Inventor
SZMUSZKOVICZ JACOB
38 patents
⚠️ This page may combine multiple inventors who share the name “SZMUSZKOVICZ JACOB”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
UPJOHN CO
36 patentsUS4212878AJul 15, 1980
Phenylacetamide derivative analgesics
UPJOHN CO69 citations96
US4145435AMar 20, 1979
2-aminocycloaliphatic amide compounds
UPJOHN CO135 citations96
US4098904AJul 4, 1978
Analgesic n-(2-aminocycloaliphatic)benzamides
UPJOHN CO78 citations96
US4359476ANov 16, 1982
Adjacently substituted cycloalkane-amide analgesics
UPJOHN CO61 citations95
US4540690ASep 10, 1985
2-(Phenylmethylene)cycloalkylamines and -azetidines
UPJOHN CO33 citations92
US4360531ANov 23, 1982
Substituted cycloalkanes
UPJOHN CO36 citations92
US4179501ADec 18, 1979
Analgesic N-(2-aminocycloaliphatic)azidobenzamides
UPJOHN CO46 citations92
US4466977AAug 21, 1984
N-[2-Amino(oxy- or thia- group-substituted-cycloaliphatic)]benzeneacetamides and -benzamide analgesics
UPJOHN CO24 citations81
US4801604AJan 31, 1989
Cis-N-(2-aminocycloaliphatic)benzamide anti-convulsants
UPJOHN CO22 citations76
US4652559AMar 24, 1987
2-(Phenylmethylene)cycloalkyl-azetidines
UPJOHN CO11 citations74
US4204003AMay 20, 1980
N-(2-Aminocyclopentyl)-N-alkanoylanilides as CNS anti-depressants
UPJOHN CO17 citations74
US4156733AMay 29, 1979
N-(2-Aminocyclopentyl) alkanoylanilides
UPJOHN CO4 citations74
US4152459AMay 1, 1979
Analgesic N-2-(aminocycloaliphatic)-hydroxy, alkoxy and (allylic)alkenyloxy-benzamides
UPJOHN CO5 citations74
US4148914AApr 10, 1979
Analgesic N-(2-aminocyclo aliphatic)cyanobenzamides
UPJOHN CO4 citations74
US3966736AJun 29, 1976
2,9-Dihydro-3H-pyrido[3,2-c]-s-triazolo[4,3-a][1,5]-benzodiazepin-3-ones
UPJOHN CO16 citations74
US3933816AJan 20, 1976
3-(Substituted aminomethyl)-7-substituted-3,5-dihydro-as-triazino[4,3-a][1,5]benzodiazepines
UPJOHN CO10 citations74
US4460600AJul 17, 1984
Adjacently substituted ketal derivatives of cycloalkane-amide analgesics
UPJOHN CO13 citations73
US4197308AApr 8, 1980
Analgesic N-(2-heterocyclic-amino cycloaliphatic) benzamides
UPJOHN CO5 citations63
US4192885AMar 11, 1980
Analgesic N-{2-[N'-(2-furylmethyl and 2-thienyl-methyl)-N'-alkylamino]cycloaliphatic}cyanobenzamides
UPJOHN CO5 citations63
US4159340AJun 26, 1979
N-(2-Aminocyclopentyl)-N-acylanilides as CNS anti-depressants
UPJOHN CO3 citations63
US4156015AMay 22, 1979
N-(2-Aminocyclopentyl)acylanilides and treating depression
UPJOHN CO2 citations63
US4153717AMay 8, 1979
Analgesic N-(2-(furylmethylamino and 2 -thienylmethylamino)cyclo aliphatic)benzamides
UPJOHN CO3 citations63
US4598088AJul 1, 1986
2-pyrrolyl-cycloalkyl-amide analgesics
UPJOHN CO4 citations62
US4590187AMay 20, 1986
Phospholipase A2 inhibition using 4,1-benzoxazepine-2-(3H)-ones
UPJOHN CO3 citations62
US4217362AAug 12, 1980
Anilide derivatives as antidepressants
UPJOHN CO0 citations52
US4212888AJul 15, 1980
Anilide derivatives as antidepressants
UPJOHN CO0 citations52
US4157398AJun 5, 1979
N-(2-Aminocyclopentyl)acylanilides and treating depression
UPJOHN CO0 citations52
US4156014AMay 22, 1979
N-(2-aminocycloheptyl)alkanoylanilides and in the treatment of depression
UPJOHN CO1 citations52
US4128663ADec 5, 1978
Anilide derivatives as antidepressants
UPJOHN CO1 citations52
US4286106AAug 25, 1981
N-[ω-(Dimethylamino)alkyl]-3',4'-dichloropropionanilides
UPJOHN CO1 citations48
US4186208AJan 29, 1980
Anti-depressant N-(3,4-dichlorophenyl)-N-dimethylaminoalkylene amides
UPJOHN CO1 citations48
US4180522ADec 25, 1979
N-(2-Dimethylaminoalkyl)-3',4'-dichloroanilides
UPJOHN CO1 citations48
US4978753ADec 18, 1990
7-phenylpyrimido[1,2-alpha][1,4]benzodiazepin-3(5H)-ones
UPJOHN CO0 citations42
US4172898AOct 30, 1979
N-(2-aminocycloheptyl)acylanilides
UPJOHN CO0 citations42
US4169156ASep 25, 1979
N-(2-aminocycloheptyl)alkanoylanilides
UPJOHN CO0 citations42
US4159339AJun 26, 1979
N-(2-Aminocycloheptyl) alkanoylanilides
UPJOHN CO0 citations42