Inventor
LEVIN JEREMY I
US42 patents
⚠️ This page may combine multiple inventors who share the name “LEVIN JEREMY I”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
AMERICAN CYANAMID CO
31 patentsUS6225311B1May 1, 2001
Acetylenic α-amino acid-based sulfonamide hydroxamic acid tace inhibitors
AMERICAN CYANAMID CO90 citations96
US5104869AApr 14, 1992
Renin inhibitors
AMERICAN CYANAMID CO120 citations95
US6313123B1Nov 6, 2001
Acetylenic sulfonamide thiol tace inhibitors
AMERICAN CYANAMID CO40 citations93
US6277885B1Aug 21, 2001
Acetylenic aryl sulfonamide and phosphinic acid amide hydroxamic acid TACE inhibitors
AMERICAN CYANAMID CO20 citations93
US6534491B2Mar 18, 2003
Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
AMERICAN CYANAMID CO32 citations92
US6326516B1Dec 4, 2001
Acetylenic β-sulfonamido and phosphinic acid amide hydroxamic acid TACE inhibitors
AMERICAN CYANAMID CO36 citations92
US6228869B1May 8, 2001
Ortho-sulfonamido bicyclic hydroxamic acids as matrix metalloproteinase and TACE inhibitors
AMERICAN CYANAMID CO17 citations92
US5294617AMar 15, 1994
Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
AMERICAN CYANAMID CO26 citations92
US5290780AMar 1, 1994
Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
AMERICAN CYANAMID CO29 citations92
US5281603AJan 25, 1994
Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
AMERICAN CYANAMID CO24 citations92
US6340691B1Jan 22, 2002
Alkynyl containing hydroxamic acid compounds as matrix metalloproteinase and tace inhibitors
AMERICAN CYANAMID CO42 citations91
US6548524B2Apr 15, 2003
Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and TACE inhibitors
AMERICAN CYANAMID CO18 citations84
US6200996B1Mar 13, 2001
Heteroaryl acetylenic sulfonamide and phosphinic acid amide hydroxamic acid tace inhibitors
AMERICAN CYANAMID CO18 citations84
US4904658AFeb 27, 1990
Substituted-6H,8H-pyrimido-[1,2,3-cd]purine-8,10-(9H)-diones and substituted-6H,10H-pyrimido[1,2-cd]purin-10-ones
AMERICAN CYANAMID CO19 citations82
US6498167B2Dec 24, 2002
Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
AMERICAN CYANAMID CO6 citations74
US5358951AOct 25, 1994
Angiotensin II receptor blocking 2, 3, 6 substituted quinazolinones
AMERICAN CYANAMID CO19 citations74
US5292742AMar 8, 1994
Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
AMERICAN CYANAMID CO7 citations74
US5284853AFeb 8, 1994
Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
AMERICAN CYANAMID CO12 citations74
US5281604AJan 25, 1994
Angiotensin II receptor blocking 2,3,6-substituted quinazolinones
AMERICAN CYANAMID CO12 citations74
US5084457AJan 28, 1992
Benzoylaminoquinazolinones
AMERICAN CYANAMID CO14 citations73
US6358980B1Mar 19, 2002
Alkynyl containing hydroxamic acid compounds as matrix metalloproteinase/tace inhibitors
AMERICAN CYANAMID CO8 citations72
US5405849AApr 11, 1995
Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
AMERICAN CYANAMID CO2 citations63
US5298517AMar 29, 1994
Angiotensin II receptor blocking agents
AMERICAN CYANAMID CO6 citations63
US5294611AMar 15, 1994
Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
AMERICAN CYANAMID CO2 citations63
US5292734AMar 8, 1994
Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
AMERICAN CYANAMID CO5 citations63
US5284852AFeb 8, 1994
Angiotensin II receptor blocking 2,3,6-substituted quinazolinones
AMERICAN CYANAMID CO2 citations63
US5013737AMay 7, 1991
2,4,8-Trisubstituted-3H,6H-1,4,5A,8A-tetraazaacenaphtylene-3,5-(4H)-diones and 2,4-8-trisubstituted-4,5-dihydro-5-thioxo-3H,6H-1,4,5A,8A-tetrazaacenaphthylen-3-ones
AMERICAN CYANAMID CO2 citations62
US4916137AApr 10, 1990
5-(Substituted-amino)-8-(phenyl or substituted-phenyl)-3H,6H-1,4,5A,8A-tetraazaacenaphthylen-3-ones and treatment of neural behavior disorders
AMERICAN CYANAMID CO5 citations62
US5338736AAug 16, 1994
Angiotensin II receptor blocking 2,3,6-substituted quinazolinones
AMERICAN CYANAMID CO1 citations52
US5286729AFeb 15, 1994
Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
AMERICAN CYANAMID CO1 citations52
US5932585AAug 3, 1999
Method of treating or inhibiting neutropenia
AMERICAN CYANAMID CO0 citations35
WYETH CORP
10 patentsUS6716833B2Apr 6, 2004
Acetylenic α-amino acid-based sulfonamide hydroxamic acid tace inhibitors
WYETH CORP6 citations72
US6762178B2Jul 13, 2004
Acetylenic aryl sulfonamide and phosphinic acid amide hydroxamic acid TACE inhibitors
WYETH CORP3 citations63
US6812227B2Nov 2, 2004
Acetylenic α-amino acid-based sulfonamide hydroxamic acid tace inhibitors
WYETH CORP4 citations61
US6753337B2Jun 22, 2004
Alkynyl containing hydroxamic acid compounds as matrix metalloproteinase/tace inhibitors
WYETH CORP5 citations61
US6946473B2Sep 20, 2005
Preparation and use of acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as TACE inhibitors
WYETH CORP3 citations59
US7179911B2Feb 20, 2007
Method for preparing hydroxamic acids
WYETH CORP3 citations57
US7488754B2Feb 10, 2009
Method for the treatment of polycystic kidney disease
WYETH CORP1 citations52
US6825354B2Nov 30, 2004
Alkynyl containing hydroxamic acid compounds as matrix metalloproteinase and TACE inhibitors
WYETH CORP1 citations51
US7576222B2Aug 18, 2009
Alkynyl-containing tryptophan derivative inhibitors of TACE/matrix metalloproteinase
WYETH CORP0 citations39
US7595327B2Sep 29, 2009
Beta-sulfonamide hydroxamic acid inhibitors of tace/matrix metalloproteinase
WYETH CORP0 citations35