US2003134866A1PendingUtilityA1
Antipsychotic pharmaceutical composition
Assignee: PHARMACEUTICAL IND TECH & DEVPriority: Jan 4, 2002Filed: May 13, 2002Published: Jul 17, 2003
Est. expiryJan 4, 2022(expired)· nominal 20-yr term from priority
A61K 31/519A61P 25/18
54
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Claims
Abstract
A pharmaceutical composition useful in treating psychosis contains a therapeutically effective amount of 2-[piperidinyl]methyl-2,3-dihydroimidazo[1,2-c]quinazolin-5(6H)-one as an active ingredient.
Claims
exact text as granted — not AI-modifiedWhat is claimed is:
1 . An antipsychotic pharmaceutical composition comprising an antipsychosis therapeutically effective amount of
2-[piperidinyl]methyl-2,3-dihydroimidazo[1,2-c]quinazolin-5(6H)-one having the following formula or a pharmaceutically acceptable salt thereof, as an active ingredient, in combination with a pharmaceutically acceptable carrier or diluent for the active ingredient: wherein R 1 is C1-C6 alkylene, carbonyl, C1-C6 alkylene carbonyl or carbonyloxy; and R 2 is hydrogen, C1-C6 alkyl, C1-C6 alkoxy or halogen.
2 . The antipsychotic pharmaceutical composition according to claim 1 , wherein R 1 is methylene or carbonyl.
3 . The antipsychotic pharmaceutical composition, wherein R 1 is carbonyl.
4 . The antipsychotic pharmaceutical composition according to claim 1 , wherein R 2 is hydrogen or halogen.
5 . The antipsychotic pharmaceutical composition according to claim 2 , wherein R 2 is hydrogen or halogen.
6 . The antipsychotic pharmaceutical composition according to claim 3 , wherein R 2 is halogen.
7 . The antipsychotic pharmaceutical composition according to claim 6 , wherein R 2 is fluorine.
8 . The antipsychotic pharmaceutical composition according to claim 6 , which is orally administered.Cited by (0)
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