1981

2,4-[1H,3H,5H]-(1)-Benzopyrano-[2,3-d]-pyrimidinediones and their use as anti-allergy agents

SCHERING CORP19 citations74
US5929236AJul 27, 1999

2-substituted morpholine and thiomorpholine derivatives as GABA-B antagonists

SCHERING CORP13 citations73
US4902693AFeb 20, 1990

Anti-allergic esters, acetal ethers, thioethers and nitrogen substituted derivatives of bicyclic compounds

SCHERING CORP4 citations63
US4866061ASep 12, 1989

Aryl-substituted naphthyridine and pyridopyrazine derivatives

SCHERING CORP4 citations63
US4775524AOct 4, 1988

Method of treating hyperproliferative skin disease with substituted heterospiro pyridine derivatives

SCHERING CORP3 citations63
US4569936AFeb 11, 1986

Anti-inflammatory substituted 9H-8-oxo-pyrimido[2,1-f]purine-2,4-diones

SCHERING CORP2 citations63
US4775686AOct 4, 1988

Naphthyridine derivatives and method for treating allergic reactions

SCHERING CORP4 citations62
US4680297AJul 14, 1987

Tricyclic positive inotropic agents

SCHERING CORP6 citations62
US4996212AFeb 26, 1991

Antiinflammatory and anti-hyperproliferative compounds

SCHERING CORP2 citations57
US4859669AAug 22, 1989

Antiinflammatory and anti-hyperproliferative naphthyridin-4-ones

SCHERING CORP2 citations57
US5760034AJun 2, 1998

Heterocyclic substituted naphthyridinones and methods and compositions employing them

SCHERING CORP0 citations52
US5461057AOct 24, 1995

Hydro-ethano-indeno-pyridines

SCHERING CORP1 citations52
US5118683AJun 2, 1992

Esters of 4-hydroxy-1,3-benzenedimethanol and compositions and methods employing such compounds

SCHERING CORP1 citations52
US4916131AApr 10, 1990

Naphthyridine derivatives and method for treating allergic reactions

SCHERING CORP1 citations52
US5350755ASep 27, 1994

Compounds and methods for treating hyperproliferative skin disease

SCHERING CORP0 citations42
US5011845AApr 30, 1991

Cyclic diesters of 4-hydroxy-1,3-benzenedimethanol and compositions and methods employing such compounds

SCHERING CORP0 citations42