US2017304403A1PendingUtilityA1
METHOD FOR INHIBITING INFLAMMATION and PRO-INFLAMMATORY CYTOKINE/CHEMOKINE EXPRESSION USING A GHRELIN ANALOGUE

Assignee: IPSEN PHARMA SASPriority: Aug 8, 2007Filed: Jun 29, 2017Published: Oct 26, 2017
Est. expiryAug 8, 2027(~1.1 yrs left)· nominal 20-yr term from priority
Inventors:Zheng Xin Dong John E. Taylor Rakesh Datta Michael Dewitt Culler
A61P 5/14A61P 3/06A61P 37/00A61P 37/02A61P 37/08A61P 43/00A61P 37/06A61P 3/10A61P 39/02A61P 35/04A61P 9/14A61P 9/10A61P 33/04A61P 31/22A61P 33/02A61P 33/06A61P 29/00A61P 25/08A61P 31/04A61P 31/14A61P 35/02A61P 35/00A61P 25/28A61P 31/18A61P 31/16A61P 31/12A61P 31/00A61P 31/10A61P 31/06A61P 31/20A61P 33/12A61P 25/00A61P 11/06A61P 17/00A61P 17/14A61P 1/18A61P 1/04A61P 17/02A61P 17/16A61P 1/00A61P 1/16A61P 19/02A61P 1/14A61K 38/05C07K 7/06A61K 38/22A61K 38/25A61K 38/06Y02A50/30
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Abstract

The present invention provides a method of ameliorating inflammation, inhibiting proinflammatory cytokine and/or chemokine expression and treating various diseases and/or conditions incidental to the onset of inflammation, in a subject in need of treatment for such conditions, by administering select analogues of native hGhrelin.
Claims

exact text as granted — not AI-modified
1 . A method of limiting myocardial damage during an acute myocardial infarction in a subject in need thereof which comprises administering to said subject an effective amount of a peptidyl analogue of ghrelin, a prodrug thereof, or a pharmaceutically acceptable salt thereof wherein said analogue or said prodrug thereof is selected from the group consisting of:
 (Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 6)   (Aib 2 , A6c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 7)   (A6c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 8)   (Aib 2,6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 9)   (Aib 2 , A5c 12 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 10)   (Aib 2 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 11)   (Aib 2 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 12)   (Aib 2 , Act 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 9)   (Aib 2 , 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Aib 2 , Dmt 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Aib 2 , Thz 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (A5c 2 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 15)   (Act 2 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 15)   (Aib 2 , A5c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 7)   (Aib 2 , A6c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 7)   (Aib 2,5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 7)   (Aib 2 , hLeu 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 7)   (Aib 2 , Cha 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 7)   (Aib 2,6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 9)   (Aib 2 ,Act 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 9)   (Aib 2 , Thr 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 9)   (Aib 2 , Abu 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 9)   (Aib 2 , 4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Aib 2 ,Thz 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Aib 2 , Pip 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Aib 2 , Dhp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Aib 2 , Ktp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Aib 2,8 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 16)   (Aib 2 , 2-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Aib 2 , 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Aib 2 , 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Aib 2 , Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Aib 2 , 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Aib 2 , 2-Fua 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Aib 2 , Apc 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Aib 2,9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Aib 2,10 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 17)   (Aib 2 , Tic 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Aib 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 18)   (A5c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 8)   (A6c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 8)   (Act 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 18)   (3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (Dmt 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 20)   (Thz 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 20)   (Aib 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 8)   (hLeu 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 8)   (Cha 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 8)   (Thr 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 18)   (Abu 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 18)   (4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 20)   (Pip 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 20)   (Dhp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 20)   (Ktp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 20)   (Aib 8 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 21)   (2-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (2-Fua 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (Apc 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (Aib 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (Aib 10 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 22)   (Aib 2 , Dap 3 (octanesulfonyl), A6c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 23)   (Dap 3 (octanesulfonyl), A6c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 24)   (Aib 2,6 , Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 25)   (Aib 2 , Dap 3 (octanesulfonyl), A5c 12 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 26)   (Aib 2 , Dap 3 (octanesulfonyl), A5c 12 ,Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 27)   (Aib 2 , Dap 3 (octanesulfonyl), A5c 12 ,Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 28)   (Aib 2 , Dap 3 (octanesulfonyl), Act 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 25)   (Aib 2 , Dap 3 (octanesulfonyl), 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 29)   (Aib 2 , Dap 3 (octanesulfonyl), Dmt 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 30)   (Aib 2 , Dap 3 (octanesulfonyl), Thz 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 30)   (A5c 2 , Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 31)   (Acte, Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 31)   (Aib 2 , Dap 3 (octanesulfonyl), A5c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 32)   (Aib 2,5 , Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 32)   (Aib 2 , Dap 3 (octanesulfonyl), hLeu 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 32)   (Aib 2 , Dap 3 (octanesulfonyl), Cha 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 32)   (Aib 2,6 , Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 25)   (Aib 2 , Dap 3 (octanesulfonyl), Thr 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 25)   (Aib 2 , Dap 3 (octanesulfonyl), Abu 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 25)   (Aib 2 , Dap 3 (octanesulfonyl), 4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 30)   (Aib 2 , Dap 3 (octanesulfonyl), Pip 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 30)   (Aib 2 , Dap 3 (octanesulfonyl), Dhp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 30)   (Aib 2 , Dap 3 (octanesulfonyl), Ktp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 30)   (Aib 2,8 , Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 33)   (Aib 2 , Dap 3 (octanesulfonyl), 2-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 29)   (Aib 2 , Dap 3 (octanesulfonyl), 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 29)   (Aib 2 , Dap 3 (octanesulfonyl), 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 29)   (Aib 2 , Dap 3 (octanesulfonyl), Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 29)   (Aib 2 , Dap 3 (octanesulfonyl), 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 29)   (Aib 2 , Dap 3 (octanesulfonyl), 2-Fua 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 29)   (Aib 2 , Dap 3 (octanesulfonyl), Apc 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 29)   (Aib 2,9 , Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 29)   (Aib 2,10 , Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 34)   (Dap 3 (octanesulfonyl), A6c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 24)   (Dap 3 (octanesulfonyl), Aib 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 35)   (Dap 3 (octanesulfonyl), A5c 12 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 36)   (Dap 3 (octanesulfonyl), A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 37)   (Dap 3 (octanesulfonyl), A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 38)   (Dap 3 (octanesulfonyl), Act 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 35)   (Dap 3 (octanesulfonyl), 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 39)   (Dap 3 (octanesulfonyl), Dmt 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 40)   (Dap 3 (octanesulfonyl), Thz 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 40)   (Dap 3 (octanesulfonyl), A5c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 24)   (Dap 3 (octanesulfonyl), Aib 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 24)   (Dap 3 (octanesulfonyl), hLeu 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 24)   (Dap 3 (octanesulfonyl), Cha 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 24)   (Dap 3 (octanesulfonyl), Thr 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 35)   (Dap 3 (octanesulfonyl), Abu 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 35)   (Dap 3 (octanesulfonyl), 4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 40)   (Dap 3 (octanesulfonyl), Pip 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 40)   (Dap 3 (octanesulfonyl), Dhp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 40)   (Dap 3 (octanesulfonyl), Ktp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 40)   (Dap 3 (octanesulfonyl), Aib 8 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 41)   (Dap 3 (octanesulfonyl), 2-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 39)   (Dap 3 (octanesulfonyl), 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 39)   (Dap 3 (octanesulfonyl), 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 39)   (Dap 3 (octanesulfonyl), Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 39)   (Dap 3 (octanesulfonyl), 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 39)   (Dap 3 (octanesulfonyl), 2-Fua 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 39)   (Dap 3 (octanesulfonyl), Apc 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 39)   (Dap 3 (octanesulfonyl), Aib 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 39)   (Dap 3 (octanesulfonyl), Aib10hGhrelin(1-28)-NH 2 ; (SEQ ID: 42)   (Dap 3 (octanesulfonyl), A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 37)   (Dab 3 (octanesulfonyl), A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 37)   (Aib 2 , A6c 5 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 43)   (A6c 5 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 44)   (Aib 2,6 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 45)   (Aib 2 , Actio, A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 45)   (Aib 2 , 3-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 46)   (Aib 2 , Dmt 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 47)   (Aib 2 , Thz 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 47)   (Aib 2 , A5c 5 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 43)   (Aib 2,5 , A5c 12 ,Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 43)   (Aib 2 , hLeu 5 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 43)   (Aib 2 , Cha 5 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 43)   (Aib 2,6 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 45)   (Aib 2 , Thr 6 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 45)   (Aib 2 , Abu 6 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 45)   (Aib 2 , 4-Hyp&#39;, A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 47)   (Aib 2 , Pip&#39;, A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 47)   (Aib 2 , Dhp 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 47)   (Aib 2 , Ktp 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 47)   (Aib 2,8 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 48)   (Aib 2 , 2-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 46)   (Aib 2 , 3-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 46)   (Aib 2 , 4-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 46)   (Aib 2 , Taz 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 46)   (Aib 2 , 2-Thi 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 46)   (Aib 2 , 2-Fua 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 46)   (Aib 2 , Apc 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 46)   (Aib 2,9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 46)   (Aib 2,10 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 49)   (Dap 3 (octanesulfonyl), A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 38)   (Dab 3 (octanesulfonyl), A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 38)   (Aib 2 , A6c 5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 50)   (A6c 5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 51)   (Aib 2,6 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 52)   (Aib 2 , Actio, A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 52)   (Aib 2 , 3-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 53)   (Aib 2 , Dmt 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 54)   (Aib 2 , Thz 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 54)   (Aib 2 , A5c 5 , 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 50)   (Aib 2,5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 50)   (Aib 2 , hLeu 5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 50)   (Aib 2 , Cha 5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 50)   (Aib 2,6 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 52)   (Aib 2 , Thr 6 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 52)   (Aib 2 , Abu 6 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 52)   (Aib 2 , 4-Hyp&#39;, A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 54)   (Aib 2 , Pip&#39;, A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 54)   (Aib 2 , Dhp 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 54)   (Aib 2 , Ktp 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 54)   (Aib 2,8 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 55)   (Aib 2 , 2-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 53)   (Aib 2 , 3-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 53)   (Aib 2 , 4-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 53)   (Aib 2 , Taz 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 53)   (Aib 2 , 2-Thi 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 53)   (Aib 2 , 2-Fua 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 53)   (Aib 2 , Apc 9,16 , A5c 12 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 53)   (Aib 2,9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 53)   (Aib 2,10 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 56)   (A6c 5 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 44)   (Aib 6 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 57)   (Act 6 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 57)   (3-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 58)   (Dmt 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 59)   (Thz 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 59)   (A5c 5,12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 44)   (Aib 5 , A5c 12 ,Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 44)   (hLeu 5 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 44)   (Cha 5 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 44)   (Aib 6 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 57)   (Thr 6 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 57)   (Abu 6 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 57)   (4-Hyp&#39;, A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 59)   (Pip 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 59)   (Dhp 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 59)   (Ktp 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 59)   (Aib 8 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 60)   (2-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 58)   (3-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 58)   (4-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 58)   (Taz 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 58)   (2-Thi 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 58)   (2-Fua 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 58)   (Apc 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 58)   (Aib 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 58)   (Aib 10 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 61)   (Aib 6 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 62)   (A5c 5,12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 51)   (Actio, A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 62)   (3-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 63)   (Dmt 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 64)   (Thz 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 64)   (Aib 5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 51)   (hLeu 5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 51)   (Cha 5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 51)   (Thr 6 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 62)   (Abu 6 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 62)   (4-Hyp A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 64)   (Pip 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 64)   (Dhp 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 64)   (Ktp 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 64)   (Aib 8 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 65)   (2-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 63)   (3-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 63)   (4-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 63)   (Taz 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 63)   (2-Thi 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 63)   (2-Fua 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 63)   (Apc 9,16 , A5c 12 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 63)   (Aib 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 63)   (Aib 10 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 66)   (Aib 2 , Glu 3 (NH-hexyl), A6c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 67)   (Glu 3 (NH-hexyl), A6c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 68)   (Aib 2,6 , Glu 3 (NH-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 69)   (Aib 2 , Glu 3 (NH-hexyl), Act 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 69)   (Aib 2 , Glu 3 (NH-hexyl), 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 