US8785390B2ActiveUtilityA1
Methods for treatment of Alzheimer's disease
Est. expiryJan 30, 2029(~2.6 yrs left)· nominal 20-yr term from priority
Inventors:Jan Johansson
C07K 14/785A61P 25/28A61K 38/1709A61K 38/00A61K 38/395
83
PatentIndex Score
4
Cited by
67
References
17
Claims
Abstract
An isolated protein selected from the group consisting of (i) proteins comprising an amino acid sequence having at least 70% identity to the C-terminal domain of lung surfactant protein C precursor (CTproSP-C, “CTC”) from a mammal; and (ii) proteins comprising an amino acid sequence having at least 70% identity to the Brichos domain of CTproSP-C from a mammal, is disclosed for treatment of Alzheimer's disease in a mammal, including man.
Claims
exact text as granted — not AI-modifiedThe invention claimed is:
1. A method of therapeutically treating or delaying progression of Alzheimer's disease in a subject in need thereof, comprising administering to the subject a therapeutically effective amount of an isolated protein, wherein the isolated protein delays or reduces amyloid fibril formation and aggregation of amyloid β peptide, and wherein the isolated protein is selected from:
(a) a protein comprising an amino acid sequence having all conserved residues of mammalian C-terminal domain of lung surfactant protein C precursor (CTproSP-C) (SEQ ID NO: 11) and having at least 70% identity to the CTproSP-C from human (SEQ ID NO: 2), bovine (SEQ ID NO: 5), rhesus (SEQ ID NO: 6), mouse (SEQ ID NO: 7), mink (SEQ ID NO: 8), rabbit (SEQ ID NO: 9) or rat (SEQ ID NO: 10); or
(b) a protein comprising an amino acid sequence having all conserved residues of the Brichos domain of mammalian CTproSP-C (SEQ ID NO: 18) and having at least 70% identity to the Brichos domain of CTproSP-C from human (SEQ ID NO: 4), bovine (SEQ ID NO: 12), rhesus (SEQ ID NO: 13), mouse (SEQ ID NO: 14), mink (SEQ ID NO: 15), rabbit (SEQ ID NO: 16) or rat (SEQ ID NO: 17).
2. The method of claim 1 , wherein the subject is human.
3. The method of claim 1 , wherein the isolated protein is selected from:
(a) a protein comprising an amino acid sequence having all conserved residues of mammalian C-terminal domain of lung surfactant protein C precursor (CTproSP-C) (SEQ ID NO: 11) and having at least 70% identity to human CTproSP-C (SEQ ID NO: 2); or
(b) a protein comprising an amino acid sequence having all conserved residues of the Brichos domain of mammalian CTproSP-C (SEQ ID NO: 18) and having at least 70% identity to the Brichos domain of human CTproSP-C (SEQ ID NO: 4).
4. The method of claim 1 , wherein the isolated protein has less than or equal to 200 amino acid residues.
5. The method of claim 4 , wherein the isolated protein has less than or equal to 150 amino acid residues.
6. The method of claim 1 , wherein the isolated protein has more than or equal to 90 amino acid residues.
7. The method of claim 6 , wherein the isolated protein has more than or equal to 100 amino acid residues.
8. The method of claim 1 , wherein the isolated protein is selected from the group consisting of:
(a) CTproSP-C from human (SEQ ID NO: 2), bovine (SEQ ID NO: 5), rhesus (SEQ ID NO: 6), mouse (SEQ ID NO: 7), mink (SEQ ID NO: 8), rabbit (SEQ ID NO: 9) or rat (SEQ ID NO: 10);
(b) the Brichos domain of CTproSP-C from human (SEQ ID NO: 4), bovine (SEQ ID NO: 12), rhesus (SEQ ID NO: 13), mouse (SEQ ID NO: 14), mink (SEQ ID NO: 15), rabbit (SEQ ID NO: 16) or rat (SEQ ID NO: 17); and
(c) an extended Brichos domain of human CTproSP-C having the amino acid sequence of SEQ ID NO: 21.
9. The method of claim 8 , wherein the isolated protein is selected from the group consisting of human CTproSP-C (SEQ ID NO: 2), the Brichos domain of human CTproSP-C (SEQ ID NO: 4), and the extended Brichos domain of human CTproSP-C having SEQ ID NO: 21.
10. The method of claim 1 , wherein a position corresponding to leucine-188 in human proSP-C (SEQ ID NO: 1) is not glutamine.
