US2021340190A1PendingUtilityA1
Flagellin compositions and uses
Est. expiryJul 30, 2034(~8 yrs left)· nominal 20-yr term from priority
Inventors:Vadim Mett
A61K 38/164A61K 2039/57A61P 9/10A61K 2039/55594A61K 2039/55516A61K 39/39A61K 2039/55583Y02A50/30A61P 37/08A61K 2039/55505A61P 37/02A61P 35/02A61K 45/06C07K 14/195A61P 37/04A61P 35/00A61P 31/04A61P 31/20A61P 31/16C07K 2319/00A61P 31/12A61K 2039/575A61K 39/0013A61P 43/00C07K 2319/21A61K 39/02
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Claims
Abstract
The present invention relates to compositions comprising improved flagellin derived constructs and methods of using the same in the treatment of various diseases.
Claims
exact text as granted — not AI-modified1 - 60 . (canceled)
61 . A composition comprising a polypeptide having an amino acid sequence that is about 95% identical to SEQ ID NO: 137.
62 . The composition of claim 61 , the composition comprising a polypeptide having an amino acid sequence that is about 98% sequence identical to SEQ ID NO: 137.
63 . The composition of claim 61 , the composition comprising a polypeptide having an amino acid sequence that is about 99% sequence identical to SEQ ID NO: 137.
64 . The composition of claim 61 , the composition comprising a polypeptide having an amino acid sequence that is SEQ ID NO: 137.
65 . A pharmaceutical composition, the pharmaceutical composition comprising a polypeptide having the amino acid sequence of SEQ ID NO: 137, and a pharmaceutically acceptable carrier.
66 . The composition of claim 61 , wherein the composition has reduced antigenicity and immunogenicity as compared to the polypeptide SEQ ID NO: 2.
67 . The composition of claim 61 , wherein the composition demonstrates improved pharmacokinetics as compared to the polypeptide SEQ ID NO: 2.
68 . The composition of claim 61 , wherein the composition activates TLR5 signaling at a level the same as, or similar to, that of the polypeptide SEQ ID NO: 2.
69 . The composition of claim 61 , wherein the polypeptide further comprises a N-terminal tag.
70 . The composition of claim 61 , wherein the polypeptide further comprises a C-terminal tag.
71 . The composition of claim 61 , wherein the composition induces NF-κB mediated expression of one or more of the cytokines selected from IL-6, IL-12, keratinocyte chemoattractant (KC), IL-10, G-CSF, MCP-1, TNF-α, MIG, and MIP-2.
72 . A pharmaceutical composition comprising the composition of claim 61 and a pharmaceutically acceptable carrier.
73 . A method of stimulating TLR5 signaling comprising administering to a subject in need thereof a composition comprising a polypeptide having an amino acid sequence that is about 95% sequence identical to SEQ ID NO: 137.
74 . The method of claim 73 , wherein the subject suffers from radiation-induced cellular damage.
75 . The method of claim 73 , wherein the subject has been subjected to a lethal dose of radiation.
76 . The method of claim 73 , wherein the subject is undergoing radiation treatment.
77 . The method of claim 73 , wherein the composition has reduced antigenicity and immunogenicity as compared to the polypeptide SEQ ID NO: 2.Cited by (0)
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