70)   (Aib 2 , Glu 3 (NH-hexyl), Dmt 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 71)   (Aib 2 , Glu 3 (NH-hexyl), Thz 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 71)   (Aib 2 , Glu 3 (NH-hexyl), A5c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 67)   (Aib 2,5 , Glu 3 (NH-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 67)   (Aib 2 , Glu 3 (NH-hexyl), hLeu 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 67)   (Aib 2 , Cha 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 7)   (Aib 2 ′ 6 , Glu 3 (NH-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 69)   (Aib 2 , Glu 3 (NH-hexyl), Thr 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 69)   (Aib 2 , Glu 3 (NH-hexyl), Abu 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 69)   (Aib 2 , Glu 3 (NH-hexyl), 4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 71)   (Aib 2 , Glu 3 (NH-hexyl), Pip 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 71)   (Aib 2 , Glu 3 (NH-hexyl), Dhp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 71)   (Aib 2 , Glu 3 (NH-hexyl), Ktp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 71)   (Aib 2,8 , Glu 3 (NH-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 72)   (Aib 2 , Glu 3 (NH-hexyl), 2-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 70)   (Aib 2 , Glu 3 (NH-hexyl), 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 70)   (Aib 2 , Glu 3 (NH-hexyl), 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 70)   (Aib 2 , Glu 3 (NH-hexyl), Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 70)   (Aib 2 , Glu 3 (NH-hexyl), 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 70)   (Aib 2 , Glu 3 (NH-hexyl), 2-Fua 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 70)   (Aib 2 , Glu 3 (NH-hexyl), Apc 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 70)   (Aib 2,9 , Glu 3 (NH-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 70)   (Aib 2,10 , Glu 3 (NH-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 73)   (Glu 3 (NH-hexyl), Aib 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 74)   (Glu 3 (NH-hexyl), A5c 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 68)   (Glu 3 (NH-hexyl), Act 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 74)   (Glu 3 (NH-hexyl), 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 75)   (Glu 3 (NH-hexyl), Dmt 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 76)   (Glu 3 (NH-hexyl), Thz 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 76)   (Glu 3 (NH-hexyl), Aib 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 68)   (Glu 3 (NH-hexyl), hLeu 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 68)   (Glu 3 (NH-hexyl), Cha 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 68)   (Glu 3 (NH-hexyl), Thr 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 74)   (Glu 3 (NH-hexyl), Abu 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 74)   (Glu 3 (NH-hexyl), 4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 76)   (Glu 3 (NH-hexyl), Pip 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 76)   (Glu 3 (NH-hexyl), Dhp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 76)   (Glu 3 (NH-hexyl), Ktp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 76)   (Glu 3 (NH-hexyl), Aib 8 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 41)   (Glu 3 (NH-hexyl), 2-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 75)   (Glu 3 (NH-hexyl), 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 75)   (Glu 3 (NH-hexyl), 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 75)   (Glu 3 (NH-hexyl), Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 75)   (Glu 3 (NH-hexyl), 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 75)   (Glu 3 (NH-hexyl), 2-Fua 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 75)   (Glu 3 (NH-hexyl), Apc 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 75)   (Glu 3 (NH-hexyl), Aib 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 75)   (Glu 3 (NH-hexyl), Aib 9 hGhrelin(1-28)-NH 2 ; (SEQ ID: 42)   (Aib 2 , Glu 3 (NH-hexyl), A6c 5 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 77)   (A6c 5 , Glu 3 (NH-hexyl), A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 78)   (Aib 2,6 , Glu 3 (NH-hexyl), A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 79)   (Aib 2 , Glu 3 (NH-hexyl), Actio, A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 79)   (Aib 2 , Glu 3 (NH-hexyl), 3-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 80)   (Aib 2 , Glu 3 (NH-hexyl), Dmt 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 81)   (Aib 2 , Glu 3 (NH-hexyl), Thz 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 81)   (Aib 2 , Glu 3 (NH-hexyl), A5c 5,12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 77)   (Aib 2,5 , Glu 3 (NH-hexyl), A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 77)   (Aib 2 , hLeu 5 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 43)   (Aib 2 , Glu 3 (NH-hexyl), Cha 5 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 77)   (Aib 2,6 , Glu 3 (NH-hexyl), A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 79)   (Aib 2 , Glu 3 (NH-hexyl), Thr 6 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 79)   (Aib 2 , Glu 3 (NH-hexyl), Abu 6 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 79)   (Aib 2 , Glu 3 (NH-hexyl), 4-Hyp&#39;, A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 81)   (Aib 2 , Glu 3 (NH-hexyl), Pip&#39;, A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 81)   (Aib 2 , Glu 3 (NH-hexyl), Dhp 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 81)   (Aib 2 , Glu 3 (NH-hexyl), Ktp 7 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 81)   (Aib 2,8 , Glu 3 (NH-hexyl), A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 82)   (Aib 2 , Glu 3 (NH-hexyl), 2-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 80)   (Aib 2 , Glu 3 (NH-hexyl), 3-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 80)   (Aib 2 , Glu 3 (NH-hexyl), 4-Pal 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 80)   (Aib 2 , Glu 3 (NH-hexyl), Taz 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 80)   (Aib 2 , Glu 3 (NH-hexyl), 2-Thi 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 80)   (Aib 2 , Glu 3 (NH-hexyl), 2-Fua 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 80)   (Aib 2 , Glu 3 (NH-hexyl), Apc 9 , A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 80)   (Aib 2,9 , Glu 3 (NH-hexyl), A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 80)   (Aib 2,12 , Glu 3 (NH-hexyl), 4-Pal 9 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 125)   (Aib 2,10 , Glu 3 (NH-hexyl), A5c 12 , Orn 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 83)   (Aib 2 , Glu 3 (NH-hexyl), A6c 5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 84)   (Glu 3 (NH-hexyl), A6c 5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 85)   (Aib 2,6 , Glu 3 (NH-hexyl), A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 86)   (Aib 2 , Glu 3 (NH-hexyl), Act 6 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 86)   (Aib 2 , Glu 3 (NH-hexyl), 3-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 87)   (Aib 2 , Glu 3 (NH-hexyl), Dmt 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 88)   (Aib 2 , Glu 3 (NH-hexyl), Thz 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 88)   (Aib 2 , Glu 3 (NH-hexyl), A5c 5 , 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 84)   (Aib 2,5 , Glu 3 (NH-hexyl), A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 84)   (Aib 2 , Glu 3 (NH-hexyl), hLeu 5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 84)   (Aib 2 , Glu 3 (NH-hexyl), Cha 5 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 84)   (Aib 2,6 , Glu 3 (NH-hexyl), A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 86)   (Aib 2 , Glu 3 (NH-hexyl), Thr 6 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 86)   (Aib 2 , Glu 3 (NH-hexyl), Abu 6 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 86)   (Aib 2 , Glu 3 (NH-hexyl), 4-Hyp&#39;, A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 88)   (Aib 2 , Glu 3 (NH-hexyl), Pip&#39;, A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 88)   (Aib 2 , Glu 3 (NH-hexyl), Dhp 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 88)   (Aib 2 , Glu 3 (NH-hexyl), Ktp 7 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 88)   (Aib 2,8 , Glu 3 (NH-hexyl), A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 89)   (Aib 2 , Glu 3 (NH-hexyl), 2-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 87)   (Aib 2 , Glu 3 (NH-hexyl), 3-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 87)   (Aib 2 , Glu 3 (NH-hexyl), 4-Pal 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 87)   (Aib 2 , Glu 3 (NH-hexyl), Taz 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 87)   (Aib 2 , Glu 3 (NH-hexyl), 2-Thi 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 87)   (Aib 2 , Glu 3 (NH-hexyl), 2-Fua 9 , A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 87)   (Aib 2 , Glu 3 (NH-hexyl), Apc 9,16 , A5c 12 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 87)   (Aib 2,9 , Glu 3 (NH-hexyl), A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 87)   (Aib 2,10 , Glu 3 (NH-hexyl), A5c 12 , Apc 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 90)   (Glu 3 (O-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 91)   (Aib 2 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 15)   (Glu 3 (NH-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 91)   (Aib 2 , Glu 3 (O-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 92)   Glu 3 (O-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 