US2013158091A1PendingUtilityA1
Polymorphs of saxagliptin hydrochloride and processes for preparing them
Est. expiryOct 4, 2030(~4.2 yrs left)· nominal 20-yr term from priority
A61P 3/08A61P 3/00A61K 31/403C07D 209/52
38
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Abstract
The invention provides polymorphs of Saxagliptin hydrochloride, processes for preparing polymorphs of Saxagliptin hydrochloride, and pharmaceutical compositions of polymorphs of Saxagliptin hydrochloride.
Claims
exact text as granted — not AI-modified1 - 18 . (canceled)
19 . Amorphous Saxagliptin hydrochloride.
20 . The amorphous Saxagliptin hydrochloride of claim 19 , characterized by an X-ray powder diffraction pattern substantially as depicted in FIG. 17 .
21 . A pharmaceutical composition comprising the amorphous Saxagliptin hydrochloride according to any one of claims 19 and 20 , and at least one pharmaceutically acceptable excipient.
22 . A method of treating a patient suffering from type 2 diabetes, comprising administering a pharmaceutical composition according to claim 21 .Cited by (0)
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