P

Inventor

HEERES JAN

124 patents
⚠️ This page may combine multiple inventors who share the name “HEERES JAN”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.

JANSSEN PHARMACEUTICA NV

41 patents
US7514445B2Apr 7, 2009

Heteroaryl amines as glycogen synthase kinase 3β inhibitors (GSK3 inhibitors)

JANSSEN PHARMACEUTICA NV117 citations97
US7125879B2Oct 24, 2006

HIV inhibiting pyrimidines derivatives

JANSSEN PHARMACEUTICA NV96 citations97
US6150360ANov 21, 2000

Trisubstituted 1,3,5-Triazine Derivatives

JANSSEN PHARMACEUTICA NV62 citations96
US4267179AMay 12, 1981

Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles

JANSSEN PHARMACEUTICA NV111 citations96
US4223036ASep 16, 1980

1-(1,3-Dioxolan-2-ylmethyl)-1H-1,2,4-triazoles

JANSSEN PHARMACEUTICA NV41 citations96
US4144346AMar 13, 1979

Novel 1-(1,3-dioxolan-2-ylmethyl)-1H-imidazoles

JANSSEN PHARMACEUTICA NV79 citations96
US3936470AFeb 3, 1976

1,3-Dioxolan-2-ylmethylimidazoles

JANSSEN PHARMACEUTICA NV40 citations96
US6440986B2Aug 27, 2002

HIV Inhibiting pyrimidine derivatives

JANSSEN PHARMACEUTICA NV74 citations95
US4916134AApr 10, 1990

4-[4-[4-[4-[[2-(2,4-difluorophenyl)-2-(1H-azolylmethyl)-1,3-dioxolan-4-yl]me]phenyl]-1-piperazinyl]phenyl]triazolones

JANSSEN PHARMACEUTICA NV52 citations95
US7037917B2May 2, 2006

HIV replication inhibiting pyrimidines

JANSSEN PHARMACEUTICA NV34 citations94
US4160838AJul 10, 1979

Antimicrobial and plant-growth-regulating triazole derivatives

JANSSEN PHARMACEUTICA NV65 citations94
US4079062AMar 14, 1978

Triazole derivatives

JANSSEN PHARMACEUTICA NV112 citations94
US5998413ADec 7, 1999

Itraconazole and stereoisomers

JANSSEN PHARMACEUTICA NV19 citations92
US5811426ASep 22, 1998

Urea and thiourea derivatives of azolones

JANSSEN PHARMACEUTICA NV28 citations92
US5639754AJun 17, 1997

Urea and thiourea derivatives of azolones

JANSSEN PHARMACEUTICA NV32 citations92
US5637592AJun 10, 1997

Acyl derivatives of azolones

JANSSEN PHARMACEUTICA NV42 citations92
US5571811ANov 5, 1996

Sulfonamide derivatives of azolones

JANSSEN PHARMACEUTICA NV23 citations92
US4931444AJun 5, 1990

5-lipoxygenase inhibiting 4-(4-phenyl-1-piperazinyl)phenols

JANSSEN PHARMACEUTICA NV55 citations92
US4619931AOct 28, 1986

[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles

JANSSEN PHARMACEUTICA NV31 citations92
US4598085AJul 1, 1986

Fungicidal 1-(2-aryl-2-R-ethyl)-1H-1,2,4-triazoles

JANSSEN PHARMACEUTICA NV57 citations92
US4335125AJun 15, 1982

1-(1,3-Dioxolan-2-ylmethyl)-1H-imidazoles

JANSSEN PHARMACEUTICA NV33 citations92
US3991201ANov 9, 1976

1-(β-Aryl-β-R-ethyl)imidazoles as antimicrobial agents

JANSSEN PHARMACEUTICA NV36 citations92
US7923554B2Apr 12, 2011

HIV inhibiting 1,2,4-triazin-6-one derivatives

JANSSEN PHARMACEUTICA NV26 citations91
US5929075AJul 27, 1999

Apolipoprotein-B synthesis inhibitors

JANSSEN PHARMACEUTICA NV26 citations91
US5728700AMar 17, 1998

Sulfonamide compounds of azolones anti-helicobacter agents

JANSSEN PHARMACEUTICA NV41 citations91
US5707977AJan 13, 1998

Watersoluble azole antifungals

JANSSEN PHARMACEUTICA NV22 citations91
US5650411AJul 22, 1997

Substituted azolone derivatives

JANSSEN PHARMACEUTICA NV24 citations90
US7399856B2Jul 15, 2008

Processes for the preparation of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-2pyrimidinyl]amino]benzonitrile

JANSSEN PHARMACEUTICA NV19 citations89
US5521186AMay 28, 1996

Apolipoprotein-β synthesis inhibitors

JANSSEN PHARMACEUTICA NV24 citations89
US4791111ADec 13, 1988

[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles having anti-microbial properties

JANSSEN PHARMACEUTICA NV52 citations89
US7034019B2Apr 25, 2006

Prodrugs of HIV replication inhibiting pyrimidines

JANSSEN PHARMACEUTICA NV14 citations83
US8003789B2Aug 23, 2011

HIV replication inhibiting pyrimidines

JANSSEN PHARMACEUTICA NV12 citations82
US4358449ANov 9, 1982

1-(1,3-Dioxolan-2-ylmethyl)-1H-1,2,4-triazoles and compositions

JANSSEN PHARMACEUTICA NV20 citations82
US4156008AMay 22, 1979

1-(4-Alkyl-2-aryl-1,3-dioxolan-2-ylmethyl)-1H-imidazoles

JANSSEN PHARMACEUTICA NV18 citations82
US4101666AJul 18, 1978

1-(2-Ar-4-R-1,3-dioxolan-2-ylmethyl)imidazoles

JANSSEN PHARMACEUTICA NV15 citations82
US4101665AJul 18, 1978

1-(2-Ar-4-aryloxymethyl-1,3-dioxolan-2-ylmethyl)imidazoles

JANSSEN PHARMACEUTICA NV14 citations82
US4490540ADec 25, 1984

(2-Aryl-4-phenylthioalkyl-1,3-dioxolan-2-ylmethyl)azole derivatives

JANSSEN PHARMACEUTICA NV23 citations81
US5710156AJan 20, 1998

Ester and carbamate derivatives of azolones

JANSSEN PHARMACEUTICA NV17 citations80
US4329342AMay 11, 1982

1-(2-Aryl-4,5-disubstituted-1,3-dioxolan-2-ylmethyl)-1H-imidazoles and 1H-1,2,4-triazoles

JANSSEN PHARMACEUTICA NV16 citations79
US5075309ADec 24, 1991

Antifungal 4-[4-[4-[4-[[2-(2,4-difluorophenyl)-2-(1H-azolylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]-1-piperazinyl]phenyl]triazolones and imidazolones

JANSSEN PHARMACEUTICA NV9 citations74
US4735942AApr 5, 1988

[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]-methyl]-1H-imidazoles and 1H-1,2,4-triazoles having antimicrobial properties

JANSSEN PHARMACEUTICA NV8 citations74

JANSSEN PHARMACEUTICA INC

2 patents

TIBOTEC PHARM LTD

2 patents

(unassigned)

2 patents

GUILLEMONT JEROME EMILE GEORGES

2 patents

CORTE BART DE

1 patent

Showing the top 50 of 124 patents by PatentIndex Score.