11. The method of claim 10 , wherein the position corresponding to leucine-188 in human proSP-C (SEQ ID NO: 1) is strictly conserved.
12. The method of claim 1 , wherein the isolated protein comprises an amino acid sequence having all conserved residues of the Brichos domain of mammalian CTproSP-C (SEQ ID NO: 18) and comprises an amino acid sequence having at least 70% identity to SEQ ID NO: 4, SEQ ID NO: 12, SEQ ID NO: 13, SEQ ID NO: 14, SEQ ID NO: 15 or SEQ ID NO: 16.
13. The method of claim 1 , wherein the isolated protein is selected from:
(a) a protein comprising an amino acid sequence having all conserved residues of mammalian CTproSP-C (SEQ ID NO: 11) and having at least 80% identity to the CTproSP-C from human (SEQ ID NO: 2), bovine (SEQ ID NO: 5), rhesus (SEQ ID NO: 6), mouse (SEQ ID NO: 7), mink (SEQ ID NO: 8), rabbit (SEQ ID NO: 9) or rat (SEQ ID NO: 10); or
(b) a protein comprising an amino acid sequence having all conserved residues of the Brichos domain of mammalian CTproSP-C (SEQ ID NO: 18) and having at least 80% identity to the Brichos domain of CTproSP-C from human (SEQ ID NO: 4), bovine (SEQ ID NO: 12), rhesus (SEQ ID NO: 13), mouse (SEQ ID NO: 14), mink (SEQ ID NO: 15), rabbit (SEQ ID NO: 16) or rat (SEQ ID NO: 17).
14. The method of claim 13 , wherein the isolated protein comprises an amino acid sequence having all conserved residues of the Brichos domain of mammalian CTproSP-C (SEQ ID NO: 18) and comprises an amino acid sequence having at least 80% identity to SEQ ID NO: 4, SEQ ID NO: 12, SEQ ID NO: 13, SEQ ID NO: 14, SEQ ID NO: 15 or SEQ ID NO: 16.
15. The method of claim 13 , wherein the isolated protein is selected from:
(a) a protein comprising an amino acid sequence having all conserved residues of mammalian CTproSP-C (SEQ ID NO: 11) and having at least 90% identity to the CTproSP-C from human (SEQ ID NO: 2), bovine (SEQ ID NO: 5), rhesus (SEQ ID NO: 6), mouse (SEQ ID NO: 7), mink (SEQ ID NO: 8), rabbit (SEQ ID NO: 9) or rat (SEQ ID NO: 10); or
(b) a protein comprising an amino acid sequence having all conserved residues of the Brichos domain of mammalian CTproSP-C (SEQ ID NO: 18) and having at least 90% identity to the Brichos domain of CTproSP-C from human (SEQ ID NO: 4), bovine (SEQ ID NO: 12), rhesus (SEQ ID NO: 13), mouse (SEQ ID NO: 14), mink (SEQ ID NO: 15), rabbit (SEQ ID NO: 16) or rat (SEQ ID NO: 17).
16. The method of claim 15 , wherein the isolated protein comprises an amino acid sequence having all conserved residues of the Brichos domain of mammalian CTproSP-C (SEQ ID NO: 18) and comprises an amino acid sequence having at least 90% identity to SEQ ID NO: 4, SEQ ID NO: 12, SEQ ID NO: 13, SEQ ID NO: 14, SEQ ID NO: 15 or SEQ ID NO: 16.
17. The method of claim 1 , wherein the isolated protein is selected from:
(a) a protein comprising an amino acid sequence having all conserved residues of mammalian CTproSP-C (SEQ ID NO: 11) and having at least 70% identity and at least 90% similarity to the CTproSP-C from human (SEQ ID NO: 2), bovine (SEQ ID NO: 5), rhesus (SEQ ID NO: 6), mouse (SEQ ID NO: 7), mink (SEQ ID NO: 8), rabbit (SEQ ID NO: 9) or rat (SEQ ID NO: 10); or
(b) a protein comprising an amino acid sequence having all conserved residues of the Brichos domain of mammalian CTproSP-C (SEQ ID NO: 18) and having at least 70% identity and at least 90% similarity to the Brichos domain of CTproSP-C from human (SEQ ID NO: 4), bovine (SEQ ID NO: 12), rhesus (SEQ ID NO: 13), mouse (SEQ ID NO: 14), mink (SEQ ID NO: 15), rabbit (SEQ ID NO: 16) or rat (SEQ ID NO: 17).Cited by (0)
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