Inventor
YAICHE PHILIPPE
FR43 patents
⚠️ This page may combine multiple inventors who share the name “YAICHE PHILIPPE”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
SANOFI AVENTIS
14 patentsUS7067521B2Jun 27, 2006
1-[alkyl], 1-[(heteroaryl)alkyl] and 1-[(aryl)alkyl]-7pyridinyl-imidazo[1,2-alpha]pyrimidin-5(1H)-one derivatives
SANOFI AVENTIS2 citations62
US7507743B2Mar 24, 2009
Substituted 8′-pyridinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a] pyrimidin-6-one and 8′-pyrimidinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a] pyrimidin-6-one derivatives
SANOFI AVENTIS1 citations52
US7465737B2Dec 16, 2008
Heteroaryl substituted 2-pyridinyl and 2-pyrimidinyl -6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one derivatives
SANOFI AVENTIS1 citations52
US7452897B2Nov 18, 2008
Use of substituted 2-(diaza-bicyclo-alkyl)-pyrimidone derivatives for the treatment of neurodegenerative diseases
SANOFI AVENTIS0 citations52
US7393853B2Jul 1, 2008
Use of substituted 8-Perfluoroalkyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one derivatives as therapeutic agents
SANOFI AVENTIS0 citations52
US7294632B2Nov 13, 2007
Substituted 8′-pyridinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a]pyrimidin-6-one and 8′-pyrimidinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a]pyrimidin-6-one derivatives
SANOFI AVENTIS0 citations52
US7781440B2Aug 24, 2010
Use of substituted 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one and 7-pyrimidinyl-2,3-dihydroimidazo[1,2-a] pyrimidin-5(1H)one derivatives
SANOFI AVENTIS1 citations51
US7608624B2Oct 27, 2009
1-[alkyl], 1-[(heteroaryl)alkyl] and 1-[(aryl)alkyl]-7-pyridinyl-imidazo[1,2-a]pyrimidin-5(1h)-one derivatives
SANOFI AVENTIS0 citations51
US7566720B2Jul 28, 2009
2-pyridinyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one and 7-pyridinyl-2,3-dihydroimidazo[1,2-a] pyrimidin-5(1H)one derivatives
SANOFI AVENTIS1 citations51
US7547705B2Jun 16, 2009
Substituted 8′-pyri(MI)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a]pyrimidin-6-one derivatives
SANOFI AVENTIS1 citations51
US7462621B2Dec 9, 2008
Use of substituted 2-pyridinyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one and 7-pyridinyl-2,3-dihydroimidazo[1,2-a] pyrimidin-5(1H)one derivatives as therapeutic agents
SANOFI AVENTIS1 citations51
US7388005B2Jun 17, 2008
Substituted 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-one and 7-pyrimidinyl-2,3-dihydroimidazo [1,2-a]pyrimidin-5(1H)one derivatives for neurodegenerative disorders
SANOFI AVENTIS0 citations51
US7294631B2Nov 13, 2007
Substituted 8′-pyri(MI)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a]pyrimidin-6-one derivatives
SANOFI AVENTIS0 citations51
US7429663B2Sep 30, 2008
7-(Pyrimidin-4-yl)-Imidazo[1,2-a]Pyrimidin-5(1H)-ones as GSK3β inhibitors
SANOFI AVENTIS0 citations42
LOCHEAD ALISTAIR
7 patentsUS8592437B2Nov 26, 2013
Heteroarylamide pyrimidone compounds
LOCHEAD ALISTAIR6 citations71
US8592580B2Nov 26, 2013
Substituted triazinone derivatives
LOCHEAD ALISTAIR2 citations62
US8598187B2Dec 3, 2013