93)   (Aib 2 , Glu 3 (NH-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 92)   (Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 6)   (Aib 2 , Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 94)   Dap 3 (octanesulfonyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 93)   (Ava 2 , Dap 3 (octanesulfonyl))hGhrelin(2-28)-NH 2 ; (SEQ ID: 126)   (Ac-Gly 1 )hGhrelin(1-5)-NH 2 ; (SEQ ID: 95)   (Ac-Gly 1 )hGhrelin(1-6)-NH 2 ; (SEQ ID: 96)   (Ac-Gly 1 )hGhrelin(1-7)-NH 2 ; (SEQ ID: 97)   (Ac-Gly 1 , Aib 2 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 98)   (Ac-Gly 1 , Aib 2 , Glu 3 (NH-hexyl))hGhrelin(1-5)-NH 2 ; (SEQ ID: 99)   (Ac-Gly 1 , Aib 2 , Glu 3 (NH-hexyl))hGhrelin(1-6)-NH 2 ; (SEQ ID: 100)   (Ac-Gly 1 , Aib 2 , Glu 3 (NH-hexyl))hGhrelin(1-7)-NH 2 ; (SEQ ID: 101)   (Ac-Gly 1 , Aib 2 , Glu 3 (NH-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 102)   (Ac-Gly 1 , Aib 2 , Glu 3 (NH-hexyl), Arg 8 )hGhrelin(1-8)-NH 2 ; (SEQ ID: 103)   (Ac-Gly 1 , Aib 2 , Glu 3 (NH-hexyl), Lys 8 )hGhrelin(1-8)-NH 2 ; (SEQ ID: 103)   (n-butyryl-Gly 1 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 104)   (n-butyryl-Gly 1 , Aib 2 , Glu 3 (NH-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 105)   (isobutyryl-Gly 1 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 104)   (n-octanoyl-Gly 1 )hGhrelin(1-28)-NH 2 , (SEQ ID: 104)   Cys 3 (S(CH 2 ) 9 CH 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 106)   (Aib 2 , Ser 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 15)   (Aib 2,6 , Ser 3 )hGhrelin(1-28)-NH 2  (SEQ ID: 9)   (Aib 2 , Ser 3 , 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Aib 2 , Ser 3 , Thz 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Aib 2 , Ser 3 , Cha 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 7)   (Aib 2 , Ser 3 , Abu 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 9)   (Aib 2 , Ser 3 , 4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Aib 2 , Ser 3 , Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Aib 2 , Ser 3 , Dhp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Aib 2,8 , Ser 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 16)   (Aib 2 , Ser 3 , Pip 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Ac-Gly 1 , Aib 2,10 , Ser 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 107)   (Aib 2,10 , Ser 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 17)   (n-butyryl-Gly 1 , Aib 2 , Ser 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 108)   (Ac-Gly 1 , Aib 2 , Ser 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 98)   (Aib 2 , Ser 3 , Tic 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Ac-Gly 1 , Aib 2 , Ser 3 , Arg 8 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 109)   (Ser 3 , Aib 8 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 110)   (Ser 3 , Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (Ser 3 , 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (Ser 3 , 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (Aib 2 , Ser 3 , 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 13)   (Ser 3 , 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 19)   (Ser 3 , 4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 20)   (Aib 2 , Ser 3 , Tic 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 14)   (Aib 2 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 111)   (Aib 2,6 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 112)   (A5c 5 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 113)   (Aib 2 , Thr 3 , 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 114)   (Aib 2 , Thr 3 , Thz 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 115)   (Aib 2 , Thr 3 , Cha 5 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 116)   (Aib 2 , Thr 3 , Abu 6 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 112)   (Aib 2 , Thr 3 , 4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 115)   (Aib 2 , Thr 3 , Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 114)   (Aib 2 , Thr 3 , Dhp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 115)   (Aib 2,8 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 117)   (Aib 2 , Thr 3 , Pip 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 115)   (Ac-Gly 1 , Aib 2,10 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 118)   (Aib 2,10 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 118)   (n-butyryl-Gly 1 , Aib 2 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 119)   (Ac-Gly 1 , Aib 2 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 119)   (Aib 2 , Thr 3 , Tic 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 115)   (Ac-Gly 1 , Aib 2 , Thr 3 , Arg 8 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 120)   (Thr 3 , Aib 8 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 121)   (Thr 3 , Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 122)   (Thr 3 , 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 122)   (Thr 3 , 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 122)   (Aib 2 , Thr 3 , 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 114)   (Thr 3 , 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 122)   (Thr 3 , 4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 123)   (Aib 2 , Thr 3 , Tic 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 115)   (Ac-Gly 1 , Glu 3 (NH-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 124)   H-Inp-D-1-Nal-D-Trp-3-Pal-Lys-NH 2 ; (SEQ ID: 128)   H-Inp-D-2-Nal-D-Trp-4-Pal-Lys-NH 2 ; (SEQ ID: 129)   H-Inp-D-2-Nal-D-Trp-Om-Lys-NH 2 ; (SEQ ID: 129)   H-Inp-D-Bip-D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 130)   H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-Lys-NH 2 ; (SEQ ID: 131)   H-Inp-D-2-Nal-D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 131)   H-Inp-D-2-Nal-D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 132)   H-Inp-D-2-Nal-D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 132)   H-Inp-D-Dip-D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 133)   H-Inp-D-Bpa-D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 133)   H-Inp-D-2-Nal-D-Bpa-Phe-Lys-NH 2 ; (SEQ ID: 134)   H-Inp-D-2-Nal-D-Trp-3-Pal-NH 2 ; (SEQ ID: 135)   H-Inp-D-2-Nal-D-Trp-4-Pal-NH 2 ; (SEQ ID: 135)   H-Inp-D-1-Nal-D-Trp-3-Pal-NH 2 ; (SEQ ID: 136)   H-Inp-D-Bip-D-Trp-Phe-NH 2 ; (SEQ ID: 137)   H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-NH 2 ; (SEQ ID: 138)   H-Inp-D-2-Nal-D-Trp-Pff-NH 2 ; (SEQ ID: 138)   H-Inp-D-2-Nal-D-Trp-2-Thi-NH 2 ; (SEQ ID: 138)   H-Inp-D-2-Nal-D-Trp-Taz-NH 2 ; (SEQ ID: 138)   H-Inp-D-Dip-D-Trp-Phe-NH 2 ; (SEQ ID: 139)   H-Inp-D-2-Nal-D-Dip-Phe-NH 2 ; (SEQ ID: 140)   H-Inp-D-Bal -D-Trp-Phe-NH 2 ; (SEQ ID: 141)   H-Inp-D-2-Nal-D-Bal -Phe-NH 2 ; (SEQ ID: 142)   H-Inp-D-2-Nal-D-Trp-3-Pal-Lys-NH 2 ; (SEQ ID: 143)   H-Inp-D-Trp-D-2-Nal(Ψ)-Pim; (SEQ ID: 127)   H-Inp-D-Bal -D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 144)   H-Inp-D-Bal -D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 144)   H-Inp-D-1-Nal-D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 128)   H-Inp-D-2-Nal-D-Trp-Phe-Apc-NH 2 ; (SEQ ID: 2)   H-Inp-D-1-Nal-D-Trp-Phe-Apc-NH 2 ; (SEQ ID: 2)   H-Inp-D-Bal-D-Trp-Phe-Apc-NH 2 ; (SEQ ID: 2)   H-Apc-D-2-Nal-D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 145)   H-Apc-D-1-Nal-D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 146)   H-Inp-D-1-Nal-D-Trp-2-Thi-NH 2 ; (SEQ ID: 147)   H-Apc-D-1-Nal-D-Trp-Phe-NH 2 ; (SEQ ID: 148)   H-Inp-D-2-Nal-D-Trp(Ψ)-Pim; (SEQ ID: 149)   H-Inp-D-1-Nal-D-Trp(Ψ)-Pim; (SEQ ID: 149)   H-Inp-D-Bal-D-Trp(Ψ)-Pim; (SEQ ID: 149)   H-Aib-D-Ser(Bzl)-D-Trp(Ψ)-Pim; (SEQ ID: 150)   H-Inp-D-1-Nal-D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 151)   H-Inp-D-Bal -D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 151)   H-Apc-D-1-Nal-D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 152)   H-Apc-D-Bal -D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 152)   H-Apc-D-Bal -D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 153)   H-Apc-D-Bal -D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 153)   H-Apc-D-1-Nal-D-Trp-Phe-Apc-NH 2 ; (SEQ ID: 154)   H-Apc-D-Bal -D-Trp-Phe-Apc-NH 2 ; (SEQ ID: 154)   H-Apc-D-1-Nal-D-1-Nal-Phe-Apc-NH 2 ; (SEQ ID: 155)   H-Apc-D-1-Nal-D-2-Nal-Phe-Apc-NH 2 ; (SEQ ID: 155)   H-Apc-D-1-Nal-D-1-Nal-Phe-Lys-NH 2 ; (SEQ ID: 156)   H-Apc-D-Bal-D-1-Nal-Phe-Apc-NH 2 ; (SEQ ID: 157)   H-Apc-D-Bal-D-2-Nal-Phe-Apc-NH 2 ; (SEQ ID: 157)   H-Apc-D-Bal-D-1-Nal-Phe-Lys-NH 2 ; (SEQ ID: 158)   H-Apc-D-Bal-D-2-Nal-Phe-Lys-NH 2 ; (SEQ ID: 158)   H-Apc-D-1-Nal-D-Trp-2-Thi-NH 2 ; (SEQ ID: 159)   H-Apc-D-Bal -D-Trp-Phe-NH 2 ; (SEQ ID: 160)   H-Apc-D-1-Nal-D-Trp-Taz-NH 2 ; (SEQ ID: 159)   H-Apc-D-Bal -D-Trp-2-Thi-NH 2 ; (SEQ ID: 161)   H-Apc-D-Bal -D-Trp-Taz-NH 2 ; (SEQ ID: 161)   H-Apc-D-2-Nal-D-Trp-2-Thi-NH 2 ; (SEQ ID: 162)   H-Apc-D-2-Nal-D-Trp-Taz-NH 2 ; (SEQ ID: 162)   H-Inp-D-1-Nal-D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 163)   H-Inp-D-Bal-D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 163)   H-Apc-D-1-Nal-D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 164)   H-Apc-D-Bal -D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 164)   H-Apc-D-1-Nal-D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 165)   H-Apc-D-1-Nal-D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 165)   H-Apc-D-1-Nal-D-Trp-2-Fua-NH 2 ; (SEQ ID: 165)   H-Apc-D-1-Nal-D-Trp-2-Pal-NH 2 ; (SEQ ID: 166)   H-Apc-D-1-Nal-D-Trp-3-Pal-NH 2 ; (SEQ ID: 166)   H-Apc-D-1-Nal-D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 167)   H-Apc-D-1-Nal-D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 167)   H-Apc-D-1-Nal-D-Trp-3-Thi-NH 2 ; (SEQ ID: 168)   H-Apc-D-1-Nal-D-Trp-4-Pal-NH 