Inventor · disambiguated record
Robert W. Desimone
Also filed as: DESIMONE ROBERT · DESIMONE ROBERT W
34 granted patents·13 pending applications·1,025 citations·filing 1995–2008
98Inventor score
Files withNEUROGEN CORP28CGI PHARMACEUTICALS INC8CURRIE KEVIN S5BAKTHAVATCHALAM RAJAGOPAL1CELLULAR GENOMICS INC1
Top patents by PatentIndex Score
47 records- 0196US7393848B2Certain heterocyclic substituted imidazo[1,2-A]pyrazin-8-ylamines and methods of inhibition of Bruton's tyrosine kinase by such compoundsCGI PHARMACEUTICALS INC·Filed 2004·Granted Jul 1, 2008·67 cites·50 claims
- 0295US7160885B2Certain 6, 8-(heteroaryl or aryl) disubstituted imidazo[1,2-a]pyrazines as modulators of Hsp90 complex activityCGI PHARMACEUTICALS INC·Filed 2004·Granted Jan 9, 2007·77 cites·41 claims
- 0395US6723730B2Capsaicin receptor ligandsNEUROGEN CORP·Filed 2001·Granted Apr 20, 2004·105 cites·185 claims
- 0495US6271241B1Cycloalkyl and aryl fused aminoalkyl-imidazole derivatives: modulators and GLP-1 receptorsNEUROGEN CORP·Filed 2000·Granted Aug 7, 2001·65 cites·51 claims
- 0594US6380210B1Heteroaryl fused aminoalkyl-imidazole derivatives: selective modulators of GABAa receptorsNEUROGEN CORP·Filed 2000·Granted Apr 30, 2002·37 cites·12 claims
- 0693US7405295B2Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of Bruton's tyrosine kinase by such compoundsCGI PHARMACEUTICALS INC·Filed 2004·Granted Jul 29, 2008·98 cites·59 claims
- 0793US6399604B1Substituted 4-OXO-napthyridine-3-carboxamides; GABA brain receptor ligandsNEUROGEN CORP·Filed 2000·Granted Jun 4, 2002·33 cites·107 claims
- 0892US7189723B2Certain 8-heteroaryl-6-phenyl-imidazo[1,2-a]pyrazines as modulators of kinase activityCGI PHARMACEUTICALS INC·Filed 2004·Granted Mar 13, 2007·48 cites·35 claims
- 0992US6646124B2Substituted 4-oxo-napthyridine-3-carboxamides: GABA brain receptor ligandsNEUROGEN CORP·Filed 2002·Granted Nov 11, 2003·24 cites·8 claims
- 1092US6143760ASubstituted 4-oxo-napthyridine-3-carboxamides: GABA brain receptor ligandsNEUROGEN CORP·Filed 1998·Granted Nov 7, 2000·47 cites·110 claims
- 1191US7312341B26-aryl-imidazo[1,2-a] pyrazin-8-ylamines, method of making, and method of use thereofCGI PHARMACEUTICALS INC·Filed 2003·Granted Dec 25, 2007·50 cites·82 claims
- 1289US6919340B2Imidazo[1,2-a]pyrazin-8-ylamines, method of making, and method of use thereofCELLULAR GENOMICS INC·Filed 2003·Granted Jul 19, 2005·54 cites·34 claims
- 1388US7259164B2Certain substituted imidazo[1,2-a]pyrazines, as modulators of kinase activityCGI PHARMACEUTICALS INC·Filed 2004·Granted Aug 21, 2007·46 cites·42 claims
- 1487US7015227B2Certain amino-substituted monocycles as kinase modulatorsCGI PHARMACEUTICALS INC·Filed 2003·Granted Mar 21, 2006·21 cites·6 claims
- 1584US6316617B1Certain amido-and amino-substituted benzylamine derivatives; a new class of Neuropeptide Y1 specific ligandsNEUROGEN CORP·Filed 2000·Granted Nov 13, 2001·17 cites·16 claims
- 1683US7160879B2Melanin concentrating hormone receptor ligands: substituted 2-(4-benzyl-piperazin-1-ylmethyl)- and 2-(4-benzyl-diazepan-1-ylmethyl)-1H-benzoimidazole analoguesNEUROGEN CORP·Filed 2003·Granted Jan 9, 2007·26 cites·24 claims
- 1783US6482844B11-benzylimidazole derivativesNEUROGEN CORP·Filed 2001·Granted Nov 19, 2002·13 cites·22 claims
- 1882US7348326B2Heteroaryl fused aminoalkyl imidazole derivatives: selective modulators of GABAa receptorsNEUROGEN CORP·Filed 2005·Granted Mar 25, 2008·6 cites·6 claims
- 1981US6448259B1Substituted cycloalkyl-4-oxonicotinic carboxamides; GABA brain receptor ligandsNEUROGEN CORP·Filed 2000·Granted Sep 10, 2002·13 cites·19 claims
- 2081US5637724ASubstituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligandsNEUROGEN CORP·Filed 1995·Granted Jun 10, 1997·21 cites·17 claims
- 2180US6358949B1Aryl and hetroaryl fused aminoalkyl-imidazole derivatives: selective modulators of bradykinin B2 receptorsNEUROGEN CORP·Filed 2000·Granted Mar 19, 2002·10 cites·56 claims
- 2279US6127395ASubstituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligandsNEUROGEN CORP·Filed 1999·Granted Oct 3, 2000·18 cites·11 claims
