Inventor
JAESCHKE GEORG
CH84 patents
⚠️ This page may combine multiple inventors who share the name “JAESCHKE GEORG”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
HOFFMANN LA ROCHE
43 patentsUS7332510B2Feb 19, 2008
Imidazole derivatives
HOFFMANN LA ROCHE15 citations92
US6451819B2Sep 17, 2002
Heterocyclic compounds useful as NMDA receptor selective subtype blockers
HOFFMANN LA ROCHE43 citations92
US6265426B1Jul 24, 2001
Triazole derivatives
HOFFMANN LA ROCHE30 citations92
US10562903B2Feb 18, 2020
Bridged piperidine derivatives
HOFFMANN LA ROCHE12 citations86
US12209091B2Jan 28, 2025
Isoindolinone derivatives as selective allosteric inhibitors of Egfr mutant cancers
HOFFMANN LA ROCHE7 citations85
US8039490B2Oct 18, 2011
Benzoyl-piperidine derivatives as dual modulators of the 5-HT2A and D3 receptors
HOFFMANN LA ROCHE7 citations84
US7153874B2Dec 26, 2006
Imidazole derivatives
HOFFMANN LA ROCHE15 citations84
US7091222B2Aug 15, 2006
Imidazole derivatives
HOFFMANN LA ROCHE13 citations84
US6339093B1Jan 15, 2002
Isoquinoline derivatives
HOFFMANN LA ROCHE17 citations84
US8618296B2Dec 31, 2013
Arylethynyl derivatives
HOFFMANN LA ROCHE4 citations74
US8513273B2Aug 20, 2013
Arylethynyl derivatives
HOFFMANN LA ROCHE4 citations74
US6610723B2Aug 26, 2003
Imidazole derivatives
HOFFMANN LA ROCHE10 citations74
US6432985B2Aug 13, 2002
Neuroprotective substituted piperidine compounds with activity as NMDA NR2B subtype selective antagonists
HOFFMANN LA ROCHE13 citations74
US9695128B2Jul 4, 2017
Ethynyl derivatives
HOFFMANN LA ROCHE4 citations73
US9682959B2Jun 20, 2017
Ethynyl derivatives
HOFFMANN LA ROCHE2 citations73
US9199971B2Dec 1, 2015
Arylethynyl pyrimidines
HOFFMANN LA ROCHE5 citations73
US8969338B2Mar 3, 2015
Ethynyl derivatives
HOFFMANN LA ROCHE4 citations73
US8716316B2May 6, 2014
Positive allosteric modulators (PAM)
HOFFMANN LA ROCHE4 citations73
US7858630B2Dec 28, 2010
D3 and 5-HT2A receptor modulators
HOFFMANN LA ROCHE7 citations73
US7414060B2Aug 19, 2008
Pyridine-2-carboxyamide derivatives
HOFFMANN LA ROCHE8 citations73
US7241760B2Jul 10, 2007
Heteroaryl-substituted imidazole derivatives
HOFFMANN LA ROCHE7 citations73
US6440995B1Aug 27, 2002
Quinolin-4-yl derivatives
HOFFMANN LA ROCHE10 citations73
US6310213B1Oct 30, 2001
Ethanesulfonyl-piperidine derivatives
HOFFMANN LA ROCHE11 citations73
US12344613B2Jul 1, 2025
EGFR inhibitor for the treatment of cancer
HOFFMANN LA ROCHE3 citations72
US11708354B2Jul 25, 2023
2-benzopyrazinyl-n-heteroaryl-2-phenyl-acetamide compounds
HOFFMANN LA ROCHE3 citations72
US11117890B2Sep 14, 2021
Substituted isoindole allosteric EGFR inhibitors
HOFFMANN LA ROCHE3 citations72
US10882848B2Jan 5, 2021
2-benzopyrazinyl-n-heteroaryl-2-phenyl-acetamide compounds
HOFFMANN LA ROCHE3 citations72
US10189848B2Jan 29, 2019
Ethynyl derivatives
HOFFMANN LA ROCHE4 citations72
US10065956B2Sep 4, 2018
Ethynyl derivatives
HOFFMANN LA ROCHE4 citations72
US9725416B2Aug 8, 2017
Ethynyl derivatives
HOFFMANN LA ROCHE4 citations72
US9359301B2Jun 7, 2016
Ethynyl derivatives
HOFFMANN LA ROCHE2 citations63
US9328090B2May 3, 2016
Arylethynyl derivatives
HOFFMANN LA ROCHE2 citations63
US9315498B2Apr 19, 2016
Arlethynyl derivatives
HOFFMANN LA ROCHE2 citations63
US9221802B2Dec 29, 2015
Arylethynyl derivatives
HOFFMANN LA ROCHE2 citations63
US9212171B2Dec 15, 2015
Ethynyl compounds
HOFFMANN LA ROCHE3 citations63
US7005432B2Feb 28, 2006
Substituted imidazol-pyridazine derivatives
HOFFMANN LA ROCHE3 citations63
US6683097B2Jan 27, 2004
Imidazole derivatives
HOFFMANN LA ROCHE2 citations63
US12195413B2Jan 14, 2025
Ethynyl derivatives
HOFFMANN LA ROCHE0 citations62
US12145940B2Nov 19, 2024
Ethynyl derivatives
HOFFMANN LA ROCHE0 citations62
US12006323B2Jun 11, 2024
Ethynyl derivatives
HOFFMANN LA ROCHE0 citations62
US11242349B2Feb 8, 2022
Ethynyl derivatives
HOFFMANN LA ROCHE1 citations62
US11059766B2Jul 13, 2021
Ethynyl derivatives
HOFFMANN LA ROCHE0 citations62
US11034699B2Jun 15, 2021
Ethynyl derivatives
HOFFMANN LA ROCHE0 citations62
C4 THERAPEUTICS INC
3 patentsUS12371442B2Jul 29, 2025
Isoindolinone and indazole compounds for the degradation of EGFR
C4 THERAPEUTICS INC1 citations74
US11673902B2Jun 13, 2023
Isoindolinone and indazole compounds for the degradation of EGFR
C4 THERAPEUTICS INC3 citations72
US12486290B2Dec 2, 2025
Isoindolinone and indazole compounds for the degradation of EGFR
C4 THERAPEUTICS INC0 citations62
JAESCHKE GEORG
3 patentsGREEN LUKE
1 patentShowing the top 50 of 84 patents by PatentIndex Score.