US2006264626A1PendingUtilityA1

INHIBITORS OF FACTOR Xa AND OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION CASCADE

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Assignee: WARNER LAMBERT COPriority: Nov 29, 2001Filed: Aug 2, 2006Published: Nov 23, 2006
Est. expiryNov 29, 2021(expired)· nominal 20-yr term from priority
Inventors:Agustin Casimiro-GarciaJeremy John EdmundsKevin James FilipskiJeffrey Thomas Kohrt
A61P 7/02A61P 9/10A61P 7/00A61P 3/10A61P 9/04A61P 35/00C07D 207/16C07D 207/24C07D 403/12C07D 401/04C07D 401/12C07D 233/56C07D 249/08C07D 213/64C07D 231/12C07D 231/06C07D 207/27C07D 207/20C07D 401/14C07D 207/26C07D 207/22C07D 237/14C07D 413/12C07D 211/76
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Claims

Abstract

Compounds useful as intermediates for synthesis of compounds of Formula (1): wherein A, B, C, G, and W 1 have any of the values defined in the specification.

Claims

exact text as granted — not AI-modified
1 . A compound selected from: 
 1-(4-Amino-3-fluorophenyl)piperidin-2-one,    2-Fluoro-4-(3-methylpyrazol-1-yl)phenylamine,    2-Fluoro-4-(5-methylpyrazol-1-yl)phenylamine,    1-(4-Amino-3-fluorophenyl)-1H-pyridin-2-one,    6′-Amino-3,4,5,6-tetrahydro-[1,3′]bipyridinyl-2-one,    6′-Amino-[1,3′]bipyridinyl-2-one,    2-(4-Amino-3-fluorophenyl)-2H-pyridazin-3-one,    1-(4-Aminophenyl)-3-methyl-1H-pyridin-2-one, and    1-(4-Amino-3-fluorophenyl)-5-methyl-1H-pyridin-2-one.    
     
     
         2 . A compound according to  claim 1  that is: 
 1-(4-Amino-3-fluorophenyl)-1H-pyridin-2-one.

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