Inventor
KOLAKOWSKI GABRIELLE R
US58 patents
⚠️ This page may combine multiple inventors who share the name “KOLAKOWSKI GABRIELLE R”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
ARRAY BIOPHARMA INC
33 patentsUS9493476B2Nov 15, 2016
Macrocyclic compounds as trk kinase inhibitors
ARRAY BIOPHARMA INC46 citations98
US10112942B2Oct 30, 2018
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC29 citations94
US9902741B2Feb 27, 2018
Macrocyclic compounds as TRK kinase inhibitors
ARRAY BIOPHARMA INC22 citations94
US9840519B2Dec 12, 2017
Macrocyclic compounds as TRK kinase inhibitors
ARRAY BIOPHARMA INC21 citations94
US9750744B2Sep 5, 2017
Macrocyclic compounds as Trk kinase inhibitors
ARRAY BIOPHARMA INC21 citations94
US9718822B2Aug 1, 2017
Macrocyclic compounds as Trk kinase inhibitors
ARRAY BIOPHARMA INC22 citations94
US10174027B2Jan 8, 2019
Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC17 citations93
US10174028B2Jan 8, 2019
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC14 citations93
US10138243B2Nov 27, 2018
Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC14 citations92
US10137124B2Nov 27, 2018
Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC12 citations92
US10023570B2Jul 17, 2018
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC14 citations92
US10584124B2Mar 10, 2020
Crystalline forms
ARRAY BIOPHARMA INC12 citations86
US10953005B1Mar 23, 2021
Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC4 citations84
US10647730B2May 12, 2020
Macrocyclic compounds as TRK kinase inhibitors
ARRAY BIOPHARMA INC4 citations84
US10555944B2Feb 11, 2020
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC10 citations84
US10172851B2Jan 8, 2019
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC8 citations84
US10172845B2Jan 8, 2019
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC4 citations83
US10144734B2Dec 4, 2018
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC6 citations83
US10688100B2Jun 23, 2020
Macrocylic compounds as ROS1 kinase inhibitors
ARRAY BIOPHARMA INC3 citations73
US10323022B2Jun 18, 2019
Pyrrolidinyl urea, pyrrolidinyl thiourea and pyrrolidinyl guanidine compounds as TrkA kinase inhibitors
ARRAY BIOPHARMA INC2 citations73
US9878997B2Jan 30, 2018
Pyrrolidinyl urea, pyrrolidinyl thiourea and pyrrolidinyl guanidine compounds as TrkA kinase inhibitors
ARRAY BIOPHARMA INC4 citations73
US10881652B2Jan 5, 2021
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC2 citations72
US10441581B2Oct 15, 2019
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC2 citations72
US9896435B2Feb 20, 2018
N-pyrrolidinyl,N′-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
ARRAY BIOPHARMA INC3 citations72
US10966985B2Apr 6, 2021
Macrocyclic compounds as ROS1 kinase inhibitors
ARRAY BIOPHARMA INC0 citations63
US11998545B2Jun 4, 2024
Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC0 citations62
US11851434B2Dec 26, 2023
Substituted pyrazolo[1,5-A]pyrazine compounds as ret kinase inhibitors
ARRAY BIOPHARMA INC0 citations62
US11648243B2May 16, 2023
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC0 citations62
US11168090B2Nov 9, 2021
Substituted pyrazolo[1,5-a]pyrazines as RET kinase inhibitors
ARRAY BIOPHARMA INC0 citations62
US10889589B2Jan 12, 2021
Bicyclic urea, thiourea, guanidine and cyanoguanidine compounds useful for the treatment of pain
ARRAY BIOPHARMA INC0 citations62
US10351575B2Jul 16, 2019
Bicyclic urea, thiourea, guanidine and cyanoguanidine compounds useful for the treatment of pain
ARRAY BIOPHARMA INC1 citations62
US11524963B2Dec 13, 2022
Substituted pyrazolo[3,4-d]pyrimidines as RET kinase inhibitors
ARRAY BIOPHARMA INC0 citations60
US9546156B2Jan 17, 2017
N-bicyclic aryl,N'-pyrazolyl urea, thiourea, guanidine cyanoguanidine compounds as TrkA kinase inhibitors
ARRAY BIOPHARMA INC1 citations52
LOXO ONCOLOGY INC
8 patentsUS10907215B2Feb 2, 2021
Point mutations in TRK inhibitor-resistant cancer and methods relating to the same
LOXO ONCOLOGY INC3 citations72
US10724102B2Jul 28, 2020
Point mutations in TRK inhibitor-resistant cancer and methods relating to the same
LOXO ONCOLOGY INC3 citations72
US10655186B2May 19, 2020
Point mutations in TRK inhibitor-resistant cancer and methods relating to the same
LOXO ONCOLOGY INC3 citations72
US10378068B2Aug 13, 2019
Point mutations in TRK inhibitor-resistant cancer and methods relating to the same
LOXO ONCOLOGY INC3 citations72
US10370727B2Aug 6, 2019
Point mutations in TRK inhibitor-resistant cancer and methods relating to the same
LOXO ONCOLOGY INC3 citations72
US10745419B2Aug 18, 2020
Process for the preparation of 6-(2-hydroxy-2-methylpropoxy)-4-(6-(6-((6-methoxypyridin-3-yl)methyl)-3,6-diazabicyclo[3.1.1]heptan-3-yl)pyridin-3-yl)pyrazolo[1,5-a]pyridine-3-carbonitrile
LOXO ONCOLOGY INC2 citations70
US11807651B2Nov 7, 2023
Process for the preparation of 6-(2-hydroxy-2-methylpropoxy)-4-(6-(6-((6-methoxypyridin-3-yl)methyl)-3,6-diazabicyclo[3.1.1]heptan-3-yl)pyridin-3-yl)pyrazolo[1,5-a]pyridine-3-carbonitrile
LOXO ONCOLOGY INC0 citations59
US11098064B2Aug 24, 2021
Process for the preparation of 6-(2-hydroxy-2-methylpropoxy)-4-(6-(6-((6-methoxypyridin-3-yl)methyl)-3,6-diazabicyclo[3.1.1]heptan-3-yl)pyridin-3-yl)pyrazolo[1,5-a]pyridine-3-carbontrile
LOXO ONCOLOGY INC1 citations59
LILLY CO ELI
4 patentsUS11964968B2Apr 23, 2024
Compounds useful for inhibiting RET kinase
LILLY CO ELI0 citations57
US11613533B2Mar 28, 2023
Compounds useful for inhibiting RET kinase
LILLY CO ELI0 citations57
US11970485B2Apr 30, 2024
RET kinase inhibitors
LILLY CO ELI0 citations56
US11697647B2Jul 11, 2023
RET kinase inhibitors
LILLY CO ELI1 citations56
PETRA PHARMA CORP
2 patentsUS11873295B2Jan 16, 2024
Allosteric chromenone inhibitors of phosphoinositide 3-kinase (PI3K) for the treatment of disease
PETRA PHARMA CORP3 citations65
US11649227B2May 16, 2023
Allosteric chromenone inhibitors of phosphoinositide 3-kinase (PI3K) for the treatment of disease
PETRA PHARMA CORP1 citations53
ANDREWS STEVEN WADE
1 patentALLEN SHELLEY
1 patentBLAKE JAMES F
1 patentShowing the top 50 of 58 patents by PatentIndex Score.