Inventor · disambiguated record
Donald W. Graham
Also filed as: GRAHAM DONALD W
39 granted patents·3 pending applications·505 citations·filing 1976–2010
98Inventor score
Top patents by PatentIndex Score
42 records- 0192US6849636B2Triazole derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1MERCK & CO INC·Filed 2003·Granted Feb 1, 2005·52 cites·49 claims
- 0288US7625937B21H-benzo[F]indazol-5-YL derivatives as selective glucocorticoid receptor modulatorsMERCK & CO INC·Filed 2007·Granted Dec 1, 2009·11 cites·21 claims
- 0387US5147868AThienamycin renal peptidase inhibitorsMERCK & CO INC·Filed 1992·Granted Sep 15, 1992·36 cites·24 claims
- 0483US5595996A7-substituted 4-aza cholanic acid derivatives and their useMERCK & CO INC·Filed 1994·Granted Jan 21, 1997·33 cites·9 claims
- 0583US5516779A17β-substituted-6-azasteroid derivatives useful as 5α-reductase inhibitorsMERCK & CO INC·Filed 1994·Granted May 14, 1996·35 cites·9 claims
- 0682US5047420A1,3-diaryl cyclopentanes and derivatives thereof as PAF antagonistsMERCK & CO INC·Filed 1989·Granted Sep 10, 1991·18 cites·8 claims
- 0782US4173631A7-Methyl-8-methylamino-10-(1'-D-ribityl)isoalloxazineMERCK & CO INC·Filed 1978·Granted Nov 6, 1979·10 cites·7 claims
- 0880US5693809ASubstituted 4-aza-5α-androstan-ones as 5α-reductase inhibitorsMERCK & CO INC·Filed 1995·Granted Dec 2, 1997·37 cites·1 claims
- 0980US4816477AAntihypercholesterolemic β-lactonesMERCK & CO INC·Filed 1987·Granted Mar 28, 1989·15 cites·19 claims
- 1078US6090836ABenzisoxazole-derived antidiabetic compoundsMERCK & CO INC·Filed 1997·Granted Jul 18, 2000·24 cites·16 claims
- 1178US5510351ADelta-17 and delta-20 olefinic and saturated 17 beta-substituted 4-aza-5 alpha-androstan-ones as 5 alpha reductase inhibitors useful in the prevention and treatment of hyperandrogenic disordersMERCK & CO INC·Filed 1993·Granted Apr 23, 1996·25 cites·14 claims
- 1276US4806564AAntihypercholesterolemic beta-lactonesMERCK & CO INC·Filed 1987·Granted Feb 21, 1989·22 cites·22 claims
- 1375US5510485A17-ester, amide, and ketone derivatives of 3-oxo-4-azasteroids as 5A-reductase inhibitorsMERCK & CO INC·Filed 1994·Granted Apr 23, 1996·25 cites·3 claims
- 1475US4407802A6-Amidino-9-substituted benzyl purinesMERCK & CO INC·Filed 1981·Granted Oct 4, 1983·13 cites·6 claims
- 1574US8178546B2Diaryltriazoles as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1ASTER SUSAN D·Filed 2010·Granted May 15, 2012·4 cites·5 claims
- 1673US7282591B21h-benzo{f}indazol-5-yl derivatives as selective glucocorticoid receptor modulatorsMERCK & CO INC·Filed 2003·Granted Oct 16, 2007·5 cites·2 claims
- 1771US7411073B2Selective non-steroidal glucocorticoid receptor modulatorsMERCK & CO INC·Filed 2004·Granted Aug 12, 2008·5 cites·11 claims
- 1870US7504402B2Triazole derivatives as inhibitors of 11-β-hydroxysteroid dehydrogenase-1MERCK & CO INC·Filed 2004·Granted Mar 17, 2009·4 cites·9 claims
- 1970US4847271AAntihypercholesterolemic β-lactonesMERCK & CO INC·Filed 1987·Granted Jul 11, 1989·41 cites·26 claims
- 2069US7732432B217-carbamoyloxy cortisol derivatives as selective glucocorticoid receptor modulatorsMERCK SHARP & DOHME·Filed 2004·Granted Jun 8, 2010·4 cites·10 claims
- 2168US5710275A7β-substituted-4-aza-5α-androstan-3-ones as 5α-reductase inhibitorsMERCK & CO INC·Filed 1993·Granted Jan 20, 1998·22 cites·2 claims