2 ; (SEQ ID: 168)   H-Apc-D-1-Nal-D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 169)   H-Apc-D-1-Nal-D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 169)   H-Apc-D-1-Nal-D-Trp-Pff-NH 2 ; (SEQ ID: 168)   H-Apc-D-2-Nal-D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 170)   H-Apc-D-2-Nal-D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 170)   H-Apc-D-2-Nal-D-Trp-2-Fua-NH 2 ; (SEQ ID: 171)   H-Apc-D-2-Nal-D-Trp-2-Pal-NH 2 ; (SEQ ID: 171)   H-Apc-D-2-Nal-D-Trp-2-Thi-Apc-NH 2 ; (SEQ ID: 172)   H-Apc-D-2-Nal-D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 172)   H-Apc-D-2-Nal-D-Trp-3-Pal-NH 2 ; (SEQ ID: 171)   H-Apc-D-2-Nal-D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 173)   H-Apc-D-2-Nal-D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 173)   H-Apc-D-2-Nal-D-Trp-3-Thi-NH 2 ; (SEQ ID: 171)   H-Apc-D-2-Nal-D-Trp-4-Pal-NH 2 ; (SEQ ID: 171)   H-Apc-D-2-Nal-D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 174)   H-Apc-D-2-Nal-D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 174)   H-Apc-D-2-Nal-D-Trp-Pff-NH 2 ; (SEQ ID: 171)   H-Apc-D-2-Nal-D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 175)   H-Apc-D-2-Nal-D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 175)   H-Apc-D-Bal -D-Bal -2-Fua-Apc-NH 2 ; (SEQ ID: 176)   H-Apc-D-Bal -D-Bal -2-Fua-Lys-NH 2 ; (SEQ ID: 176)   H-Apc-D-Bal -D-Bal -2-Fua-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -2-Pal-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -2-Thi-Apc-NH 2 ; (SEQ ID: 178)   H-Apc-D-Bal -D-Bal -2-Thi-Lys-NH 2 ; (SEQ ID: 178)   H-Apc-D-Bal -D-Bal -2-Thi-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -3-Pal-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -3-Thi-Apc-NH 2 ; (SEQ ID: 179)   H-Apc-D-Bal -D-Bal -3-Thi-Lys-NH 2 ; (SEQ ID: 179)   H-Apc-D-Bal -D-Bal -3-Thi-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -4-Pal-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -Pff-Apc-NH 2 ; (SEQ ID: 180)   H-Apc-D-Bal -D-Bal -Pff-Lys-NH 2 ; (SEQ ID: 180)   H-Apc-D-Bal -D-Bal -Pff-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal-D-Bal-Phe-Apc-NH 2 ; (SEQ ID: 181)   H-Apc-D-Bal -D-Bal -Phe-Lys-NH 2 ; (SEQ ID: 181)   H-Apc-D-Bal -D-Bal -Phe-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -Taz-Apc-NH 2 ; (SEQ ID: 182)   H-Apc-D-Bal -D-Bal -Taz-Lys-NH 2 ; (SEQ ID: 182)   H-Apc-D-Bal -D-Bal -Taz-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 183)   H-Apc-D-Bal -D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 183)   H-Apc-D-Bal -D-Trp-2-Fua-NH 2 ; (SEQ ID: 184)   H-Apc-D-Bal -D-Trp-2-Pal-NH 2 ; (SEQ ID: 184)   H-Apc-D-Bal -D-Trp-3-Pal-NH 2 ; (SEQ ID: 184)   H-Apc-D-Bal -D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 185)   H-Apc-D-Bal -D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 185)   H-Apc-D-Bal -D-Trp-3-Thi-NH 2 ; (SEQ ID: 184)   H-Apc-D-Bal -D-Trp-4-Pal-NH 2 ; (SEQ ID: 184)   H-Apc-D-Bal -D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 186)   H-Apc-D-Bal -D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 186)   H-Apc-D-Bal -D-Trp-Pff-NH 2 ; (SEQ ID: 184)   H-Inp-D-1-Nal-D-Bal -2-Fua-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-1-Nal-D-Bal -2-Fua-NH 2 ; (SEQ ID: 188)   H-Inp-D-1-Nal-D-Bal -2-Thi-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-1-Nal-D-Bal -3-Thi-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-1-Nal-D-Bal -Pff-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-1-Nal-D-Bal -Pff-NH 2 ; (SEQ ID: 188)   H-Inp-D-1-Nal-D-Bal -Phe-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-1-Nal-D-Bal -Taz-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-1-Nal-D-Bal -Taz-NH 2 ; (SEQ ID: 188)   H-Inp-D-1-Nal-D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 189)   H-Inp-D-1-Nal-D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 189)   H-Inp-D-1-Nal-D-Trp-2-Fua-NH 2 ; (SEQ ID: 189)   H-Inp-D-1-Nal-D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 190)   H-Inp-D-1-Nal-D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 190)   H-Inp-D-1-Nal-D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 191)   H-Inp-D-1-Nal-D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 191)   H-Inp-D-1-Nal-D-Trp-Pff-NH 2 ; (SEQ ID: 192)   H-Inp-D-1-Nal-D-Trp-Taz-NH 2 ; (SEQ ID: 192)   H-Inp-D-2-Nal-D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 193)   H-Inp-D-2-Nal-D-Trp-2-Fua-NH 2 ; (SEQ ID: 194)   H-Inp-D-2-Nal-D-Trp-2-Thi-Apc-NH 2 ; (SEQ ID: 193)   H-Inp-D-2-Nal-D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 193)   H-Inp-D-2-Nal-D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 195)   H-Inp-D-2-Nal-D-Trp-3-Thi-NH 2 ; (SEQ ID: 194)   H-Inp-D-2-Nal-D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 193)   H-Inp-D-2-Nal-D-Trp-Pff-NH 2 ; (SEQ ID: 194)   H-Inp-D-2-Nal-D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 193)   H-Inp-D-2-Nal-D-Trp-Taz-NH 2 ; (SEQ ID: 194)   H-Inp-D-Bal -D-Bal -2-Fua-Lys-NH 2 ; (SEQ ID: 196)   H-Inp-D-Bal -D-Bal -2-Fua-NH 2 ; (SEQ ID: 197)   H-Inp-D-Bal -D-Bal -2-Thi-Lys-NH 2 ; (SEQ ID: 196)   H-Inp-D-Bal -D-Bal -3-Thi-Lys-NH 2 ; (SEQ ID: 196)   H-Inp-D-Bal -D-Bal -Pff-Lys-NH 2 ; (SEQ ID: 196)   H-Inp-D-Bal -D-Bal -Pff-NH 2 ; (SEQ ID: 197)   H-Inp-D-Bal -D-Bal -Phe-Lys-NH 2 ; (SEQ ID: 196)   H-Inp-D-Bal -D-Bal -Taz-Lys-NH 2 ; (SEQ ID: 196)   H-Inp-D-Bal -D-Bal -Taz-NH 2 ; (SEQ ID: 197)   H-Inp-D-Bal -D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 198)   H-Inp-D-Bal -D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 198)   H-Inp-D-Bal -D-Trp-2-Fua-NH 2 ; (SEQ ID: 199)   H-Inp-D-Bal -D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 200)   H-Inp-D-Bal -D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 200)   H-Inp-D-Bal-D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 201)   H-Inp-D-Bal -D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 201)   H-Inp-D-Bal -D-Trp-Pff-NH 2 ; (SEQ ID: 199)   H-Inp-D-Bal -D-Trp-Taz-NH 2 ; (SEQ ID: 199)   H-Inp-D-Bip-D-Bal -2-Fua-Lys-NH 2 ; (SEQ ID: 202)   H-Inp-D-Bip-D-Bal -2-Fua-NH 2 ; (SEQ ID: 203)   H-Inp-D-Bip-D-Bal -2-Thi-Lys-NH 2 ; (SEQ ID: 202)   H-Inp-D-Bip-D-Bal -3-Thi-Lys-NH 2 ; (SEQ ID: 202)   H-Inp-D-Bip-D-Bal -Pff-Lys-NH 2 ; (SEQ ID: 202)   H-Inp-D-Bip-D-Bal -Pff-NH 2 ; (SEQ ID: 203)   H-Inp-D-Bip-D-Bal -Taz-Lys-NH 2 ; (SEQ ID: 204)   H-Inp-D-Bip-D-Bal -Taz-NH 2 ; (SEQ ID: 205)   H-Inp-D-Bip-D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 206)   H-Inp-D-Bip-D-Trp-2-Fua-NH 2 ; (SEQ ID: 207)   H-Inp-D-Bip-D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 206)   H-Inp-D-Bip-D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 206)   H-Inp-D-Bip-D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 206)   H-Inp-D-Bip-D-Trp-Pff-NH 2 ; (SEQ ID: 207)   H-Inp-D-Bip-D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 206)   H-Inp-D-Bip-D-Trp-Taz-NH 2 ; (SEQ ID: 207)   H-Inp-D-1-Nal-D-Trp-3-Pal-Lys-NH 2 ; (SEQ ID: 128)   H-Inp-D-2-Nal-D-Trp-4-Pal-Lys-NH 2 ; (SEQ ID: 129)   H-Inp-D-2-Nal-D-Trp-Om-Lys-NH 2 ; (SEQ ID: 129)   H-Inp-D-Bip-D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 130)   H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-Lys-NH 2 ; (SEQ ID: 131)   H-Inp-D-2-Nal-D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 131)   H-Inp-D-2-Nal-D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 132)   H-Inp-D-2-Nal-D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 132)   H-Inp-D-Dip-D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 133)   H-Inp-D-Bpa-D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 133)   H-Inp-D-2-Nal-D-Bpa-Phe-Lys-NH 2 ; (SEQ ID: 134)   H-Inp-D-2-Nal-D-Trp-Thr(Bzl)-NH 2 ; (SEQ ID: 138)   H-Inp-D-2-Nal-D-Trp-Pff-NH 2 ; (SEQ ID: 138)   H-Inp-D-2-Nal-D-Trp-Taz-NH 2 ; (SEQ ID: 138)   H-Inp-D-2-Nal-D-Dip-Phe-NH 2 ; (SEQ ID: 140)   H-Inp-D-2-Nal-D-Trp-3-Pal-Lys-NH 2 ; (SEQ ID: 143)   H-Inp-D-Trp-D-2-Nal(Ψ)-Pim; (SEQ ID: 127)   H-Inp-D-Bal -D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 144)   H-Inp-D-Bal -D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 144)   H-Inp-D-1-Nal-D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 128)   H-Inp-D-2-Nal-D-Trp-Phe-Apc-NH 2 ; (SEQ ID: 2)   H-Inp-D-1-Nal-D-Trp-Phe-Apc-NH 2 ; (SEQ ID: 2)   H-Inp-D-Bal-D-Trp-Phe-Apc-NH 2 ; (SEQ ID: 2)   H-Apc-D-2-Nal-D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 145)   H-Apc-D-1-Nal-D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 146)   H-Inp-D-2-Nal-D-Trp(Ψ)-Pim; (SEQ ID: 149)   H-Inp-D-1-Nal-D-Trp(Ψ)-Pim; (SEQ ID: 149)   H-Inp-D-Bal-D-Trp(Ψ)-Pim; (SEQ ID: 149)   H-Aib-D-Ser(Bzl)-D-Trp(Ψ)-Pim; (SEQ ID: 150)   H-Inp-D-1-Nal-D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 151)   H-Inp-D-Bal -D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 151)   H-Apc-D-1-Nal-D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 152)   H-Apc-D-Bal -D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 152)   H-Apc-D-Bal -D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 153)   H-Apc-D-Bal -D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 153)   H-Apc-D-1-Nal-D-Trp-Phe-Apc-NH 2 ; (SEQ ID: 154)   H-Apc-D-Bal -D-Trp-Phe-Apc-NH 2 ; (SEQ ID: 154)   H-Apc-D-1-Nal-D-1-Nal-Phe-Apc-NH 2 ; (SEQ ID: 155)   H-Apc-D-1-Nal-D-2-Nal-Phe-Apc-NH 2 ; (SEQ ID: 155)   H-Apc-D-1-Nal-D-1-Nal-Phe-Lys-NH 2 ; (SEQ ID: 156)   H-Apc-D-Bal-D-1-Nal-Phe-Apc-NH 2 ; (SEQ ID: 157)   H-Apc-D-Bal-D-2-Nal-Phe-Apc-NH 2 ; (SEQ ID: 157)   H-Apc-D-Bal-D-1-Nal-Phe-Lys-NH 2 ; (SEQ ID: 158)   H-Apc-D-Bal-D-2-Nal-Phe-Lys-NH 2 ; (SEQ ID: 158)   H-Apc-D-1-Nal-D-Trp-2-Thi-NH 2 ; (SEQ ID: 159)   H-Apc-D-Bal -D-Trp-Phe-NH 2 ; (SEQ ID: 160)   H-Apc-D-1-Nal-D-Trp-Taz-NH 2 ; (SEQ ID: 159)   H-Apc-D-Bal -D-Trp-2-Thi-NH 2 ; (SEQ ID: 