Inventor
VAN DAELE GEORGES H P
BE33 patents
Patents
33 patentsUS5374637ADec 20, 1994
N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
JANSSEN PHARMACEUTICA NV86 citations97
US5576448ANov 19, 1996
N-(3-hydroxy-4-piperidinyl) (dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
JANSSEN PHARMACEUTICA NV24 citations96
US4179569ADec 18, 1979
N-(4-piperidinyl)-N-phenylamides
JANSSEN PHARMACEUTICA NV34 citations92
US4990521AFeb 5, 1991
4-(aroylamino)piperidine-butanimide derivatives
JANSSEN PHARMACEUTICA NV47 citations91
US5041454AAug 20, 1991
Novel substituted N-(1-alkyl-3-hydroxy-4-piperidinyl)benzamides
JANSSEN PHARMACEUTICA NV23 citations90
US4975439ADec 4, 1990
Novel substituted N-(1-alkyl-3-hydroxy-4-piperidinyl)benzamides
JANSSEN PHARMACEUTICA NV24 citations90
US4968684ANov 6, 1990
Method of improving sleep
JANSSEN PHARMACEUTICA NV20 citations81
US5130312AJul 14, 1992
Substituted N-(3-hydroxy-4-piperidinyl)benzamides
JANSSEN PHARMACEUTICA NV21 citations79
US5610157AMar 11, 1997
N-(3-hydroxy-4-piperidinyl) (dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzo-dioxin) carboxamide derivatives
JANSSEN PHARMACEUTICA NV4 citations73
US5026853AJun 25, 1991
4-substituted-2(or 3)aminocarbonyl-1-piperazineacetamide
JANSSEN PHARMACEUTICA NV18 citations72
US4880808ANov 14, 1989
N-aryl-piperazinealkanamides useful for improving sleep
JANSSEN PHARMACEUTICA NV15 citations72
US5948794ASep 7, 1999
Enterokinetic benzamide
JANSSEN PHARMACEUTICA NV7 citations71
US5854260ADec 29, 1998
Enterokinetic benzamide
JANSSEN PHARMACEUTICA NV5 citations71
US4906643AMar 6, 1990
Substituted N-(3-hydroxy-4-piperidinyl)benzamides as gastrointestinal agents
JANSSEN PHARMACEUTICA NV13 citations71
US5498618AMar 12, 1996
4-amino-N-(4-methyl-4-piperidinyl)-2-methoxybenzamides for treating smooth muscle contraction disorders
JANSSEN PHARMACEUTICA NV5 citations66
US5739134AApr 14, 1998
N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2h-benzopyran, dihydrobenzodioxin, benzodioxole, dihydrobenzodioxepin, or tetrahydrobenzoxepin)carboxamide derivatives
JANSSEN PHARMACEUTICA NV4 citations64
US5616738AApr 1, 1997
N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2-H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
JANSSEN PHARMACEUTICA NV1 citations62
US5616583AApr 1, 1997
N- (3-hydroxy-4-piperidinyl) (benzodioxolane, benzodioxane or benzodioxepane) carboxamide derivatives
JANSSEN PHARMACEUTICA NV2 citations62
US5602129AFeb 11, 1997
N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
JANSSEN PHARMACEUTICA NV1 citations62
US5565582AOct 15, 1996
N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
JANSSEN PHARMACEUTICA NV1 citations62
US5554772ASep 10, 1996
N-(3-hydroxy-4-piperidinyl) dihydrobenzofuran, (dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
JANSSEN PHARMACEUTICA NV1 citations62
US5536733AJul 16, 1996
N-(3-hydroxy-4-piperidinyl) (dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
JANSSEN PHARMACEUTICA NV2 citations62
US5521314AMay 28, 1996
N-(3-hydroxy)-4-piperidinyl) (Dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
JANSSEN PHARMACEUTICA NV1 citations62
US5480997AJan 2, 1996
Pyridine-substituted benzenemethanamine derivatives
JANSSEN PHARMACEUTICA NV1 citations61
US5480912AJan 2, 1996
Method of treating HIV-1 with α-substituted benzenemethanamine derivatives
JANSSEN PHARMACEUTICA NV2 citations59
US6310077B1Oct 30, 2001
Enterokinetic benzamide
JANSSEN PHARMACEUTICA NV1 citations58
US5552553ASep 3, 1996
N-(3-hydroxy-4-piperidinyl) (dihydrobenzofuran, dihydro-2H-benzopyran or dehydrobenzodioxin) carboxamide derivatives
JANSSEN PHARMACEUTICA NV1 citations54
US5604230AFeb 18, 1997
Heterocycle-substituted benzenemethanamine derivatives
JANSSEN PHARMACEUTICA NV0 citations50
US5587387ADec 24, 1996
Heterocycle-substituted benzenemethanamine derivatives
JANSSEN PHARMACEUTICA NV0 citations50
US5552430ASep 3, 1996
Heterocycle-substituted benzenemethanamine derivatives
JANSSEN PHARMACEUTICA NV0 citations50
US5550135AAug 27, 1996
Heterocycle-substituted benzenemethanamine derivatives
JANSSEN PHARMACEUTICA NV0 citations50
US5541215AJul 30, 1996
Heterocycle-substituted benzenemethanamine derivatives
JANSSEN PHARMACEUTICA NV0 citations50
US5407961AApr 18, 1995
α-substituted benzenemethanamine derivatives and pharmaceutical use
JANSSEN PHARMACEUTICA NV1 citations49