Inventor
HEERES JAN
124 patents
⚠️ This page may combine multiple inventors who share the name “HEERES JAN”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
JANSSEN PHARMACEUTICA NV
41 patentsUS7514445B2Apr 7, 2009
Heteroaryl amines as glycogen synthase kinase 3β inhibitors (GSK3 inhibitors)
JANSSEN PHARMACEUTICA NV117 citations97
US7125879B2Oct 24, 2006
HIV inhibiting pyrimidines derivatives
JANSSEN PHARMACEUTICA NV96 citations97
US6150360ANov 21, 2000
Trisubstituted 1,3,5-Triazine Derivatives
JANSSEN PHARMACEUTICA NV62 citations96
US4267179AMay 12, 1981
Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV111 citations96
US4223036ASep 16, 1980
1-(1,3-Dioxolan-2-ylmethyl)-1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV41 citations96
US4144346AMar 13, 1979
Novel 1-(1,3-dioxolan-2-ylmethyl)-1H-imidazoles
JANSSEN PHARMACEUTICA NV79 citations96
US3936470AFeb 3, 1976
1,3-Dioxolan-2-ylmethylimidazoles
JANSSEN PHARMACEUTICA NV40 citations96
US6440986B2Aug 27, 2002
HIV Inhibiting pyrimidine derivatives
JANSSEN PHARMACEUTICA NV74 citations95
US4916134AApr 10, 1990
4-[4-[4-[4-[[2-(2,4-difluorophenyl)-2-(1H-azolylmethyl)-1,3-dioxolan-4-yl]me]phenyl]-1-piperazinyl]phenyl]triazolones
JANSSEN PHARMACEUTICA NV52 citations95
US7037917B2May 2, 2006
HIV replication inhibiting pyrimidines
JANSSEN PHARMACEUTICA NV34 citations94
US4160838AJul 10, 1979
Antimicrobial and plant-growth-regulating triazole derivatives
JANSSEN PHARMACEUTICA NV65 citations94
US4079062AMar 14, 1978
Triazole derivatives
JANSSEN PHARMACEUTICA NV112 citations94
US5998413ADec 7, 1999
Itraconazole and stereoisomers
JANSSEN PHARMACEUTICA NV19 citations92
US5811426ASep 22, 1998
Urea and thiourea derivatives of azolones
JANSSEN PHARMACEUTICA NV28 citations92
US5639754AJun 17, 1997
Urea and thiourea derivatives of azolones
JANSSEN PHARMACEUTICA NV32 citations92
US5637592AJun 10, 1997
Acyl derivatives of azolones
JANSSEN PHARMACEUTICA NV42 citations92
US5571811ANov 5, 1996
Sulfonamide derivatives of azolones
JANSSEN PHARMACEUTICA NV23 citations92
US4931444AJun 5, 1990
5-lipoxygenase inhibiting 4-(4-phenyl-1-piperazinyl)phenols
JANSSEN PHARMACEUTICA NV55 citations92
US4619931AOct 28, 1986
[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV31 citations92
US4598085AJul 1, 1986
Fungicidal 1-(2-aryl-2-R-ethyl)-1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV57 citations92
US4335125AJun 15, 1982
1-(1,3-Dioxolan-2-ylmethyl)-1H-imidazoles
JANSSEN PHARMACEUTICA NV33 citations92
US3991201ANov 9, 1976
1-(β-Aryl-β-R-ethyl)imidazoles as antimicrobial agents
JANSSEN PHARMACEUTICA NV36 citations92
US7923554B2Apr 12, 2011
HIV inhibiting 1,2,4-triazin-6-one derivatives
JANSSEN PHARMACEUTICA NV26 citations91
US5929075AJul 27, 1999
Apolipoprotein-B synthesis inhibitors
JANSSEN PHARMACEUTICA NV26 citations91
US5728700AMar 17, 1998
Sulfonamide compounds of azolones anti-helicobacter agents
JANSSEN PHARMACEUTICA NV41 citations91
US5707977AJan 13, 1998
Watersoluble azole antifungals
JANSSEN PHARMACEUTICA NV22 citations91
US5650411AJul 22, 1997
Substituted azolone derivatives
JANSSEN PHARMACEUTICA NV24 citations90
US7399856B2Jul 15, 2008
Processes for the preparation of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-2pyrimidinyl]amino]benzonitrile
JANSSEN PHARMACEUTICA NV19 citations89
US5521186AMay 28, 1996
Apolipoprotein-β synthesis inhibitors
JANSSEN PHARMACEUTICA NV24 citations89
US4791111ADec 13, 1988
[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles having anti-microbial properties
JANSSEN PHARMACEUTICA NV52 citations89
US7034019B2Apr 25, 2006
Prodrugs of HIV replication inhibiting pyrimidines
JANSSEN PHARMACEUTICA NV14 citations83
US8003789B2Aug 23, 2011
HIV replication inhibiting pyrimidines
JANSSEN PHARMACEUTICA NV12 citations82
US4358449ANov 9, 1982
1-(1,3-Dioxolan-2-ylmethyl)-1H-1,2,4-triazoles and compositions
JANSSEN PHARMACEUTICA NV20 citations82
US4156008AMay 22, 1979
1-(4-Alkyl-2-aryl-1,3-dioxolan-2-ylmethyl)-1H-imidazoles
JANSSEN PHARMACEUTICA NV18 citations82
US4101666AJul 18, 1978
1-(2-Ar-4-R-1,3-dioxolan-2-ylmethyl)imidazoles
JANSSEN PHARMACEUTICA NV15 citations82
US4101665AJul 18, 1978
1-(2-Ar-4-aryloxymethyl-1,3-dioxolan-2-ylmethyl)imidazoles
JANSSEN PHARMACEUTICA NV14 citations82
US4490540ADec 25, 1984
(2-Aryl-4-phenylthioalkyl-1,3-dioxolan-2-ylmethyl)azole derivatives
JANSSEN PHARMACEUTICA NV23 citations81
US5710156AJan 20, 1998
Ester and carbamate derivatives of azolones
JANSSEN PHARMACEUTICA NV17 citations80
US4329342AMay 11, 1982
1-(2-Aryl-4,5-disubstituted-1,3-dioxolan-2-ylmethyl)-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV16 citations79
US5075309ADec 24, 1991
Antifungal 4-[4-[4-[4-[[2-(2,4-difluorophenyl)-2-(1H-azolylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]-1-piperazinyl]phenyl]triazolones and imidazolones
JANSSEN PHARMACEUTICA NV9 citations74
US4735942AApr 5, 1988
[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]-methyl]-1H-imidazoles and 1H-1,2,4-triazoles having antimicrobial properties
JANSSEN PHARMACEUTICA NV8 citations74
JANSSEN PHARMACEUTICA INC
2 patentsTIBOTEC PHARM LTD
2 patents(unassigned)
2 patentsGUILLEMONT JEROME EMILE GEORGES
2 patentsCORTE BART DE
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