Inventor

NISHINO YUKISHIGE

DE28 patents

Patents

28 patents

US5569652AOct 29, 1996

Dihydrospirorenone as an antiandrogen

SCHERING AG80 citations96

US5807899ASep 15, 1998

Triphenylethylenes, process for their production, pharmaceutical preparations that contain these triphenylethylenes as well as their use for the production of pharmaceutical agents

SCHERING AG56 citations94

US4916144AApr 10, 1990

N-substituted imidazoles as aromatase inhibitors

SCHERING AG30 citations92

US6495607B2Dec 17, 2002

Benzocycloheptenes, process for their production, pharmaceutical preparations that contain the latter as well as their use for the production of pharmaceutical agents

SCHERING AG14 citations83

US6288051B1Sep 11, 2001

7 α-(5-methylaminopentyl)-estratrienes, process for their production, pharmaceutical preparations that contain these 7 α(5-methylaminopentyl)-estratrienes as well as their use for the production of pharmaceutical agents

SCHERING AG17 citations82

US5986115ANov 16, 1999

7α-(ξ-aminoalkyl)-estratrienes, process for their production, pharmaceutical preparations which contain these 7α-(ξ-aminoalkyl)-estratrienes as well as their use for the production of pharmaceutical agents

SCHERING AG16 citations82

US5280035AJan 18, 1994

Cycloalkylene azoles and their use as aromatase inhibitors

SCHERING AG5 citations74

US5045558ASep 3, 1991

N-substituted imidazoles and their use in pharmaceutical agents

SCHERING AG7 citations74

US4925834AMay 15, 1990

3-methylene-4-androsten-17-ones, process for their production and pharmaceutical preparations containing them

SCHERING AG8 citations74

US4591585AMay 27, 1986

1-alkyl-androsta-1,4-diene-3,17-diones their production and pharmaceutical preparations containing same

SCHERING AG9 citations74

US6271403B1Aug 7, 2001

7α-(xi-aminoalkyl)-estratrienes, process for their production, pharmaceutical preparations which contain these 7α-(xi-aminoalkyl-estratrienes as well as their use for the production of pharmaceutical agents

SCHERING AG7 citations73

US5866560AFeb 2, 1999

7α-(ξ-aminoalkyl)-estratrienes, process for their production, pharmaceutical preparations which contain these 7α-(ξ-aminoalkyl)-estratrienes as well as their use for the production of pharmaceutical agents

SCHERING AG14 citations73

US3960841AJun 1, 1976

11β-HALOGEN-7α-SUBSTITUTED ESTRATRIENES, PROCESS FOR THE PRODUCTION OF PHARMACEUTICAL PREPARATIONS THAT CONTAIN THESE 11β-HALOGEN-7α-SUBSTITUTED ESTRATRIENES AS WELL AS THEIR USE FOR THE PRODUCTION OF PHARMACEUTICAL AGENTS

SCHERING AG8 citations72

US4011314AMar 8, 1977

7-hydroxyestradiols

SCHERING AG10 citations72

US5502046AMar 26, 1996

11β-substituted 14,17-ethanoestratrienes, process for their production and their use as pharmaceutical agents

SCHERING AG8 citations70

US5145847ASep 8, 1992

14,17α-etheno- and -ethanoestratrienes, processes for the preparation of these compounds, as well as their use for the production of medicinal agents

SCHERING AG5 citations63

US6878750B2Apr 12, 2005

Benzocycloheptenes, process for their production, pharmaceutical preparations that contain the latter as well as their use for the production of pharmaceutical agents

SCHERING AG4 citations62

US5344834ASep 6, 1994

Functionalized vinyl azoles and methods of use

SCHERING AG2 citations60

US5236912AAug 17, 1993

Antiandrogenic [3,2-c]pyrazole and [3,2-d]triazole steroids

SCHERING AG5 citations60

US4178381ADec 11, 1979

C-homoestratrienes

SCHERING AG2 citations60

US5411982AMay 2, 1995

Cycloalkylene azoles, and their use as aromatase inhibitors

SCHERING AG0 citations52

US5135937AAug 4, 1992

Cycloalkylene azoles and pharmaceutical preparations obtained therefrom

SCHERING AG0 citations52

US4871725AOct 3, 1989

1-methyl-15α-(1-oxyalkyl)androsta-1,4-diene-3,17-diones, processes for their production, and pharmaceutical preparations containing them

