US2010160620A1PendingUtilityA1

N-pyrazole a2a receptor agonists

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Assignee: GILEAD PALO ALTO INCPriority: Jun 22, 1999Filed: Dec 14, 2009Published: Jun 24, 2010
Est. expiryJun 22, 2019(expired)· nominal 20-yr term from priority
Inventors:Jeff ZablockiElfatih ElzeinVenkata P. PalleLuiz Belardinelli
A61P 7/02A61P 9/10A61P 7/00A61P 9/08A61P 9/00A61P 43/00A61P 29/00C07D 473/34C07H 19/16
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Abstract

2-adenosine N-pyrazole compounds having the following formula: and methods for using the compounds as A2A receptor agonists to stimulate mammalian coronary vasodilatation for therapeutic purposes and for purposes of imaging the heart.

Claims

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1 .- 7 . (canceled) 
     
     
         8 . A compound having the following formula: 
       
         
           
           
               
               
           
         
         namely (1-{9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-6-aminopurin-2-yl}pyrazol-4-yl)-N-methylcarboxamide.

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