161)   H-Apc-D-Bal -D-Trp-Taz-NH 2 ; (SEQ ID: 161)   H-Apc-D-2-Nal-D-Trp-2-Thi-NH 2 ; (SEQ ID: 162)   H-Apc-D-2-Nal-D-Trp-Taz-NH 2 ; (SEQ ID: 162)   H-Inp-D-1-Nal-D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 163)   H-Inp-D-Bal-D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 163)   H-Apc-D-1-Nal-D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 164)   H-Apc-D-Bal -D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 164)   H-Inp-D-2-Nal-D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 195)   H-Inp-D-Bal -D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 200)   H-Inp-D-Bal -D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 198)   H-Inp-D-Bal -D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 201)   H-Inp-D-Bal -D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 200)   H-Inp-D-Bal -D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 198)   H-Inp-D-Bal-D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 201)   H-Apc-D-Bal -D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 185)   H-Apc-D-Bal -D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 183)   H-Apc-D-Bal -D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 186)   H-Inp-D-Bal -D-Bal -Phe-Lys-NH 2 ; (SEQ ID: 196)   H-Inp-D-Bal -D-Bal -2-Thi-Lys-NH 2 ; (SEQ ID: 196)   H-Inp-D-Bal -D-Bal -3-Thi-Lys-NH 2 ; (SEQ ID: 196)   H-Inp-D-Bal -D-Bal -Taz-Lys-NH 2 ; (SEQ ID: 196)   H-Inp-D-Bal -D-Bal -2-Fua-Lys-NH 2 ; (SEQ ID: 196)   H-Inp-D-Bal -D-Bal -Pff-Lys-NH 2 ; (SEQ ID: 196)   H-Apc-D-Bal -D-Bal -Phe-Lys-NH 2 ; (SEQ ID: 181)   H-Apc-D-Bal -D-Bal -2-Thi-Lys-NH 2 ; (SEQ ID: 178)   H-Apc-D-Bal -D-Bal -3-Thi-Lys-NH 2 ; (SEQ ID: 179)   H-Apc-D-Bal -D-Bal -Taz-Lys-NH 2 ; (SEQ ID: 182)   H-Apc-D-Bal -D-Bal -2-Fua-Lys-NH 2 ; (SEQ ID: 176)   H-Apc-D-Bal -D-Bal -Pff-Lys-NH 2 ; (SEQ ID: 180)   H-Inp-D-1-Nal-D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 190)   H-Inp-D-1-Nal-D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 189)   H-Inp-D-1-Nal-D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 191)   H-Inp-D-1-Nal-D-Bal -Phe-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-1-Nal-D-Bal -2-Thi-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-1-Nal-D-Bal -3-Thi-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-1-Nal-D-Bal -Taz-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-1-Nal-D-Bal -2-Fua-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-1-Nal-D-Bal -Pff-Lys-NH 2 ; (SEQ ID: 187)   H-Inp-D-2-Nal-D-Trp-2-Thi-Apc-NH 2 ; (SEQ ID: 193)   H-Inp-D-2-Nal-D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 193)   H-Inp-D-2-Nal-D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 193)   H-Inp-D-2-Nal-D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 193)   H-Inp-D-2-Nal-D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 193)   H-Inp-D-1-Nal-D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 190)   H-Inp-D-1-Nal-D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 189)   H-Inp-D-1-Nal-D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 191)   H-Apc-D-1-Nal-D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 167)   H-Apc-D-1-Nal-D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 165)   H-Apc-D-1-Nal-D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 169)   H-Apc-D-2-Nal-D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 172)   H-Apc-D-2-Nal-D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 173)   H-Apc-D-2-Nal-D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 175)   H-Apc-D-2-Nal-D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 170)   H-Apc-D-2-Nal-D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 174)   H-Inp-D-Bip-D-Trp-2-Thi-Lys-NH 2 ; (SEQ ID: 206)   H-Inp-D-Bip-D-Trp-3-Thi-Lys-NH 2 ; (SEQ ID: 206)   H-Inp-D-Bip-D-Trp-Taz-Lys-NH 2 ; (SEQ ID: 206)   H-Inp-D-Bip-D-Trp-2-Fua-Lys-NH 2 ; (SEQ ID: 206)   H-Inp-D-Bip-D-Trp-Pff-Lys-NH 2 ; (SEQ ID: 206)   H-Inp-D-Bip-D-Bal -2-Thi-Lys-NH 2 ; (SEQ ID: 202)   H-Inp-D-Bip-D-Bal -3-Thi-Lys-NH 2 ; (SEQ ID: 202)   H-Inp-D-Bip-D-Bal -Taz-Lys-NH 2 ; (SEQ ID: 204)   H-Inp-D-Bip-D-Bal -2-Fua-Lys-NH 2 ; (SEQ ID: 202)   H-Inp-D-Bip-D-Bal-Pff-Lys-NH 2 ; (SEQ ID: 202)   H-Apc-D-Bal -D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 185)   H-Apc-D-Bal -D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 183)   H-Apc-D-Bal -D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 186)   H-Apc-D-Bal-D-Bal-Phe-Apc-NH 2 ; (SEQ ID: 181)   H-Apc-D-Bal -D-Bal -2-Thi-Apc-NH 2 ; (SEQ ID: 178)   H-Apc-D-Bal -D-Bal -3-Thi-Apc-NH 2 ; (SEQ ID: 179)   H-Apc-D-Bal -D-Bal -Taz-Apc-NH 2 ; (SEQ ID: 182)   H-Apc-D-Bal -D-Bal -2-Fua-Apc-NH 2 ; (SEQ ID: 176)   H-Apc-D-Bal -D-Bal -Pff-Apc-NH 2 ; (SEQ ID: 180)   H-Apc-D-1-Nal-D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 167)   H-Apc-D-1-Nal-D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 165)   H-Apc-D-1-Nal-D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 169)   H-Apc-D-2-Nal-D-Trp-2-Thi-Apc-NH 2 ; (SEQ ID: 172)   H-Apc-D-2-Nal-D-Trp-3-Thi-Apc-NH 2 ; (SEQ ID: 173)   H-Apc-D-2-Nal-D-Trp-Taz-Apc-NH 2 ; (SEQ ID: 175)   H-Apc-D-2-Nal-D-Trp-2-Fua-Apc-NH 2 ; (SEQ ID: 170)   H-Apc-D-2-Nal-D-Trp-Pff-Apc-NH 2 ; (SEQ ID: 174)   H-Inp-D-Bal -D-Trp-Taz-NH 2 ; (SEQ ID: 199)   H-Inp-D-Bal -D-Trp-2-Fua-NH 2 ; (SEQ ID: 199)   H-Inp-D-Bal -D-Trp-Pff-NH 2 ; (SEQ ID: 199)   H-Apc-D-Bal -D-Trp-3-Thi-NH 2 ; (SEQ ID: 184)   H-Apc-D-Bal -D-Trp-2-Fua-NH 2 ; (SEQ ID: 184)   H-Apc-D-Bal -D-Trp-Pff-NH 2 ; (SEQ ID: 184)   H-Apc-D-Bal -D-Trp-4-Pal-NH 2 ; (SEQ ID: 184)   H-Apc-D-Bal -D-Trp-3-Pal-NH 2 ; (SEQ ID: 184)   H-Apc-D-Bal -D-Trp-2-Pal-NH 2 ; (SEQ ID: 184)   H-Inp-D-Bal -D-Bal -Taz-NH 2 ; (SEQ ID: 197)   H-Inp-D-Bal -D-Bal -2-Fua-NH 2 ; (SEQ ID: 197)   H-Inp-D-Bal -D-Bal -Pff-NH 2 ; (SEQ ID: 197)   H-Apc-D-Bal -D-Bal -Phe-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -2-Thi-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -3-Thi-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -Taz-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -2-Fua-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -Pff-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -4-Pal-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -3-Pal-NH 2 ; (SEQ ID: 177)   H-Apc-D-Bal -D-Bal -2-Pal-NH 2 ; (SEQ ID: 177)   H-Inp-D-1-Nal-D-Trp-Taz-NH 2 ; (SEQ ID: 192)   H-Inp-D-1-Nal-D-Trp-2-Fua-NH 2 ; (SEQ ID: 189)   H-Inp-D-1-Nal-D-Trp-Pff-NH 2 ; (SEQ ID: 192)   H-Inp-D-1-Nal-D-Bal -Taz-NH 2 ; (SEQ ID: 188)   H-Inp-D-1-Nal-D-Bal -2-Fua-NH 2 ; (SEQ ID: 188)   H-Inp-D-1-Nal-D-Bal -Pff-NH 2 ; (SEQ ID: 188)   H-Inp-D-2-Nal-D-Trp-Taz-NH 2 ; (SEQ ID: 194)   H-Inp-D-2-Nal-D-Trp-2-Fua-NH 2 ; (SEQ ID: 194)   H-Inp-D-2-Nal-D-Trp-Pff-NH 2 ; (SEQ ID: 194)   H-Apc-D-1-Nal-D-Trp-3-Thi-NH 2 ; (SEQ ID: 168)   H-Apc-D-1-Nal-D-Trp-2-Fua-NH 2 ; (SEQ ID: 165)   H-Apc-D-1-Nal-D-Trp-Pff-NH 2 ; (SEQ ID: 168)   H-Apc-D-1-Nal-D-Trp-4-Pal-NH 2 ; (SEQ ID: 168)   H-Apc-D-1-Nal-D-Trp-3-Pal-NH 2 ; (SEQ ID: 166)   H-Apc-D-1-Nal-D-Trp-2-Pal-NH 2 ; (SEQ ID: 166)   H-Apc-D-2-Nal-D-Trp-3-Thi-NH 2 ; (SEQ ID: 171)   H-Apc-D-2-Nal-D-Trp-2-Fua-NH 2 ; (SEQ ID: 171)   H-Apc-D-2-Nal-D-Trp-Pff-NH 2 ; (SEQ ID: 171)   H-Apc-D-2-Nal-D-Trp-4-Pal-NH 2 ; (SEQ ID: 171)   H-Apc-D-2-Nal-D-Trp-3-Pal-NH 2 ; (SEQ ID: 171)   H-Apc-D-2-Nal-D-Trp-2-Pal-NH 2 ; (SEQ ID: 171)   H-Inp-D-Bip-D-Trp-Taz-NH 2 ; (SEQ ID: 207)   H-Inp-D-Bip-D-Trp-2-Fua-NH 2 ; (SEQ ID: 207)   H-Inp-D-Bip-D-Trp-Pff-NH 2 ; (SEQ ID: 207)   H-Inp-D-Bip-D-Bal -Taz-NH 2 ; (SEQ ID: 205)   H-Inp-D-Bip-D-Bal -2-Fua-NH 2 ; (SEQ ID: 203)   H-Inp-D-Bip-D-Bal -Pff-NH 2 ; (SEQ ID: 203)   H-Inp-D-1-Nal-D-Trp-2-Thi-Apc-NH 2 ; (SEQ ID: 208)   H-Inp-D-Bal -D-Trp-2-Thi-Apc-NH 2 ; (SEQ ID: 208)   H-Apc-D-1-Nal-D-Trp-2-Thi-Apc-NH 2 ; (SEQ ID: 209)   H-Apc-D-Bal -D-Trp-2-Thi-Apc-NH 2 ; (SEQ ID: 209)   H-Apc-D-1-Nal-D-Trp-Phe-Lys-NH 2 ; (SEQ ID: 145)   (Ser(n-octanoyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 210)   (Glu(NH-hexyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 211)   (Glu(NH-hexyl) 3,15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 212)   (Glu(NH-hexyl) 3 , Ser(n-octanoyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 213)   (Aib 2 , Glu(NH-hexyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 214)   (Aib 2 , Glu(NH-hexyl) 3,15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 215)   (Aib 2,8 , Glu(NH-hexyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 216)   (Aib 2,8 , Glu(NH-hexyl) 3,15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 217)   (Aib 2,10 , Glu(NH-hexyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 218)   (Aib 2,10 , Glu(NH-hexyl) 3,15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 219)   (Ser(n-octanoyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 220)   (Glu(NH-hexyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 221)   (Glu(NH-hexyl) 3,16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 222)   (Glu(NH-hexyl) 3 , Ser(n-octanoyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 223)   (Aib 2 , Glu(NH-hexyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 224)   (Aib 2 , Glu(NH-hexyl) 3,16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 225)   (Aib 2,8 , Glu(NH-hexyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 226)   (Aib 2,8 , Glu(NH-hexyl) 3,16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 227)   (Aib 2,10 , Glu(NH-hexyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 228)   (Aib 2,10 , Glu(NH-hexyl) 3,16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 229)   (Ser(n-octanoyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 230)   (Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 231)   (Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 