Arylamide pyrimidone compounds
LOCHEAD ALISTAIR1 citations51
US8211903B2Jul 3, 2012
Substituted pyrimido isoquinoline derivatives
LOCHEAD ALISTAIR0 citations51
US8202874B2Jun 19, 2012
Substituted N-oxide pyrazine derivatives
LOCHEAD ALISTAIR0 citations51
US8093256B2Jan 10, 2012
Use of 8-substituted-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one derivatives
LOCHEAD ALISTAIR0 citations51
US9073915B2Jul 7, 2015
Substituted pyrimidone derivatives
LOCHEAD ALISTAIR0 citations41
FAYOL AUDE
7 patentsUS8507476B2Aug 13, 2013
Substituted arylamide diazepinopyrimidone derivatives
FAYOL AUDE1 citations50
US9073914B2Jul 7, 2015
Substituted alkyl pyrimidin-4-one derivatives
FAYOL AUDE0 citations39
US8614219B2Dec 24, 2013
Substituted pyrimidin-4-one derivatives
FAYOL AUDE0 citations39
US8507475B2Aug 13, 2013
Substituted heteroarylamide diazepinopyrimidone derivatives
FAYOL AUDE0 citations39
US8507470B2Aug 13, 2013
Substituted arylamide oxazepinopyrimidone derivatives
FAYOL AUDE0 citations39
US8501728B2Aug 6, 2013
Substituted heteroarylamide oxazepinopyrimidone derivatives
FAYOL AUDE0 citations39
US8198287B2Jun 12, 2012
Substituted heteroaryl pyridopyrimidone derivatives
FAYOL AUDE0 citations39
MITSUBISHI PHARMA CORP
6 patentsUS7247638B2Jul 24, 2007
8-Substituted-6,7,8,9-tetrahydropyrimido [1,2-a] pyrimidin-4-one derivatives.
MITSUBISHI PHARMA CORP2 citations62
US7232827B2Jun 19, 2007
Heteroaryl substituted 2-pyridinyl and 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-one derivatives
MITSUBISHI PHARMA CORP5 citations62
US7217715B2May 15, 2007
Substituted 8-perfluoroalkyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one derivatives
MITSUBISHI PHARMA CORP2 citations62
US7214682B2May 8, 2007
Substituted 2-pyridinyl-6,7,8,9-tetrahydropyrimido{1,2-a}pyrimidin-4-one and 7-pyridinyl-2,3-dihydroimidazo{1,2-a}pyrimidin-5(1h)one derivatives
MITSUBISHI PHARMA CORP2 citations61
US6974819B2Dec 13, 2005
2-pyridinyl-6,7,8,9-tetrahydropyrimido{1,2-a}pyrimidin-4-one and 7-pyridinyl-2,3-dihydoimidazo{1,2-a}pyrimidin-5(1H)one derivatives
MITSUBISHI PHARMA CORP2 citations61
US7211581B2May 1, 2007
Substituted 2-(diaza-bicyclo-alkyl)-pyrimidone derivatives
MITSUBISHI PHARMA CORP0 citations52
ABOUABDELLAH AHMED
5 patentsUS8697883B2Apr 15, 2014
Cyclopenta[C]pyrrole-2-carboxylate derivatives, preparation thereof and therapeutic use thereof
ABOUABDELLAH AHMED19 citations82
US8394787B2Mar 12, 2013
7-aza-spiro[3.5]nonane-7-carboxylate derivatives, preparation thereof and therapeutic use thereof
ABOUABDELLAH AHMED6 citations71
US8889702B2Nov 18, 2014
Derivatives of azaspiranyl-alkylcarbamates of 5-member heterocyclic compounds, preparation thereof and therapeutic use thereof
ABOUABDELLAH AHMED2 citations61
US8865738B2Oct 21, 2014
5-membered heterocyclic compound cyclopenta[C]pyrrolylalkylcarbamate derivatives, preparation thereof, and therapeutic use thereof
ABOUABDELLAH AHMED3 citations61
US8716289B2May 6, 2014
Carbamate derivatives of alkyl-heterocycles, preparation thereof and therapeutic use thereof
ABOUABDELLAH AHMED1 citations50