Inventor · disambiguated record
Josephus H. M. Lange
Also filed as: LANGE JOSEPHUS H · LANGE JOSEPHUS H M
27 granted patents·7 pending applications·193 citations·filing 1992–2011
95Inventor score
Top patents by PatentIndex Score
34 records- 0192US6476060B24,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activitySOLVAY PHARM BV·Filed 2001·Granted Nov 5, 2002·78 cites·24 claims
- 0287US6974810B24,5-Dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activitySOLVAY PHARM BV·Filed 2002·Granted Dec 13, 2005·31 cites·9 claims
- 0386US7524867B2Tetrasubstituted imidazole derivatives as cannabinoid CB1 receptor modulators with a high CB1/CB2 receptor subtype selectivitySOLVAY PHARM BV·Filed 2005·Granted Apr 28, 2009·10 cites·11 claims
- 0482US7528162B24,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activitySOLVAY PHARM BV·Filed 2002·Granted May 5, 2009·20 cites·16 claims
- 0581US7109216B21H-imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activitySOLVAY PHARM BV·Filed 2004·Granted Sep 19, 2006·14 cites·13 claims
- 0679US7319110B21H-1,2,4-triazole-3-carboxamide derivatives having cannabinoid-CB1 receptor agonistic, partial agonistic, inverse agonistic or antagonistic activitySOLVAY PHARM BV·Filed 2003·Granted Jan 15, 2008·14 cites·4 claims
- 0777US8138174B2Compounds with a combination of cannabinoid CB1 antagonism and serotonin reuptake inhibitionLANGE JOSEPHUS H M·Filed 2008·Granted Mar 20, 2012·2 cites·5 claims
- 0876US7786144B2Sulphur containing pyrazole derivatives as selective cannabinoid CB1 receptor antagonistsSOLVAY PHARM BV·Filed 2007·Granted Aug 31, 2010·2 cites·13 claims
- 0976US7608718B24,5-dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activitySOLVAY PHARM BV·Filed 2005·Granted Oct 27, 2009·2 cites·2 claims
- 1070US7186741B2Neurotensin active 2,3,diaryl-pyrazolidine derivativesSOLVAY PHARM BV·Filed 2003·Granted Mar 6, 2007·6 cites·4 claims
- 1167US8063062B2Compounds with a combination of cannabinoid-CB1 antagonism and acetylcholinesterase inhibitionLANGE JOSEPHUS H M·Filed 2007·Granted Nov 22, 2011·1 cites·11 claims
- 1260US7495108B2Imidazoline derivatives having CB1-antagonistic activitySOLVAY PHARM BV·Filed 2007·Granted Feb 24, 2009·0 cites·5 claims
- 1358US7928134B25-aryl-4,5-dihydro-(1H)-pyrazolines as cannabinoid CB1 receptor agonistsSOLVAY PHARM BV·Filed 2008·Granted Apr 19, 2011·0 cites·11 claims
- 1457US7342032B2Thiazole derivatives having CB1-antagonistic, agonistic or partial agonistic activitySOLVAY PHARMACEUTICALS INC·Filed 2003·Granted Mar 11, 2008·1 cites·9 claims
- 1555US7498348B21 H-imidazole derivatives as cannabinoid receptor modulatorsSOLVAY PHARM BV·Filed 2007·Granted Mar 3, 2009·0 cites·3 claims
- 1655US7173044B2Imidazoline derivatives having CB1-antagonistic activitySOLVAY PHARM BV·Filed 2005·Granted Feb 6, 2007·0 cites·7 claims
- 1753US7271189B21H-imidazole derivatives as cannabinoid receptor modulatorsSOLVAY PHARM BV·Filed 2004·Granted Sep 18, 2007·0 cites·9 claims
- 1853US2011137040A1Synthesis of 3,4-diaryl-4,5-dihydro-(h)-pyrazole-1-carboxamidine derivativesLANGE JOSEPHUS H M·Filed 2009·Application pending·0 cites
- 1951US8729101B21H-imidazole derivative having CB1, agonistic, CB1 partial agonistic or CB1 antagnistic activityKRUSE CORNELIS G·Filed 2008·Granted May 20, 2014·0 cites·6 claims
- 2049US6335326B1Benzisoxazole derivatives having d4-antagonistic activityDUPHAR INT RES·Filed 1999·Granted Jan 1, 2002·9 cites·13 claims
- 2147US2004235854A11H-imidazole derivatives having cb1 agonistic, cb1 partial agonistic or cb1 antagonistic activityFiled 2002·Application pending·0 cites
- 2245US2011160459A15-aryl-4,5-dihydro-(1h)-pyrazolines as cannabinoid cb1 receptor agonistsSOLVAY PHARM BV·Filed 2011·Application pending·0 cites
- 2344US8937184B21H-imidazole derivatives as cannabinoid CB2 receptor modulatorsLANGE JOSEPHUS H M·Filed 2006·Granted Jan 20, 2015·0 cites·8 claims
- 2444US8575148B2Spiro azepane-oxazolidinones as Kv1.3 potassium channel blockersSMID PIETER·Filed 2009·Granted Nov 5, 2013·0 cites·14 claims
- 2544US7745476B21,3,5-trisubstituted 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activitySOLVAY PHARM BV·Filed 2005·Granted Jun 29, 2010·0 cites·17 claims
- 2643US2007142362A14,5-Dihydro-(1H)-pyrazole derivatives as cannabinoid CB1 receptor modulatorsSOLVAY PHARM BV·Filed 2006·Application pending·0 cites
- 2743US2005065189A1Thiazole derivatives as cannabinoid receptor modulatorsSOLVAY PHARM BV·Filed 2004·Application pending·0 cites
- 2842US2011053983A1(5r)-1,5-diaryl-4,5-dihydro-1h-pyrazole-3-carboxamidine derivatives having cb1-antagonistic activityLANGE JOSEPHUS H M·Filed 2009·Application pending·0 cites
- 2941US2011172274A1Fluoro-substituted 3,4-diaryl-4,5-dihydro-1h-pyrazole-1-carboxamidine derivatives having cb1-antagonistic activityLANGE JOSEPHUS H M·Filed 2009·Application pending·0 cites
- 3039US8461184B2Sulphur containing pyrazole derivatives as selective cannabinoid CB1 receptor antagonistsLANGE JOSEPHUS H M·Filed 2010·Granted Jun 11, 2013·0 cites·5 claims
- 3137US8410135B24,5 dihydro-(1H)-pyrazole derivatives as cannabinoid CB1 receptor modulatorsLANGE JOSEPHUS H M·Filed 2008·Granted Apr 2, 2013·0 cites·14 claims
- 3237US5281595AAlkylenedioxyphenyl ether derivatives having anti-ischaemic, memory enhancing and anti-convulsive activityDUPHAR INT RES·Filed 1992·Granted Jan 25, 1994·2 cites·6 claims
- 3332US9422244B2Synthesis of substituted pyrazoline carboxamidine derivativesVAN LOEVEZIJN ARNOLD·Filed 2011·Granted Aug 23, 2016·0 cites·6 claims
- 3428US5356891APhenylalkyl amine derivatives having anti-ischaemic activityWITIAK DONALD T·Filed 1992·Granted Oct 18, 1994·1 cites·3 claims
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Identity basis: PatentsView inventor disambiguation (2025Q4-odp release). How scoring works →