Inventor
EPSTEIN JOSEPH W
US32 patents
⚠️ This page may combine multiple inventors who share the name “EPSTEIN JOSEPH W”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
AMERICAN CYANAMID CO
26 patentsUS4131611ADec 26, 1978
Azabicyclohexanes
AMERICAN CYANAMID CO70 citations94
US4847256AJul 11, 1989
4,5-dihydro and 4,5,6,7-tetrahydropyrazolo(1,5-A)-pyrimidines
AMERICAN CYANAMID CO34 citations92
US4435419AMar 6, 1984
Method of treating depression using azabicyclohexanes
AMERICAN CYANAMID CO94 citations92
US5594027AJan 14, 1997
Aminocycloalkanobenzodioxoles as beta-3 selective adrenergic agents
AMERICAN CYANAMID CO21 citations91
US5510376AApr 23, 1996
Aminocycloalkanobenzodioxoles as beta-3 selective adrenergic agents
AMERICAN CYANAMID CO24 citations91
US4231935ANov 4, 1980
1-Phenyl-3-azabicyclo[3.1.0]hexanes
AMERICAN CYANAMID CO50 citations91
US4196120AApr 1, 1980
Azabicyclohexanes, method of use and preparation of the same
AMERICAN CYANAMID CO44 citations91
US5482971AJan 9, 1996
Beta3 -adrenergic agents and their use in pharmaceutical compositions
AMERICAN CYANAMID CO24 citations88
US4904658AFeb 27, 1990
Substituted-6H,8H-pyrimido-[1,2,3-cd]purine-8,10-(9H)-diones and substituted-6H,10H-pyrimido[1,2-cd]purin-10-ones
AMERICAN CYANAMID CO19 citations82
US5480908AJan 2, 1996
β3 -adrenergic agents benzodioxole dicarboxylates and their use in pharmaceutical compositions
AMERICAN CYANAMID CO16 citations81
US4544665AOct 1, 1985
1-Aryl-3-azabicyclo[3.2.0]heptanes
AMERICAN CYANAMID CO22 citations81
US5219857AJun 15, 1993
Method of treating cognitive and related neural behavioral problems
AMERICAN CYANAMID CO15 citations73
US5126340AJun 30, 1992
4-[(substituted)alkylcarbonyl]-4,5-dihydro and -4,5,6,7-tetrahydro-7-[(substituted)-phenyl]pyrazolo[1,5-a]pyrimidine-3-carbonitriles
AMERICAN CYANAMID CO13 citations73
US5084457AJan 28, 1992
Benzoylaminoquinazolinones
AMERICAN CYANAMID CO14 citations73
US4963553AOct 16, 1990
4-[(substituted) alkylcarbonyl]-4,5-dihydro- and -4,5,6,7-tetrahydro-7-[(substituted)phenyl]pyrazolo[1,5-a]pyrimidines
AMERICAN CYANAMID CO14 citations73
US4168269ASep 18, 1979
Substituted thieno-benzodiazepines
AMERICAN CYANAMID CO9 citations73
US4977189ADec 11, 1990
Substituted guanidinedicarbonyl derivatives
AMERICAN CYANAMID CO18 citations72
US4529736AJul 16, 1985
3a-(Substituted phenyl)-2,3,3a,4,7,7a-hexahydro[or 3a-(substituted-phenyl)octahydro]-4,7-alkano-1H-isoindoles for treating depression in warm-blooded animals
AMERICAN CYANAMID CO15 citations72
US4431661AFeb 14, 1984
5-Aryl-3-azabicyclo[3.2.0]heptan-6-one acetals, and analgesic use therefor
AMERICAN CYANAMID CO16 citations72
US5013737AMay 7, 1991
2,4,8-Trisubstituted-3H,6H-1,4,5A,8A-tetraazaacenaphtylene-3,5-(4H)-diones and 2,4-8-trisubstituted-4,5-dihydro-5-thioxo-3H,6H-1,4,5A,8A-tetrazaacenaphthylen-3-ones
AMERICAN CYANAMID CO2 citations62
US4916137AApr 10, 1990
5-(Substituted-amino)-8-(phenyl or substituted-phenyl)-3H,6H-1,4,5A,8A-tetraazaacenaphthylen-3-ones and treatment of neural behavior disorders
AMERICAN CYANAMID CO5 citations62
US4888345ADec 19, 1989
4,8-disubstituted-1,2-dihydro and 1,2,3,4-tetrahydroimidazo-[1,5-a] pyrimidines
AMERICAN CYANAMID CO2 citations62
US5606069AFeb 25, 1997
β3 -adrenergic agents, benzodioxole dicarboxylates and their use in pharmaceutical compositions
AMERICAN CYANAMID CO4 citations61
US4963552AOct 16, 1990
1-substitute-1,2-dihydro-4-((substituted)phenyl)imidazo-[1,5-a]pyrimidine-8-carbonitriles
AMERICAN CYANAMID CO2 citations60
US5001157AMar 19, 1991
Substituted N-[[2-(aminocarbonyl)phenylamino]thioxomethyl]benzamides
AMERICAN CYANAMID CO0 citations51
US5932585AAug 3, 1999
Method of treating or inhibiting neutropenia
AMERICAN CYANAMID CO0 citations35
NEUROVANCE INC
3 patentsUS9737506B2Aug 22, 2017
1-aryl-3-azabicyclo[3.1.0]hexanes: preparation and use to treat neuropsychiatric disorders
NEUROVANCE INC5 citations82
US9205074B2Dec 8, 2015
1-aryl-3-azabicyclo[3.1.0]hexanes: preparation and use to treat neuropsychiatric disorders
NEUROVANCE INC9 citations82
US8877798B2Nov 4, 2014
1-aryl-3-azabicyclo[3.1.0]hexanes: preparation and use to treat neuropsychiatric disorders
NEUROVANCE INC11 citations82