US2005288327A1PendingUtilityA1

Small molecule inhibitors of HER2 expression

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Assignee: UESUGI MOTONARIPriority: May 14, 2002Filed: Jul 20, 2005Published: Dec 29, 2005
Est. expiryMay 14, 2022(expired)· nominal 20-yr term from priority
Inventors:Motonari UesugiShinichi Asada
C07D 401/14C07D 211/26A61P 35/00
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Claims

Abstract

Peptide mimetic small molecule inhibitors of Sur-2 are provided having the general formula:

Claims

exact text as granted — not AI-modified
1 - 4 . (canceled)  
     
     
         5 . A compound of the formula:  
       
         
           
           
               
               
           
         
         wherein the R 1  is selected from the group of β blockers consisting of propanolol, indenolol, carpindolol, bupranolol, and mepindolol;  
         and pharmaceutically acceptable salts thereof.  
       
     
     
         6 . The compound of  claim 5  wherein the β blocker substituent group is propanolol.  
     
     
         7 - 19 . (canceled)

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