Inventor
BACKX LEO J J
25 patents
Patents
25 patentsUS4267179AMay 12, 1981
Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV111 citations96
US4223036ASep 16, 1980
1-(1,3-Dioxolan-2-ylmethyl)-1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV41 citations96
US4144346AMar 13, 1979
Novel 1-(1,3-dioxolan-2-ylmethyl)-1H-imidazoles
JANSSEN PHARMACEUTICA NV79 citations96
US4916134AApr 10, 1990
4-[4-[4-[4-[[2-(2,4-difluorophenyl)-2-(1H-azolylmethyl)-1,3-dioxolan-4-yl]me]phenyl]-1-piperazinyl]phenyl]triazolones
JANSSEN PHARMACEUTICA NV52 citations95
US4931444AJun 5, 1990
5-lipoxygenase inhibiting 4-(4-phenyl-1-piperazinyl)phenols
JANSSEN PHARMACEUTICA NV55 citations92
US4619931AOct 28, 1986
[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV31 citations92
US4598085AJul 1, 1986
Fungicidal 1-(2-aryl-2-R-ethyl)-1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV57 citations92
US4335125AJun 15, 1982
1-(1,3-Dioxolan-2-ylmethyl)-1H-imidazoles
JANSSEN PHARMACEUTICA NV33 citations92
US3991201ANov 9, 1976
1-(β-Aryl-β-R-ethyl)imidazoles as antimicrobial agents
JANSSEN PHARMACEUTICA NV36 citations92
US5521186AMay 28, 1996
Apolipoprotein-β synthesis inhibitors
JANSSEN PHARMACEUTICA NV24 citations89
US4791111ADec 13, 1988
[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles having anti-microbial properties
JANSSEN PHARMACEUTICA NV52 citations89
US4358449ANov 9, 1982
1-(1,3-Dioxolan-2-ylmethyl)-1H-1,2,4-triazoles and compositions
JANSSEN PHARMACEUTICA NV20 citations82
US5075309ADec 24, 1991
Antifungal 4-[4-[4-[4-[[2-(2,4-difluorophenyl)-2-(1H-azolylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]-1-piperazinyl]phenyl]triazolones and imidazolones
JANSSEN PHARMACEUTICA NV9 citations74
US4735942AApr 5, 1988
[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]-methyl]-1H-imidazoles and 1H-1,2,4-triazoles having antimicrobial properties
JANSSEN PHARMACEUTICA NV8 citations74
US4524110AJun 18, 1985
Antimicrobial imidazole derivatives
JANSSEN PHARMACEUTICA NV7 citations74
US4490530ADec 25, 1984
Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)-methyl-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV10 citations74
US4368200AJan 11, 1983
Heterocyclic derivatives of (4-phenyl-piperazine-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)-methyl-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV10 citations74
US4160841AJul 10, 1979
Heterocyclic derivatives of 1-(1,3-dioxolan-2-ylmethyl)-1H-imidazoles
JANSSEN PHARMACEUTICA NV13 citations74
US4861879AAug 29, 1989
[[4-[4-Phenyl-1-piperazinyl)phenoxymethyl]-1-3-dioxolan-2-yl]-methyl]-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV6 citations63
US4483865ANov 20, 1984
Antimicrobial imidazole derivatives
JANSSEN PHARMACEUTICA NV2 citations63
US4244964AJan 13, 1981
Heterocyclic derivatives of 1-(1,3-dioxolan-2-ylmethyl)-1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV4 citations63
US4229460AOct 21, 1980
Heterocyclic derivatives of 1-(1,3-dioxolan-2-ylmethyl)-1H-1,2,4-triazoles having antifungal and antibacterial properties
JANSSEN PHARMACEUTICA NV5 citations63
US4268680AMay 19, 1981
Heterocyclic derivatives of 1-(1,3-dioxolan-2-ylmethyl)-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV1 citations52
US4232034ANov 4, 1980
Heterocyclic derivatives of 1-(1,3-dioxolan-2-ylmethyl)-1H-imidazoles
JANSSEN PHARMACEUTICA NV1 citations52
US4229581AOct 21, 1980
Hydrazine carboxamide derivatives of 1-(1,3-dioxolan-2-ylmethyl)-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV0 citations52