US2013195782A1PendingUtilityA1

Novel Glycine Derivative Capable Of Inhibiting Melanin Formation And Composition Using The Same

Assignee: HSU NAI-HSUANPriority: Oct 22, 2010Filed: Oct 22, 2010Published: Aug 1, 2013
Est. expiryOct 22, 2030(~4.2 yrs left)· nominal 20-yr term from priority
A61K 8/44C07C 233/47A61Q 19/08C07C 237/22A61Q 19/02A61P 17/00A61K 8/30A61K 31/198
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Claims

Abstract

The invention provides a glycine derivative, having a structure shown in the following general equation (I): wherein R 1 represents a C1˜C4 alkyl group; R 2 represents a hydrogen atom or a methyl group; and n represents an integer of 1˜6.

Claims

exact text as granted — not AI-modified
What is claimed is: 
     
         1 . A glycine derivative capable of inhibiting melanin formation, having a structure shown in the following general equation (I): 
       
         
           
           
               
               
           
         
         wherein R 1  represents a C1˜C4 alkyl group; R 2  represents a hydrogen atom or a methyl group; and n represents an integer of 1˜6. 
       
     
     
         2 . The glycine derivative according to  claim 1 , wherein the glycine derivative is 3(2-acetylamino-acetylamino)-propionic acid having a structure shown in the following equation (II): 
       
         
           
           
               
               
           
         
       
     
     
         3 . The glycine derivative according to  claim 1 , wherein the glycine derivative is 4-(2-Acetylamino-acetylamino)-butyric acid having a structure shown in the following equation (III): 
       
         
           
           
               
               
           
         
       
     
     
         4 . The glycine derivative according to  claim 1 , wherein the glycine derivative is [(2-Acetylamino-acetyl)-methyl-amino]-acetic acid having a structure shown in the following general equation (IV): 
       
         
           
           
               
               
           
         
       
     
     
         5 . The glycine derivative according to  claim 1 , wherein a solution or a buffer solution containing the glycine derivative with addition amount of 0.05˜10 wt % (weight ratio) has light transmittance more than or equal to 97% in the wavelength range of 420˜500 nm. 
     
     
         6 . The glycine derivative according to  claim 5 , wherein the buffer solution comprises citric acid and salts thereof. 
     
     
         7 . The glycine derivative according to  claim 5 , wherein solution or the buffer solution containing the glycine derivative with addition amount of 0.05˜10 wt % (weight ratio) has light transmittance more than or equal to 98% at the specific wavelength 440 nm. 
     
     
         8 . A whitening composition, comprising:
 a glycine derivative with addition amount of 0.05˜10 wt % (weight ratio) wherein the glycine derivative has a function of inhibiting melanin formation and has a structure shown in the following general equation (I):   
       
         
           
           
               
               
           
         
         wherein R 1  represents a C1˜C4 alkyl group; R 2  represents a hydrogen atom or a methyl group; and n represents an integer of 1˜6. 
       
     
     
         9 . The composition according to  claim 8 , wherein the composition comprises the glycine derivative with addition amount of 0.1˜2 wt % (weight ratio) and has a function of inhibiting melanin formation. 
     
     
         10 . The composition according to  claim 8 , wherein the glycine derivative is 3(2-acetylamino-acetylamino)-propionic acid having a structure shown in the following general equation (II): 
       
         
           
           
               
               
           
         
       
     
     
         11 . The composition according to  claim 8 , wherein the glycine derivative is 4-(2-Acetylamino-acetylamino)-butyric acid having a structure shown in the following general equation (III): 
       
         
           
           
               
               
           
         
       
     
     
         12 . The composition according to  claim 8 , wherein the glycine derivative is [(2-Acetylamino-acetyl)-methyl-amino]-acetic acid having a structure shown in the following equation (IV):

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