232)   (Glu(NH-hexyl) 3 , Ser(n-octanoyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 233)   (Dap(octanesulfonyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 234)   (Dap(octanesulfonyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 235)   (Dap(octanesulfonyl) 3 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 236)   (Dap(octanesulfonyl) 3 , Ser(n-octanoyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 237)   (Glu(NH-hexyl) 3 , Dap(octanesulfonyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 238)   (Cys(S—(CH 2 ) 9 CH 3 ) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 239)   (Cys(S—(CH 2 ) 9 CH 3 ) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 240)   (Glu(NH-hexyl) 3 , Cys(S—(CH 2 ) 9 CH 3 ) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 241)   (Cys(S—(CH 2 ) 9 CH 3 ) 3 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 242)   (Cys(S—(CH 2 ) 9 CH 3 ) 3 , Ser(n-octanoyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 243)   (Aib 2 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 244)   (Aib 2 , Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 245)   (Aib 2 , Thz 7 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 246)   (Aib 2 , 4-Hyp 7 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 246)   (Aib 2 , Dhp 7 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 246)   (Aib 2 , Pip 7 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 246)   (Aib 2 , Tic 7 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 246)   (Aib 2 , Glu(NH-hexyl) 3,17 , Thz 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 247)   (Aib 2 , Glu(NH-hexyl) 3,17 , 4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 247)   (Aib 2 , Glu(NH-hexyl) 3,17 , Dhp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 247)   (Aib 2 , Glu(NH-hexyl) 3,17 , Pip 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 247)   (Aib 2 , Glu(NH-hexyl) 3,17 , Tic 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 247)   (Aib 2,8 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 248)   (Aib 2,8 , Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 249)   (Aib 2 , 3-Pal 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 250)   (Aib 2 , 4-Pal 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 250)   (Aib 2 , Taz 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 250)   (Aib 2 , 2-Thi 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 250)   (Aib 2 , Glu(NH-hexyl) 3,17 , 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 251)   (Aib 2 , Glu(NH-hexyl) 3,17 , 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 251)   (Aib 2 , Glu(NH-hexyl) 3,17 , Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 251)   (Aib 2 , Glu(NH-hexyl) 3,17 , 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 251)   (Aib 2,10 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 252)   (Aib 2,10 , Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 253)   (Aib 8 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 254)   (Taz 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 255)   (3-Pal 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 255)   (4-Pal 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 255)   (2-Thi 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 255)   (Glu(NH-hexyl) 3,17 , Aib 8 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 256)   (Glu(NH-hexyl) 3,17 , Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 257)   (Glu(NH-hexyl) 3,17 , 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 257)   (Glu(NH-hexyl) 3,17 , 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 257)   (Glu(NH-hexyl) 3,17 , 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 257)   (Aib 1,2,10 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 258)   (Aib 1,2,10 , Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 259)   (A5c 2 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 260)   (A5c 2 , Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 261)   (Glu(1-heptanol) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 262)   (Asp (1-heptanol) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 263)   (Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 264)   (Asp(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 265)   (Aib 2 , Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 266)   (Lys(biotinyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 267)   (Ser(n-octanoyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 268)   (Glu(NH-hexyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 269)   (Glu(NH-hexyl) 3,18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 270)   (Glu(NH-hexyl) 3 , Ser(n-octanoyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 271)   (Aib 2 , Glu(NH-hexyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 272)   (Aib 2 , Glu(NH-hexyl) 3,18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 273)   (Aib 2,8 , Glu(NH-hexyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 274)   (Aib 2,8 , Glu(NH-hexyl) 3,18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 275)   (Aib 2,10 , Glu(NH-hexyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 276)   (Aib 2,10 , Glu(NH-hexyl) 3,18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 277)   (Ser(n-octanoyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 278)   (Glu(NH-hexyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 279)   (Glu(NH-hexyl) 3,19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 280)   (Glu(NH-hexyl) 3 , Ser(n-octanoyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 281)   (Aib 2 , Glu(NH-hexyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 282)   (Aib 2 , Glu(NH-hexyl) 3,19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 283)   (Aib 2,8 , Glu(NH-hexyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 284)   (Aib 2,8 , Glu(NH-hexyl) 3,19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 285)   (Aib 2,10 , Glu(NH-hexyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 286)   (Aib 2,10 , Glu(NH-hexyl) 3,19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 287)   (Ser(n-octanoyl) 20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 288)   (Glu(NH-hexyl) 20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 289)   (Glu(NH-hexyl) 3,20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 290)   (Glu(NH-hexyl) 3 , Ser(n-octanoyl) 20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 291)   (Aib 2 , Glu(NH-hexyl) 2 1hGhrelin(1-28)-NH 2 ; (SEQ ID: 292)   (Aib 2 , Glu(NH-hexyl) 3,20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 293)   (Aib 2,8 , Glu(NH-hexyl) 9 hGhrelin(1-28)-NH 2 ; (SEQ ID: 294)   (Aib 2,8 , Glu(NH-hexyl) 3,20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 295)   (Aib 2,10 , Glu(NH-hexyl) 2,20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 296)   (Aib 2,10 , Glu(NH-hexyl) 3,20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 297)   (Ac-Gly 1 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 298)   (Ac-Gly 1 , Ser(n-octanoyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 299)   (Ac-Gly 1 , Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 300)   Glu(NH-hexyl) 3 , Ser(n-octanoyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 301)   (Ac-Gly 1 , Dap(octanesulfonyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 302)   (Ac-Gly 1 , Dap(octanesulfonyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 303)   Dap(octanesulfonyl) 3 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 304)   (Ac-Gly 1 , Dap(octanesulfonyl) 3 , Ser(n-octanoyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 305)   (Ac-Gly 1 , Glu(NH-hexyl) 3 , Dap(octanesulfonyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 306)   (Ac-Gly 1 , Cys(S—(CH 2 ) 9 CH 3 ) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 307)   (Ac-Gly 1 , Cys(S—(CH 2 ) 9 CH 3 ) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 308)   (Ac-Gly 1 , Glu(NH-hexyl) 3 , Cys(S—(CH 2 ) 9 CH 3 ) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 309)   (Ac-Gly 1 , Cys(S—(CH 2 ) 9 CH 3 ) 3 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 310)   (Ac-Gly 1 , Cys(S—(CH 2 ) 9 CH 3 ) 3 , Ser(n-octanoyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 311)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 312)   (Ac-Gly 1 , Aib 2 , Thz 7 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 313)   (Ac-Gly 1 , Aib 2 , 4-Hyp 7 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 313)   (Ac-Gly 1 , Aib 2 , Dhp 7 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 313)   (Ac-Gly 1 , Aib 2 , Pip 7 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 313)   (Ac-Gly 1 , Aib 2 , Tic 7 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 313)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,17 , Thz 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 314)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,17 , 4-Hyp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 314)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,17 , Dhp 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 314)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,17 , Pip 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 314)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,17 , Tic 7 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 314)   (Ac-Gly 1 , Aib 2,8 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 315)   (Ac-Gly 1 , Aib 2 , 3-Pal 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 316)   (Ac-Gly 1 , Aib 2 , 4-Pal 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 316)   (Ac-Gly 1 , Aib 2 , Taz 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 316)   (Ac-Gly 1 , Aib 2 , 2-Thi 