- 2263US2009181994A1Triazole derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1MERCK & CO INC·Filed 2009·Application pending·0 cites
- 2358US5741795A16-substituted-6-aza-androsten-4-ene-3-ones as 5-α-reductase inhibitorsMERCK & CO INC·Filed 1996·Granted Apr 21, 1998·14 cites·13 claims
- 2454US5621104ASubstituted 3-phenanthridinone derivatives as 5-alpha-reductase inhibitorsMERCK & CO INC·Filed 1994·Granted Apr 15, 1997·4 cites·1 claims
- 2554US5438061A7-substituted-δ4-6-azasteroid derivatives as 5α-reductase inhibitorsMERCK & CO INC·Filed 1993·Granted Aug 1, 1995·9 cites·4 claims
- 2652US4752611AAnticoccidial 1,2,3-trazole compoundsMERCK & CO INC·Filed 1985·Granted Jun 21, 1988·3 cites·17 claims
- 2752US4079069A5-Deazariboflavin and its derivativesMERCK & CO INC·Filed 1977·Granted Mar 14, 1978·3 cites·3 claims
- 2848US4094976AAnticoccidial cyclicamino ethanols and esters thereofMERCK & CO INC·Filed 1976·Granted Jun 13, 1978·7 cites·15 claims
- 2947US7662846B2Selective spirocyclic glucocorticoid receptor modulatorsMERCK SHARP & DOHME·Filed 2004·Granted Feb 16, 2010·0 cites·5 claims
- 3047US5760045ADelta-17 and delta-20 olefinic and saturated 17β-substituted-4-aza-5α-androstan-3-ones as 5α-reductase inhibitors useful in the prevention and treatment of hyperandrogenic disordersMERCK & CO INC·Filed 1996·Granted Jun 2, 1998·6 cites·9 claims
- 3146US8026264B2Triazole derivatives as inhibitors of 11-β hydroxysteroid dehydrogenase-1MERCK SHARP & DOHME·Filed 2004·Granted Sep 27, 2011·0 cites·15 claims
- 3244US4091094A9-Azariboflavin and pharmaceutical composition containing sameMERCK & CO INC·Filed 1976·Granted May 23, 1978·1 cites·6 claims
- 3344US2008255216A1Diaryltriazoles as Inhibitors of 11-Beta-Hydroxysteroid Dehydrogenase-1ASTER SUSAN D·Filed 2005·Application pending·0 cites
- 3443US2005245588A1Octahydro-2-h-naphtho[1,2-f]indole-4-carboxamide derivatives as selective glucocorticoid receptor modulatorsALI AMJAD·Filed 2003·Application pending·0 cites
- 3542US5843953A7-substituted 4-aza cholanic acid derivatives and their useMERCK & CO INC·Filed 1995·Granted Dec 1, 1998·6 cites·8 claims
- 3639US7329683B211-β-hydroxysteroid dehydrogenase 1 inhibitors useful for the treatment of diabetes, obesity and dyslipidemiaMERCK & CO INC·Filed 2003·Granted Feb 12, 2008·0 cites·2 claims
- 3738US6048869ATricyclic compoundsMERCK & CO INC·Filed 1999·Granted Apr 11, 2000·3 cites·32 claims
- 3838US5886005A4-Aza-19-norandrostane derivativesMERCK & CO INC·Filed 1996·Granted Mar 23, 1999·3 cites·8 claims
- 3936US4406902ADipeptidase inhibitorsMERCK & CO INC·Filed 1981·Granted Sep 27, 1983·5 cites·12 claims
- 4032US4053602ACompositions for treating coccidiosis containing 5-deazariboflavin and its derivativesMERCK & CO INC·Filed 1976·Granted Oct 11, 1977·0 cites·11 claims
- 4130US5132463A1,3-diaryl cyclopentanes and derivatives thereof as PAF antagonistsMERCK & CO INC·Filed 1991·Granted Jul 21, 1992·0 cites·8 claims
- 4229US4290966AProcess for the preparation of traumatinMERCK & CO INC·Filed 1980·Granted Sep 22, 1981·0 cites·6 claims
Join the waitlist — get patent alerts
Get an alert when Donald W. Graham files or is granted a new patent.
We store only your email — no account needed. See our privacy policy.
Identity basis: PatentsView inventor disambiguation (2025Q4-odp release). How scoring works →