Inventor
BLYTHIN DAVID J
US39 patents
Patents
39 patentsUS5795894AAug 18, 1998
Piperazino derivatives as neurokinn antagonists
SCHERING CORP109 citations98
US5968929AOct 19, 1999
Piperazino derivatives as neurokinin antagonists
SCHERING CORP70 citations96
US5869488AFeb 9, 1999
Piperazino derivatives as neurokinin antagonists
SCHERING CORP78 citations96
US5798359AAug 25, 1998
Piperazino derivatives as neurokinin antagonists
SCHERING CORP56 citations95
US5719156AFeb 17, 1998
Piperazino derivatives as neurokinin antagonists
SCHERING CORP55 citations95
US6635630B2Oct 21, 2003
Selective neurokinin antagonists
SCHERING CORP41 citations92
US6436928B1Aug 20, 2002
Selective neurokinin antagonists
SCHERING CORP17 citations92
US5037826AAug 6, 1991
1-substituted naphthyridine and pyridopyrazine derivatives
SCHERING CORP36 citations92
US4680298AJul 14, 1987
Tricyclic anti-allergy and use as anti-inflammatory agents
SCHERING CORP27 citations92
US4897397AJan 30, 1990
Aryl-alkynoic, alkenoic or alkanoic compounds and compositions useful as antiallergy and anti-inflammatory agents
SCHERING CORP33 citations86
US7956189B2Jun 7, 2011
Maleate, tosylate, fumarate and oxalate salts of 5-(1-(S)-amino-2-hydroxyethyl)-N-[(2,4-difluorophenyl)-methy]-2-[8-methoxy-2-(triflouromethy)-5-quinoline]-4-oxazolecarboxamide and preparation process therefore
SCHERING CORP7 citations80
US6051575AApr 18, 2000
Piperazino derivatives as neurokinin antagonists
SCHERING CORP15 citations74
US5981520ANov 9, 1999
Piperazino derivatives as neurokinin antagonists
SCHERING CORP13 citations74
US5892039AApr 6, 1999
Piperazino derivatives as neurokinin antagonists
SCHERING CORP13 citations74
US5011860AApr 30, 1991
Aryl-substituted naphthyridine and pyridopyrazine derivatives and their use in treating hyperproliferative skin diseases
SCHERING CORP8 citations74
US4794116ADec 27, 1988
Anti-allergic esters, acetal ethers, thioethers and nitrogen substituted derivatives of bicyclic compounds
SCHERING CORP5 citations74
US4782067ANov 1, 1988
Anti-allergic composition containing zwitterionic bicyclic compounds
SCHERING CORP12 citations74
US4760073AJul 26, 1988
Aryl-substituted naphthyridine and pyridopyrazine derivatives, useful as anti-allergic agents
SCHERING CORP13 citations74
US4740511AApr 26, 1988
Method of treating hyperproliferative skin disease
SCHERING CORP9 citations74
US4684727AAug 4, 1987
Zwitterionic 1,8-naphthyridine and pyrazino[2,3-b]pyridine containing compounds useful as anti-allergic, anti-inflammatory and cycloprotective agents
SCHERING CORP7 citations74
US4652564AMar 24, 1987
Substituted spiro pyridine derivatives as anti-allergy and antiinflammatory agents
SCHERING CORP15 citations74
US4632923ADec 30, 1986
Substituted hetero spiro pyridine derivatives as anti-allergy and anti-inflammatory agents
SCHERING CORP13 citations74
US4297355AOct 27, 1981
(1H,3H,5H)-(1)-Benzopyrano-(2,3-d)-pyrimidine-4-one-2-thiones and their use as anti-allergy agents
SCHERING CORP7 citations74
US4272535AJun 9, 1981
2,4-[1H,3H,5H]-(1)-Benzopyrano-[2,3-d]-pyrimidinediones and their use as anti-allergy agents
SCHERING CORP19 citations74
US5929236AJul 27, 1999
2-substituted morpholine and thiomorpholine derivatives as GABA-B antagonists
SCHERING CORP13 citations73
US4902693AFeb 20, 1990
Anti-allergic esters, acetal ethers, thioethers and nitrogen substituted derivatives of bicyclic compounds
SCHERING CORP4 citations63
US4866061ASep 12, 1989
Aryl-substituted naphthyridine and pyridopyrazine derivatives
SCHERING CORP4 citations63
US4775524AOct 4, 1988
Method of treating hyperproliferative skin disease with substituted heterospiro pyridine derivatives
SCHERING CORP3 citations63
US4569936AFeb 11, 1986
Anti-inflammatory substituted 9H-8-oxo-pyrimido[2,1-f]purine-2,4-diones
SCHERING CORP2 citations63
US4775686AOct 4, 1988
Naphthyridine derivatives and method for treating allergic reactions
SCHERING CORP4 citations62
US4680297AJul 14, 1987
Tricyclic positive inotropic agents
SCHERING CORP6 citations62
US4996212AFeb 26, 1991
Antiinflammatory and anti-hyperproliferative compounds
SCHERING CORP2 citations57
US4859669AAug 22, 1989
Antiinflammatory and anti-hyperproliferative naphthyridin-4-ones
SCHERING CORP2 citations57
US5760034AJun 2, 1998
Heterocyclic substituted naphthyridinones and methods and compositions employing them
SCHERING CORP0 citations52
US5461057AOct 24, 1995
Hydro-ethano-indeno-pyridines
SCHERING CORP1 citations52
US5118683AJun 2, 1992
Esters of 4-hydroxy-1,3-benzenedimethanol and compositions and methods employing such compounds
SCHERING CORP1 citations52
US4916131AApr 10, 1990
Naphthyridine derivatives and method for treating allergic reactions
SCHERING CORP1 citations52
US5350755ASep 27, 1994
Compounds and methods for treating hyperproliferative skin disease
SCHERING CORP0 citations42
US5011845AApr 30, 1991
Cyclic diesters of 4-hydroxy-1,3-benzenedimethanol and compositions and methods employing such compounds
SCHERING CORP0 citations42