Inventor
KADIN SAUL B
35 patents
Patents
35 patentsUS4556672ADec 3, 1985
3-Substituted 2-oxindole-1-carboxamides as analgesic and anti-inflammatory agents
PFIZER90 citations96
US4721712AJan 26, 1988
1,3-disubstituted 2-oxindoles as analgesic and anti-inflammatory agents
PFIZER30 citations92
US4569942AFeb 11, 1986
N,3-Disubstituted 2-oxindole-1-carboxamides as analgesic and antiinflammatory agents
PFIZER36 citations92
US4725616AFeb 16, 1988
1,3-dicarboxamide-oxindoles as antiinflammatory agents
PFIZER20 citations82
US4658037AApr 14, 1987
Intermediates for 1,3-disubstituted 2-oxindoles as analgesic and antiinflammatory agents
PFIZER18 citations82
US4535081AAug 13, 1985
Antiallergic and antiulcer 1-oxo-1H-thiazolo[3,2-a]pyrimidine-2-carboxamides and intermediates therefor
PFIZER19 citations82
US4075343AFeb 21, 1978
Anti-allergenic 5-alkoxyimidazo[1,2-A]quinoline-2-carboxylic acids and derivatives thereof
PFIZER26 citations82
US4808601AFeb 28, 1989
Analgesic and antiinflammatory 1,3-diacyl-2-oxindole compounds
PFIZER10 citations74
US4791129ADec 13, 1988
1,3-dicarboxamidooxindoles as analgesic and antiinflammatory agents
PFIZER15 citations74
US4752609AJun 21, 1988
Analgesic and antiinflammatory 1,3-diacyl-2-oxindole compounds
PFIZER8 citations74
US4690943ASep 1, 1987
Analgesic and antiinflammatory 1,3-diacyl-2-oxindole compounds
PFIZER15 citations74
US4678802AJul 7, 1987
1-acylcarbamoyloxindole-3-carboxamides as antiinflammatory agents
PFIZER13 citations74
US4623725ANov 18, 1986
[1,2,4]Triazolo[4,3-a]quinoxaline-4-amine derivatives
PFIZER10 citations74
US4423048ADec 27, 1983
Antiallergic and antiulcer 1-oxo-1H-thiazolo[3,2-a]pyrimidine-2-carboxamides and intermediates therefor
PFIZER7 citations74
US4321372AMar 23, 1982
Antiulcer thiazol-2-ylcarbamoyl-carboxylic acids, esters and amides
PFIZER8 citations74
US4296129AOct 20, 1981
(Carboxyacylamino)phenylalkenamides and esters thereof as SRS-A antagonists
PFIZER11 citations74
US4296120AOct 20, 1981
(Carboxy-oxo-pyrrolidino)phenylalkenamides and esters thereof as SRS-A antagonists
PFIZER9 citations74
US4066766AJan 3, 1978
1-Oxo-6-substituted pyrimido [1,2-a]quinoline-2-carboxylic acids and derivatives thereof and their use as antiallergy agents
PFIZER9 citations74
US4041163AAug 9, 1977
N-(5-Tetrazolyl)-4-oxo-4H-pyrimido(2,1-b)benzothiazole-3-carboxamide antiallergy agents
PFIZER14 citations74
US4017625AApr 12, 1977
Anti-allergic N-(5-tetrazolyl)-1-oxo-1H-6-alkoxypyrimido-[1,2-a]quinoline-2-carboxamides and intermediates therefor
PFIZER13 citations74
US3998954ADec 21, 1976
1,3(2H,4H)-Dioxoisoquinoline-4-carboxamides used as anti-inflammatory agents
PFIZER12 citations74
US4791131ADec 13, 1988
Analgesic and antiinflammatory 1-acyl-2-oxindole-3-carboxamides
PFIZER2 citations63
US4730004AMar 8, 1988
Analgesic and anti-inflammatory 1-acyl-2-oxindole-3-carboxamides
PFIZER5 citations63
US4414388ANov 8, 1983
1-Oxo-1H-thiazolo[3,2-a]pyrimidine-2-carboxamides
PFIZER2 citations63
US4247699AJan 27, 1981
Process for making 2-amino-4-hydroxyquinolines
PFIZER6 citations63
US4175193ANov 20, 1979
2-Amino-3-cyano-4-hydroxyquinolines
PFIZER4 citations63
US4134981AJan 16, 1979
Pyrimidal [2,3,d]Pyrimidin-4(3H)-ones as antiallergy agents
PFIZER2 citations62
US4044134AAug 23, 1977
Fused pyrimidin-4(3H)-ones as antiallergy agents
PFIZER5 citations62
US3974161AAug 10, 1976
Fused pyrimidin-4(3H)-ones as antiallergy agents
PFIZER4 citations62
US4031217AJun 21, 1977
1-Oxo-1H-6-substituted-pyrimido(1,2-a)-quinoline-2-carboxylic acids and esters useful as antiulcer agents
PFIZER3 citations57
US4014881AMar 29, 1977
1-Oxo-1H-6-piperidinopyrimido[1,2-a]quinoline-2-carboxylic acids and esters
PFIZER3 citations57
US4343813AAug 10, 1982
Carboxamide compounds as SRS-A antagonists
PFIZER0 citations52
US4342781AAug 3, 1982
Diphenylpropenamides as SRS-A antagonists
PFIZER1 citations52
US4331683AMay 25, 1982
Carboxamide compounds as SRS-A antagonists
PFIZER0 citations52
US4120962AOct 17, 1978
Fused pyrimidin-4(3H)-ones as antiallergy agents
PFIZER0 citations51