- 2378US5637725ASubstituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligandsNEUROGEN CORP·Filed 1995·Granted Jun 10, 1997·16 cites·15 claims
- 2477US5936095ASubstituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligandsNEUROGEN CORP·Filed 1997·Granted Aug 10, 1999·15 cites·3 claims
- 2576US5849927ASubstituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligandsNEUROGEN CORP·Filed 1997·Granted Dec 15, 1998·16 cites·1 claims
- 2675US6509366B2Substituted imidazoles as selective modulators of Bradykinin B2 receptorsNEUROGEN CORP·Filed 2001·Granted Jan 21, 2003·7 cites·46 claims
- 2775US6133265ACertain amido- and amino- substituted benzylamine derivatives; a new class of neuropeptide Y1 specific ligandsNEUROGEN CORP·Filed 1997·Granted Oct 17, 2000·33 cites·20 claims
- 2869US6972293B2Heteroaryl fused aminoalkyl-imidazole derivatives: selective modulators of GABAa receptorsNEUROGEN CORP·Filed 2003·Granted Dec 6, 2005·3 cites·10 claims
- 2968US6627624B1Aryl fused aminoalkyl-imidazole derivatives: selective modulators of GABAa receptorsNEUROGEN CORP·Filed 2000·Granted Sep 30, 2003·4 cites·33 claims
- 3066US6906075B2Melanin concentrating hormone receptor ligands: substituted benzoimidazole analoguesNEUROGEN CORP·Filed 2003·Granted Jun 14, 2005·3 cites·16 claims
- 3165US6194427B1Substituted cycloalkyl-4-Oxonicotinic carboxamides; gaba brain receptor ligandsNEUROGEN CORP·Filed 1999·Granted Feb 27, 2001·19 cites·22 claims
- 3265US6156898ASubstituted 1,4-dihydro-4-oxonicotinic carboxamides; GABA brain receptor ligandsNEUROGEN CORP·Filed 1999·Granted Dec 5, 2000·13 cites·38 claims
- 3358US2008182849A1Certain Heterocyclic Substituted Imidazo[1,2-A]Pyrazin-8-Ylamines And Methods Of Inhibition Of Bruton's Tyrosine Kinase By Such CompoundsCURRIE KEVIN S·Filed 2008·Application pending·0 cites
- 3456US7241765B2Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analoguesNEUROGEN CORP·Filed 2006·Granted Jul 10, 2007·0 cites·44 claims
- 3555US2004176443A1Capsaicin receptor ligandsNEUROGEN CORP·Filed 2004·Application pending·0 cites
- 3654US2009082362A1Use of capsaicin receptor antagonists to treat symptoms of tear gas exposureBAKTHAVATCHALAM RAJAGOPAL·Filed 2008·Application pending·0 cites
- 3751US2011177011A1Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of bruton's tyrosine kinase by such compoundsCURRIE KEVIN S·Filed 2008·Application pending·0 cites
- 3849US2003092912A1Heteroaryl fused aminoalkyl-imidazole derivatives: selective modulators of GABAa ReceptorsNEUROGEN CORP A CORP OF THE ST·Filed 2002·Application pending·0 cites
- 3947US2002082425A1Aryl and heteroaryl fused aminoalkyl-imidazole derivativesNEUROGEN CORP·Filed 2001·Application pending·0 cites
- 4047US2003229076A1Substituted imidazoles as selective modulators of bradykinin B2 receptorsFiled 2002·Application pending·0 cites
- 4145US2005288295A1Certain imidazo[1,2-a]pyrazin-8-ylamines, method of making, and method of use thereofCURRIE KEVIN S·Filed 2004·Application pending·0 cites
- 4245US2002151550A1Aryl and heteroaryl fused aminoalkyl-imidazole derivatives: selective modulators of bradykinin B2 receptorsNEUROGEN CORP·Filed 2002·Application pending·0 cites
- 4344US7625931B2Certain substituted diphenyl ureas, as modulators of kinase activityCGI PHARMACEUTICALS INC·Filed 2006·Granted Dec 1, 2009·0 cites·46 claims
- 4443US2006199846A1Certain substituted ureas as modulators of kinase activityMITCHELL SCOTT A·Filed 2006·Application pending·0 cites
- 4542US2004082627A1Certain aromatic monocycles as kinase modulatorsFiled 2003·Application pending·0 cites
- 4640US2006183746A1Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of Bruton's tyrosine kinase by such compoundsCURRIE KEVIN S·Filed 2005·Application pending·0 cites
- 4740US2006178367A1Certain imidazo[1,2-a]pyrazin-8-ylamines, method of making, and method of use thereofCURRIE KEVIN S·Filed 2005·Application pending·0 cites
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Identity basis: PatentsView inventor disambiguation (2025Q4-odp release). How scoring works →