Inventor
BAGGIOLINI ENRICO G
US26 patents
Patents
26 patentsUS5512554AApr 30, 1996
Method of treating hyperproliferative skin diseases with fluorinated vitamin D3 analogs
HOFFMANN LA ROCHE43 citations96
US4804502AFeb 14, 1989
Vitamin D compounds
HOFFMANN LA ROCHE88 citations96
US5451574ASep 19, 1995
Vitamin D3 Flourinated Analogs
HOFFMANN LA ROCHE36 citations95
US5145846ASep 8, 1992
Vitamin D3 analogs
HOFFMANN LA ROCHE72 citations95
US4508651AApr 2, 1985
Synthesis of 1α,25-dihydroxyergocalciferol
HOFFMANN LA ROCHE57 citations95
US5087619AFeb 11, 1992
Vitamin D3 analogs
HOFFMANN LA ROCHE71 citations94
US5120722AJun 9, 1992
Trihydroxy-cholecacliferol and trihydroxy-ergocalciferol for treating leukemia
HOFFMANN LA ROCHE30 citations92
US4594432AJun 10, 1986
Process for the synthesis of 1α,23(S),25-trihydroxycholecalciferol and 1α,23(R),25-trihydroxycholecalciferol
HOFFMANN LA ROCHE33 citations92
US4898855AFeb 6, 1990
Deuterated analogs of 1,25-dihydroxycholecalciferol
HOFFMANN LA ROCHE21 citations81
US4612308ASep 16, 1986
25,26-Dehydro-1α,23(S,R)-dihydroxycholecalciferol and its epimers
HOFFMANN LA ROCHE21 citations81
US4225525ASep 30, 1980
Vitamin D3 metabolite derivatives
HOFFMANN LA ROCHE7 citations74
US5247123ASep 21, 1993
Deuterated analogs of 1,25-dihydroxycholecalciferol
HOFFMANN LA ROCHE8 citations73
US5149846ASep 22, 1992
Deuterated analogs of 1,25-dihydroxycholecalciferol
HOFFMANN LA ROCHE8 citations73
US5039671AAug 13, 1991
Trifluorinated-1α,25S-dihydroxy vitamin D3 compounds
HOFFMANN LA ROCHE8 citations73
US4595776AJun 17, 1986
Synthesis of 1α,25-dihydroxyergocalciferol
HOFFMANN LA ROCHE10 citations73
US4130713ADec 19, 1978
Biotin intermediates
HOFFMANN LA ROCHE13 citations73
US4632784ADec 30, 1986
Process for the preparation of 1α,23,25-trihydroxycholecalciferol-26-oic acid 23,26-lactone
HOFFMANN LA ROCHE5 citations62
US4284557AAug 18, 1981
Intermediate racemates for the preparation of biotin and a process for their preparation
HOFFMANN LA ROCHE2 citations62
US4247704AJan 27, 1981
Hexahydro thieno imadazole intermediates for the synthesis of biotin
HOFFMANN LA ROCHE3 citations62
US4245104AJan 13, 1981
Isoxazolines and isoxazolidines
HOFFMANN LA ROCHE2 citations62
US4189586AFeb 19, 1980
Preparation of biotin
HOFFMANN LA ROCHE4 citations62
US4906785AMar 6, 1990
Novel trifluorinated vitamin D3 intermediates
HOFFMANN LA ROCHE4 citations58
US5110958AMay 5, 1992
Compounds, process and intermediates
HOFFMANN LA ROCHE1 citations51
US4382031AMay 3, 1983
Intermediates for the preparation of biotin
HOFFMANN LA ROCHE0 citations51
US4337345AJun 29, 1982
Preparation of biotin via thieno [3,2c] isoxazoles
HOFFMANN LA ROCHE1 citations51
US4320056AMar 16, 1982
Certain thia-diazatricyclo[3,3,3,08,11 ]tridecanes, and their preparation
HOFFMANN LA ROCHE1 citations51