Inventor
RAEYMAEKERS ALFONS H M
BE40 patents
⚠️ This page may combine multiple inventors who share the name “RAEYMAEKERS ALFONS H M”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
JANSSEN PHARMACEUTICA NV
38 patentsUS5521187AMay 28, 1996
1,3-Dihydro-2H-imidazo[4,5-B]quinolin-2-one derivatives
JANSSEN PHARMACEUTICA NV41 citations95
US5037829AAug 6, 1991
(1H-azol-1-ylmethyl) substituted quinazoline derivatives
JANSSEN PHARMACEUTICA NV57 citations95
US4859684AAug 22, 1989
(1H-imidazol-1-ylmethyl) substituted benzimidazole derivatives and use thereof in treating androgen dependent disorders
JANSSEN PHARMACEUTICA NV65 citations95
US5491161AFeb 13, 1996
Pyrroloimidazolyl and imidazopyridinyl substituted 1H-benzimidazole derivatives
JANSSEN PHARMACEUTICA NV24 citations92
US5151421ASep 29, 1992
(1h-azol-1-ylmethyl) substituted quinoxaline derivatives
JANSSEN PHARMACEUTICA NV29 citations92
US5028606AJul 2, 1991
(1H-azol-1-ylmethyl)substituted quinoxaline derivatives
JANSSEN PHARMACEUTICA NV44 citations92
US5157046AOct 20, 1992
Method of treating epithelial disorders
JANSSEN PHARMACEUTICA NV30 citations91
US4631278ADec 23, 1986
Anti-protozoal α-aryl-4-(4,5-dihydro-3,5-dioxo-1,2,4-triazin-2(3H)-yl)-benzeneacetonitrile derivatives, pharmaceutical compositions, and method of use therefor
JANSSEN PHARMACEUTICA NV31 citations91
US4943574AJul 24, 1990
(1H-azol-1-ylmethyl) substituted benzotriazole derivatives and pharmaceutical compositions containing them
JANSSEN PHARMACEUTICA NV23 citations89
US4243806AJan 6, 1981
5-[4-(Diarylmethyl)-1-piperazinylalkyl]benzimidazole derivatives
JANSSEN PHARMACEUTICA NV31 citations89
US5516908AMay 14, 1996
1,3-dihydro-2H-imidazo-[4,5-β]quinolin-2-one derivatives and intermediates
JANSSEN PHARMACEUTICA NV17 citations81
US5500435AMar 19, 1996
Method of treating epithelial disorders
JANSSEN PHARMACEUTICA NV15 citations81
US5342957AAug 30, 1994
Benzimidazoles useful in treating epithelial disorders
JANSSEN PHARMACEUTICA NV16 citations81
US4767760AAug 30, 1988
Anti-protozoal 5,6-dihydro-2-(substituted phenyl)-1,2,4-triazine-3,5(2H,4H)-dione derivatives, compositions, and method of use therefor
JANSSEN PHARMACEUTICA NV16 citations81
US5043327AAug 27, 1991
Positive inotropic and lusitropic 3,5-dihydroimidazo[2,1-b]quinazolin-2(1H)-one derivatives, compositions and use
JANSSEN PHARMACEUTICA NV17 citations74
US4826862AMay 2, 1989
Anthelminthic [(5(6) (1H-azole-1-ylmethyl)benzimidazole]carbamates
JANSSEN PHARMACEUTICA NV11 citations74
US5612354AMar 18, 1997
(1H-azol-1-ylmethyl)substituted quinoline derivatives
JANSSEN PHARMACEUTICA NV13 citations73
US5541325AJul 30, 1996
Intermediates for the preparation of 1,3,dihydro-2H-imidazo[4,5-B]quinolin-2-one derivatives
JANSSEN PHARMACEUTICA NV7 citations73
US5420147AMay 30, 1995
Method of treating epithelial disorders
JANSSEN PHARMACEUTICA NV11 citations72
US5270464ADec 14, 1993
Anti-HIV-1 tetrahydroimidazo[1,4]benzodiazepin-2-(thi) ones
JANSSEN PHARMACEUTICA NV7 citations72
US4952570AAug 28, 1990
5,6-dihydro-2-(substituted phenyl)-1,2,4-triazine-3,5(2H,4H)-diones
JANSSEN PHARMACEUTICA NV9 citations72
US4179505ADec 18, 1979
5-[4-(Diarylmethyl)-1-piperazinylalkyl]benzimidazole derivatives
JANSSEN PHARMACEUTICA NV15 citations71
US4032536AJun 28, 1977
(1h-benzimidazol-2-yl)carbamates
JANSSEN PHARMACEUTICA NV15 citations67
US5220023AJun 15, 1993
Glycine derivatives
JANSSEN PHARMACEUTICA NV2 citations63
US5120845AJun 9, 1992
Positive inotropic and lusitropic 3,5-dihydroimidazo[2,1-b]quinazolin-2(1H)-one derivatives
JANSSEN PHARMACEUTICA NV2 citations63
US5457102AOct 10, 1995
Pyrroloimidazolyl and imidazopyridinyl substituted 1H-benzimidazole derivatives
JANSSEN PHARMACEUTICA NV3 citations62
US5256681AOct 26, 1993
[5(6)-(benzisoxa-,benzisothia-or indazol-3-yl)-1H-benzimidazol-2-yl]carbamates
JANSSEN PHARMACEUTICA NV5 citations62
US5371079ADec 6, 1994
Antiretroviral tetrahydroimidazo[1,4]benzodiazepin-2-(thi)ones
JANSSEN PHARMACEUTICA NV3 citations61
US5039677AAug 13, 1991
6-(1H-azol-1-ylmethyl)-1-(pyrimidinyloxy)-1H benzotriazoles
JANSSEN PHARMACEUTICA NV2 citations61
US4778887AOct 18, 1988
α-aryl-4-(4,5-dihydro-3,5-dioxo-1,2,4-triazin-2(3H)-yl)-benzeneacetonitriles
JANSSEN PHARMACEUTICA NV3 citations61
US5212192AMay 18, 1993
Immunostimulating 6-aryl-5,6-dihydroimidazo[2,1-b]thiazole derivatives
JANSSEN PHARMACEUTICA NV6 citations56
US6201119B1Mar 13, 2001
Antiretroviral tetrahydroimidazo[1,4]benzodiazepin-2(thi) ones
JANSSEN PHARMACEUTICA NV0 citations51
US5441954AAug 15, 1995
(1h-azol-1-ylmethyl) substituted quinoline derivatives
JANSSEN PHARMACEUTICA NV0 citations51
US5180832AJan 19, 1993
(3-pyridinyl)methanone oxime derivatives
JANSSEN PHARMACEUTICA NV0 citations51
US4963573AOct 16, 1990
[[[(3-pyridinyl)methylen]amino]oxy]alkanoic acids and esters
JANSSEN PHARMACEUTICA NV0 citations51
US4746671AMay 24, 1988
Pharmaceutical use of [[[(3-pyridinyl)methylen]amino]oxy]alkanoic acids and esters
JANSSEN PHARMACEUTICA NV1 citations51
US5602134AFeb 11, 1997
Positive inotropic and lusitropic pyrroloquinolinone derivatives
JANSSEN PHARMACEUTICA NV0 citations42
US5527915AJun 18, 1996
Immunostimulating 6-aryl-5,6-dihydroimidazo[2,1-beta]thiazole derivatives
JANSSEN PHARMACEUTICA NV0 citations30