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 316)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,17 , 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 317)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,17 , 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 317)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,17 , Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 317)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,17 , 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 317)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 318)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 319)   (Ac-Gly 1 , Aib 8 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 320)   (Ac-Gly 1 , Taz 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 321)   (Ac-Gly 1 , 3-Pal 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 321)   (Ac-Gly 1 , 4-Pal 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 321)   (Ac-Gly 1 , 2-Thi 9 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 321)   (Ac-Gly 1 , Glu(NH-hexyl) 3,17 , Aib 8 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 322)   (Ac-Gly 1 , Glu(NH-hexyl) 3,17 , Taz 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 323)   (Ac-Gly 1 , Glu(NH-hexyl) 3,17 , 3-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 323)   (Ac-Gly 1 , Glu(NH-hexyl) 3,17 , 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 323)   (Ac-Gly 1 , Glu(NH-hexyl) 3,17 , 2-Thi 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 323)   (Ac-Gly 1 , Aib Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 324)   (Ac-Gly 1 , Aib Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 325)   (Ac-Gly 1 , A5c 2 , Glu(NH-hexyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 326)   (Ac-Gly 1 , A5c 2 , Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 327)   (Ac-Gly 1 , Glu(1-heptanol) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 328)   (Ac-Gly 1 , Asp(1-heptanol) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 329)   (Ac-Gly 1 , Glu(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 330)   (Ac-Gly 1 , Asp(NH-hexyl) 3,17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 331)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 3 , Lys(biotinyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 332)   (Ac-Gly 1 , Glu(NH-hexyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 333)   (Ac-Gly 1 , Ser(n-octanoyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 334)   (Ac-Gly 1 , Glu(NH-hexyl) 3,15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 335)   (Ac-Gly 1 , Glu(NH-hexyl) 3 , Ser(n-octanoyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 336)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 337)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 338)   (Ac-Gly 1 , Glu(NH-hexyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 339)   (Ac-Gly 1 , Glu(NH-hexyl) 3,15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 340)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 341)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 3,15 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 342)   (Ac-Gly 1 , Glu(NH-hexyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 343)   (Ac-Gly 1 , Ser(n-octanoyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 344)   (Ac-Gly 1 , Glu(NH-hexyl) 3,16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 345)   (Ac-Gly 1 , Glu(NH-hexyl) 3 , Ser(n-octanoyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 346)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 347)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 348)   (Ac-Gly 1 , Glu(NH-hexyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 349)   (Ac-Gly 1 , Glu(NH-hexyl) 3,16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 350)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 351)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 3,16 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 352)   (Ac-Gly 1 , Glu(NH-hexyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 353)   (Ac-Gly 1 , Ser(n-octanoyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 354)   (Ac-Gly 1 , Glu(NH-hexyl) 3,18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 355)   (Ac-Gly 1 , Glu(NH-hexyl) 3 , Ser(n-octanoyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 356)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 357)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 358)   (Ac-Gly 1 , Glu(NH-hexyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 359)   (Ac-Gly 1 , Glu(NH-hexyl) 3,18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 360)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 361)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 3,18 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 362)   (Ac-Gly 1 , Glu(NH-hexyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 363)   (Ac-Gly 1 , Ser(n-octanoyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 364)   (Ac-Gly 1 , Glu(NH-hexyl) 3,19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 365)   (Ac-Gly 1 , Glu(NH-hexyl) 3 , Ser(n-octanoyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 366) (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 367)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 368)   (Ac-Gly 1 , Glu(NH-hexyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 369)   (Ac-Gly 1 , Glu(NH-hexyl) 3,19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 370)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 371)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 3,19 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 372)   (Ac-Gly 1 , Glu(NH-hexyl) 9 hGhrelin(1-28)-NH 2 ; (SEQ ID: 373)   (Ac-Gly 1 , Ser(n-octanoyl) 20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 374)   (Ac-Gly 1 , Glu(NH-hexyl) 3,20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 375)   (Ac-Gly 1 , Glu(NH-hexyl) 3 , Ser(n-octanoyl) 20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 376)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 9 hGhrelin(1-28)-NH 2 ; (SEQ ID: 377)   (Ac-Gly 1 , Aib 2 , Glu(NH-hexyl) 3,20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 378)   (Ac-Gly 1 , Glu(NH-hexyl) 20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 379)   (Ac-Gly 1 , Glu(NH-hexyl) 3,20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 380)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 2 1hGhrelin(1-28)-NH 2 ; (SEQ ID: 381)   (Ac-Gly 1 , Aib 2,10 , Glu(NH-hexyl) 3,20 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 382)   (Ac-Gly 1 , Aib Glu(NH-hexyl) 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 385)   (1-Apc 1 , Aib 2,10 , Glu(NH-hexyl) 3 )-hGhrelin(1-28)NH 2 ; (SEQ ID: 385)   (Inp 1 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 386)   (Inp 1 , Aib 2 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 386)   (Inp 1 , Aib 2 , Glu(NH-hexyl) 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 387)   (Inp 1 , Aib 2,10 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 388)   (Inp 1 , Aib 2,8 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 389)   (Inp 1 , Aib 2 , Ser(n-octanoyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 390)   (Inp 1 , Ser(n-octanoyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 390)   (Inp 1 , Aib 2,8 , Ser(n-octanoyl) 17 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 389)   Ac-(Inp 1 , Aib Glu(NH-hexyl) 3 )hGhrelin(1-28)-NH 2 ;   Ac-(1-Apc 1 , Aib 2,10 , Glu(NH-hexyl) 3 )hGhrelin(1-28)-NH 2 ;   (Asp 3 (NH-heptyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 391)   (des-Ser 2 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 392)   (des-Gly 1 , des-Ser 2 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 392)   (Aib 1 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 393)   (Asp 3 (O-hexyl))hGhrelin(1-28)-NH 2 ; (SEQ ID: 394)   Ser 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 395)   (A5c 5 , Ser 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 396)   (Aib 2 ′ 4 , Sera, 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 397)   (n-octanoyl-Gly 1 , Ser 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 398)   (isobutyryl-Gly 1 , Ser 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 398)   (n-butyryl-Gly 1 , Ser 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 398)   (Aib 1 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 395)   (Aib 2,4 , Thr 3 , 4-Pal 9 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 397)   (n-octanoyl-Gly 1 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 399)   (isobutyryl-Gly 1 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 399)   (n-butyryl-Gly 1 , Thr 3 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 399)   (Ac-Gly 1 )hGhrelin(1-28)-NH 2 ; (SEQ ID: 400)   (Ac-Gly 1 , Ser 3 )hGhrelin(1-28)-NH 2 , (SEQ ID: 400)   (Aib 2 , Lys(myristyl) 17 )hGhrelin-(1-28)-NH 2 ; and (SEQ ID: 383)   [Gly(myristyl) 1 , Aib 2 , Lys(myristyl) 17 ]hGhrelin-(1-28)-NH 2 ; (SEQ ID: 384)   
       or a pharmaceutically acceptable salt thereof. 
     
     
         2 . A method of limiting myocardial damage during an acute myocardial infarction in a subject in need thereof according to  claim 1  wherein said analogue or said prodrug thereof is H-Inp-D-Bal-D-Trp-Phe-Apc-NH 2  (SEQ ID: 2) or a pharmaceutically acceptable salt thereof. 
     
     
         3 . The method of  claim 1 , wherein said peptidyl analogue of ghrelin or said prodrug thereof inhibits C-reactive protein. 
     
     
         4 . The method of  claim 3  wherein said C-reactive protein is synthesized in response to inflammation.
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