SCHERING AG0 citations52

US7145015B2Dec 5, 2006

Benzocycloheptenes, process for their production, pharmaceutical preparations that contain that latter as well as their use for the production of pharmaceutical agents

SCHERING AG0 citations51

US5389624AFeb 14, 1995

Antiandrogenic [3,2-c]pyrazole and [3,2-d]triazole steroids

SCHERING AG0 citations50

NISHINO YUKISHIGE

Patents

Dihydrospirorenone as an antiandrogen

Triphenylethylenes, process for their production, pharmaceutical preparations that contain these triphenylethylenes as well as their use for the production of pharmaceutical agents

N-substituted imidazoles as aromatase inhibitors

Benzocycloheptenes, process for their production, pharmaceutical preparations that contain the latter as well as their use for the production of pharmaceutical agents

7 α-(5-methylaminopentyl)-estratrienes, process for their production, pharmaceutical preparations that contain these 7 α(5-methylaminopentyl)-estratrienes as well as their use for the production of pharmaceutical agents

7α-(ξ-aminoalkyl)-estratrienes, process for their production, pharmaceutical preparations which contain these 7α-(ξ-aminoalkyl)-estratrienes as well as their use for the production of pharmaceutical agents

Cycloalkylene azoles and their use as aromatase inhibitors

N-substituted imidazoles and their use in pharmaceutical agents

3-methylene-4-androsten-17-ones, process for their production and pharmaceutical preparations containing them

1-alkyl-androsta-1,4-diene-3,17-diones their production and pharmaceutical preparations containing same

7α-(xi-aminoalkyl)-estratrienes, process for their production, pharmaceutical preparations which contain these 7α-(xi-aminoalkyl-estratrienes as well as their use for the production of pharmaceutical agents

7α-(ξ-aminoalkyl)-estratrienes, process for their production, pharmaceutical preparations which contain these 7α-(ξ-aminoalkyl)-estratrienes as well as their use for the production of pharmaceutical agents

3,17,18-Trihydroxy-1,3,5(10)-estratrienes

1,3-Oxygenated 8α-estratrienes

1,3-Oxygenated-8α-estratrienes

11β-HALOGEN-7α-SUBSTITUTED ESTRATRIENES, PROCESS FOR THE PRODUCTION OF PHARMACEUTICAL PREPARATIONS THAT CONTAIN THESE 11β-HALOGEN-7α-SUBSTITUTED ESTRATRIENES AS WELL AS THEIR USE FOR THE PRODUCTION OF PHARMACEUTICAL AGENTS

7-hydroxyestradiols

11β-substituted 14,17-ethanoestratrienes, process for their production and their use as pharmaceutical agents

14,17α-etheno- and -ethanoestratrienes, processes for the preparation of these compounds, as well as their use for the production of medicinal agents

Benzocycloheptenes, process for their production, pharmaceutical preparations that contain the latter as well as their use for the production of pharmaceutical agents

Functionalized vinyl azoles and methods of use

Antiandrogenic [3,2-c]pyrazole and [3,2-d]triazole steroids

C-homoestratrienes

Cycloalkylene azoles, and their use as aromatase inhibitors

Cycloalkylene azoles and pharmaceutical preparations obtained therefrom

1-methyl-15α-(1-oxyalkyl)androsta-1,4-diene-3,17-diones, processes for their production, and pharmaceutical preparations containing them

Benzocycloheptenes, process for their production, pharmaceutical preparations that contain that latter as well as their use for the production of pharmaceutical agents

Antiandrogenic [3,2-c]pyrazole and [3,2-d]triazole steroids