US2012071496A1PendingUtilityA1
Aminopyrimidinamides As Pest Control Agents
Est. expiryFeb 17, 2029(~2.6 yrs left)· nominal 20-yr term from priority
Inventors:Simon MaechlingArnd VoersteEva-Maria FrankenAngela BeckerUlrich GörgensMazen Es-SayedMarkus HeilGraham HolmwoodJohannes-Rudolf JansenOtto SchallnerUlrich Ebbinghaus-KintscherPeter LümmenSilvia Cerezo-GalvezSachio KudoTakashi HashihayataEiichi ShimojoTeruyuki IchiharaMasashi AtakaKatsuhiko Shibuya
A61P 33/00A61P 33/14C07D 401/12C07D 403/12C07D 239/48A01N 43/54
38
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Claims
Abstract
The present application relates to novel aminopyrimidinamides, to processes for their preparation and to their use for controlling animal pests, especially arthropods, in particular insects.
Claims
exact text as granted — not AI-modified1 . Compounds of the formula (I)
in which
R 1 represents a radical from the group consisting of hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, cyanoalkyl, cycloalkyl, halocycloalkyl, cycloalkenyl, halocycloalkenyl, hydroxyalkyl, alkoxyalkyl, haloalkoxyalkyl, alkoxyhaloalkyl, alkylcarbonylalkyl, alkoxycarbonylalkyl, alkylsulphanylalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, haloalkylsulphanylalkyl, haloalkylsulphinylalkyl, haloalkylsulphonylalkyl, halocycloalkylalkyl, cycloalkylalkyl and in each case optionally substituted phenyl, naphthyl, phenylalkyl, heteroaryl, heteroarylalkyl, heterocyclyl and heterocyclylalkyl.
R 2 represents a radical from the group consisting of hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, cyanoalkyl, cycloalkyl, halocycloalkyl, cycloalkenyl, halocycloalkenyl, hydroxyalkyl, alkoxyalkyl, haloalkoxyalkyl, alkoxyhaloalkyl, alkylcarbonylalkyl, alkoxycarbonylalkyl, alkylsulphanylalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, haloalkylsulphanylalkyl, haloalkylsulphinylalkyl, haloalkylsulphonylalkyl, cycloalkylalkyl and in each case optionally substituted phenyl, naphthyl, phenylalkyl, heteroaryl, heteroarylalkyl, heterocyclyl and heterocyclylalkyl,
R 3 represents a radical from the group consisting of hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, cyanoalkyl, cycloalkyl, halocycloalkyl, cycloalkenyl, halocycloalkenyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, haloalkoxyalkyl, alkoxyhaloalkyl, alkylcarbonylalkyl, alkoxycarbonylalkyl, alkylsulphanylalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, haloalkylsulphanylalkyl, haloalkylsulphinylalkyl, haloalkylsulphonylalkyl, cycloalkylalkyl and in each case optionally substituted phenyl, naphthyl, phenylalkyl, heteroaryl, heteroarylalkyl, heterocyclyl and hererocyclylalkyl,
R 4 represents a radical from the group consisting of in each case optionally substituted phenyl, naphthyl, heteroaryl, heteroarylalkyl, heterocyclyl and heterocyclylalkyl,
R 5 represents a radical from the group consisting of hydrogen, halogen, cyano and in each case optionally substituted alkyl, cycloalkyl, phenyl, naphthyl, heteroaryl, heteroarylalkyl, heterocyclyl and heterocyclylalkyl,
R 6 represents a radical from the group consisting of hydrogen, halogen, alkyl, haloalkyl, cyanoalkyl, alkoxyalkyl, alkylcarbonyl, haloalkylcarbonyl, cycloalkyl, halocycloalkyl, cycloalkylalkyl, alkylsulphonyl, alkenyl, alkynyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, alkoxycarbonylalkyl; optionally substituted phenyl, optionally substituted naphthyl, optionally substituted phenylalkyl, optionally substituted heterocyclylalkyl, optionally substituted heteroarylalkyl and optionally substituted phenylcarbonyl and
X represents oxygen or sulphur.
2 . Composition, characterized in that it comprises at least one compound of the formula (I) according to claim 1 and customary extenders and/or surfactants.
3 . Method for controlling pests, characterized in that a compound of the formula (I) according to claim 1 or a composition according to claim 2 is allowed to act on the pests and/or their habitat.
4 . Use of compounds of the formula (I) according to claim 1 or of compositions according to claim 2 for controlling pests.
5 . Pharmaceutical compositions comprising at least one compound according to claim 1 .
6 . Use of at least one compound according to claim 1 for preparing pharmaceutical compositions for controlling parasites on animals.Cited by (0)
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