Inventor
STOKBROEKX RAYMOND A
BE24 patents
Patents
24 patentsUS4329353AMay 11, 1982
1-(4-Aryl-cyclohexyl)piperidine derivatives, method of use thereof and pharmaceutical compositions thereof
JANSSEN PHARMACEUTICA NV58 citations95
US5637592AJun 10, 1997
Acyl derivatives of azolones
JANSSEN PHARMACEUTICA NV42 citations92
US5571811ANov 5, 1996
Sulfonamide derivatives of azolones
JANSSEN PHARMACEUTICA NV23 citations92
US5112825AMay 12, 1992
Antirhinoviral heteroamine-substituted pyridazines
JANSSEN PHARMACEUTICA NV25 citations92
US5001125AMar 19, 1991
Anti-virally active pyridazinamines
JANSSEN PHARMACEUTICA NV57 citations92
US4619931AOct 28, 1986
[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV31 citations92
US5231184AJul 27, 1993
Pridazinamine derivatives
JANSSEN PHARMACEUTICA NV54 citations91
US4992433AFeb 12, 1991
Novel pyridazinamine derivatives
JANSSEN PHARMACEUTICA NV46 citations91
US5100893AMar 31, 1992
Antipicornaviral pyridazinamines
JANSSEN PHARMACEUTICA NV23 citations90
US5070090ADec 3, 1991
Antipicorpaviral herterocyclic-substituted morpholinyl alkylphenol ethers
JANSSEN PHARMACEUTICA NV20 citations81
US4735942AApr 5, 1988
[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]-methyl]-1H-imidazoles and 1H-1,2,4-triazoles having antimicrobial properties
JANSSEN PHARMACEUTICA NV8 citations74
US4861785AAug 29, 1989
Benzoxazol-and benzothiazolamine derivatives, useful as anti-anoxic agents
JANSSEN PHARMACEUTICA NV12 citations73
US5292738AMar 8, 1994
Anti-virally active pyridazinamines
JANSSEN PHARMACEUTICA NV8 citations72
US5157035AOct 20, 1992
Anti-virally active pyridazinamines
JANSSEN PHARMACEUTICA NV6 citations72
US5106973AApr 21, 1992
Pyridzainamine derivatives
JANSSEN PHARMACEUTICA NV18 citations72
US4826848AMay 2, 1989
Antidepressive substituted N-[(4-piperidinyl)alkyl] bicyclic condensed oxazol- and thiazolamines
JANSSEN PHARMACEUTICA NV10 citations72
US4689330AAug 25, 1987
Antidepressive substituted N-[(4-piperidinyl)alkyl] bicyclic condensed oxazol- and thiazolamines
JANSSEN PHARMACEUTICA NV20 citations72
US4369184AJan 18, 1983
1-(Cyclohexyl)-4-aryl-4-piperidinecarboxylic acid derivatives
JANSSEN PHARMACEUTICA NV17 citations72
US5196535AMar 23, 1993
Intermediates for producing antipicornaviral pyridazinamines
JANSSEN PHARMACEUTICA NV14 citations71
US4861879AAug 29, 1989
[[4-[4-Phenyl-1-piperazinyl)phenoxymethyl]-1-3-dioxolan-2-yl]-methyl]-1H-imidazoles and 1H-1,2,4-triazoles
JANSSEN PHARMACEUTICA NV6 citations63
US5010198AApr 23, 1991
Intermediates for the synthesis of benzoxazol- and benzothiazolamine derivatives, useful as anti-anoxic agents
JANSSEN PHARMACEUTICA NV3 citations62
US5607932AMar 4, 1997
Heterocyclic derivatives of azolones
JANSSEN PHARMACEUTICA NV3 citations61
US4749702AJun 7, 1988
Antidepressive substituted N-[(4-piperidinyl)alkyl] bicyclic condensed oxazol- and thiazolamines
JANSSEN PHARMACEUTICA NV4 citations61
US5530011AJun 25, 1996
4-[(2-benzothiazolyl)methylamino]-α-[(3,4-difluorophenoxy)methyl]-1-piperidineethanol
JANSSEN PHARMACEUTICA NV1 citations51