US2019359557A1PendingUtilityA1
Picolinamides with fungicidal activity
Est. expiryDec 30, 2034(~8.5 yrs left)· nominal 20-yr term from priority
Inventors:Chenglin YaoKevin G. MeyerYu LuBrian A. LoyDavid M. JonesRonald J. HeemstraJeffrey B. EppJohnathan E. DelorbeKyle A. DekorverJohn F. Daeuble, Sr.
C07C 69/02A61K 31/44A01N 37/44C07C 229/36C07C 229/08A01N 43/40C07D 213/81C07B 2200/07C07C 229/22C07C 2601/02C07C 271/22A01N 47/12A01N 43/10
70
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Claims
Abstract
The invention relates to picolinamides of Formula I and their use as fungicides.
Claims
exact text as granted — not AI-modifiedWhat is claimed is:
1 . A compound of Formula I
X is hydrogen or C(O)R 5 ;
Y is hydrogen, C(O)R 5 , or Q;
Q is
R 1 is CH 2 OCH 3 , or hydrogen or alkyl, where alkyl is optionally substituted with 0, 1 or multiple R 8 ;
R 2 is methyl;
R 3 is chosen from C(O)OCH 3 or alkyl, alkenyl, or aryl, each optionally substituted with 0, 1 or multiple R 8 ;
R 4 is chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 ;
R 5 is alkoxy, optionally substituted with 0, 1, or multiple R 8 ;
R 6 is chosen from hydrogen or alkoxy, where alkoxy is optionally substituted with 0, 1, or multiple R 8 ;
R 7 is chosen from hydrogen, C(O)R 9 , or CH 2 OC(O)R 9 ;
R 8 is chosen from hydrogen, alkyl, aryl, halo, alkenyl, or phenoxy, each optionally substituted with 0, 1, or multiple R 10 ,
R 9 is chosen from alkyl, alkoxy, or aryl, each optionally substituted with 0, 1, or multiple R 8 ;
R 10 is chosen from alkyl, aryl, halo, haloalkyl, haloaryl, alkenyl, or alkoxy;
R 11 is chosen from hydrogen or methyl.
2 . A compound according to claim 1 , wherein X and Y are hydrogen.
3 . A compound according to claim 2 , wherein R 1 and R 11 are independently chosen from hydrogen or methyl.
4 . A compound according to claim 2 , wherein R 3 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .
5 . A compound according to claim 2 , wherein R 4 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .
6 . A compound according to claim 2 , wherein R 1 and R 11 are independently chosen from hydrogen or methyl, R 3 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 , and R 4 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .
7 . A compound according to claim 1 , wherein X is C(O)R 5 and Y is hydrogen.
8 . A compound according to claim 7 , wherein R 1 and R 11 are independently chosen from hydrogen or methyl.
9 . A compound according to claim 7 , wherein R 3 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .
10 . A compound according to claim 7 , wherein R 4 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .
11 . A compound according to claim 7 , wherein R 1 and R 11 are independently chosen from hydrogen or methyl, R 3 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 , and R 4 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .
12 . A compound according to claim 1 , wherein X is hydrogen and Y is Q.
13 . A compound according to claim 12 , wherein R 7 is hydrogen.
14 . A compound according to claim 13 , wherein R 6 is OCH 3 .
15 . A compound according to claim 14 , wherein R 1 and R 11 are independently chosen from hydrogen or methyl.
16 . A compound according to claim 14 , wherein R 3 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .
17 . A compound according to claim 14 , wherein R 4 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .
18 . A compound according to claim 14 , wherein R 1 and R 11 are independently chosen from hydrogen or methyl, R 3 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 , and R 4 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .
19 . A compound according to claim 13 , wherein R 7 is C(O)R 9 , or CH 2 OC(O)R 9.
20 . A compound according to claim 19 , wherein R 1 and R 11 are independently chosen from hydrogen or methyl.
21 . A compound according to claim 19 , wherein R 3 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .
22 . A compound according to claim 19 , wherein R 4 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .
23 . A compound according to claim 19 , wherein R 1 and R 11 are independently chosen from hydrogen or methyl, R 3 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 , and R 4 is independently chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .Cited by (0)
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