US2010249145A1PendingUtilityA1

Inhibitors of VEGF Receptor and HGF Receptor Signaling

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Assignee: METHYLGENE INCPriority: May 20, 2005Filed: Mar 25, 2010Published: Sep 30, 2010
Est. expiryMay 20, 2025(expired)· nominal 20-yr term from priority
A61P 43/00C07D 495/04A61P 35/00A61P 9/00A61K 31/519A61K 31/522A61K 31/4365
41
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Claims

Abstract

The invention relates to the inhibition of VEGF receptor signaling and HGF receptor signaling. The invention provides compounds and methods for inhibiting VEGF receptor signaling and HGF receptor signaling. The invention also provides compositions and methods for treating cell proliferative diseases and conditions

Claims

exact text as granted — not AI-modified
1 . A hydrate or solvate of a compound selected from the group consisting of 
       
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
         
           
           
               
               
           
         
       
     
     
         2 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         3 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         4 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         5 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         6 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         7 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         8 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         9 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         10 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         11 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         12 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         13 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         14 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         15 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         16 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         17 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         18 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         19 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         20 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         21 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         22 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         23 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         24 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         25 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         26 . The hydrate or solvate according to  claim 1 , wherein the compound has the structure 
       
         
           
           
               
               
           
         
       
     
     
         27 . A pharmaceutical composition comprising a hydrate or solvate according to  claim 1  and a pharmaceutically acceptable carrier. 
     
     
         28 . A method of inhibiting VEGF receptor signaling and HGF receptor signaling in an animal, the method comprising administering to the animal a receptor inhibiting amount of a hydrate or solvate according to  claim 1 , or a composition thereof. 
     
     
         29 . A method of treating an angiogenesis-mediated cell proliferative disease in a patient or inhibiting solid tumor growth in a patient, the method comprising administering to the patient in need thereof an effective therapeutical amount of a hydrate or solvate according to  claim 1  or a composition thereof.

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