Inventor

SAARI WALFRED S

52 patents

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SAARI WALFRED S

MERCK & CO INC

Inhibitors of HIV reverse transcriptase

Inhibitors of HIV reverse transcriptase

Bone acting agents

Acyloxymethyl esters of bisphosphonic acids as bone resorption inhibitors

Inhibitors of farnesyl-protein transferase

Gastrin releasing peptide antagonist

N-alkyl(and cycloalkyl)oxamic acid and derivatives as inhibitors of glycolic acid oxidase

Gastrin releasing peptide antagonist

Piperazinylpyrazines

Carbamates of 4-hydroxyanisole as prodrugs for chemotherapy of melanoma

Tetrahydro-1H-1,4-diazepino(1,7-a)benzimidazoles useful as analgesic agents

6-chloro-2-(1-piperazinyl)pyrazine

Piperazinylpyrazines

Piperazinylpyridines

Antihypertensive amino acid esters

Halogenated pyrimidine nucleosides and their derivatives

Dinitrobenzenesulfonamides

α-nitroalkylnitrobenzenesulfonamides

Amides and esters of 2-(N-(hydroxypiperidinoalkyl) and (hydroxypyrrolidinoalkyl)-aminosulfonyl)-6-nitrobenzoic acids useful as adjuncts to radiation therapy

Amides and esters of 2-[N-(morpholinoalkyl)aminosulfonyl]-6-nitrobenzoic acids and compositions useful as adjuncts to radiation therapy

4-[2-Pyridinylthio(oxy or amino)methyl]-1H-imidazoles and derivatives

Treating sedation with 1-(3-substituted-2-pyridinyl) piperazines

Use of piperazinyl-imidazo[1,2-a]pyrazines in sedation

3-(1-Piperazinyl)-pyrido[2,3-b]pyrazines

Amino acid esters

(6aα,10aα,11aα)-2-(2-Pyridinyl)-1,3,4,6,6a,7,8,9,10,10a,11,11a-dodecahydro-2H-pyrazino]1,2-b]isoquinoline and derivatives

2-(4-Aminopiperidino)pyrazines

2-{[4-(6-Substituted-2-pyrazinyl)-1-piperazinyl]alkyl}-5-substituted-1,2,4-triazolo[4,3-a]pyridin-3(2H)-one analgesic agents

Esterification process

Gastrin releasing peptide antagonist

Derivatives of 2-(substituted sulfamyl)-6-nitrobenzoic acids and pharmaceutical compositions

Esters of 2-(substituted sulfamyl)-6-nitro-benzoic acid and pharmaceutical compositions

2-(substituted sulfamyl)-6-nitrobenzoic acid amides and pharmaceutical compositions

2-[2-Pyridinyloxy(thio or amino)methyl]-1H-imidazoles and derivatives

8-[2-Imidazolylmethyloxy(thio, or amino)]-imidazo[1,2-a]pyrazines and derivatives for treating hypertension

1-(3-Halo-2-pyridinyl) piperazine

Esters of α-methyl-3,4-OR-phenylalanines

Novel N-carboxy-alpha-amino acid anhydrides

6-(1-Piperazinyl)quinoxaline

Amino acid esters

3-(2,5-Dihydroxyphenyl)-alanine as a cardiac stimulant

N-substituted-3-nitro-4-(ureidooxymethyl)-benzenesulfonamides as radiation enhancers

Derivatives of 3-nitropyridines useful as adjuncts to radiation therapy

2-(substituted sulfamyl) derivatives of 4-nitrobenzamide as radiation sensitizers

Derivatives of 2-(substituted sulfamyl)-6-nitrobenzoic acids, useful as adjuncts to radiation therapy

Substituted 3-nitrobenzenesulfonamides useful as adjuncts in radiation therapy

Novel nitropyrazinyl- and nitropyridinyl- substituted piperazin-3-one and hexahydro-1H-1,4-diazepin-5-one compounds useful as adjuncts to radiation therapy

Amino acid esters

Process for preparing novel N-carboxyl-α-amino acid anhydrides

MERCK SHARP & DOHME

Fused tricyclic compounds, pharmaceutical compositions containing them and their use in therapy