Inventor
PITTS WILLIAM J
US46 patents
⚠️ This page may combine multiple inventors who share the name “PITTS WILLIAM J”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
BRISTOL MYERS SQUIBB CO
38 patentsUS6399773B1Jun 4, 2002
Compounds derived from an amine nucleus that are inhibitors of IMPDH enzyme
BRISTOL MYERS SQUIBB CO105 citations98
US6838559B2Jan 4, 2005
Purine inhibitors of phosphodiesterase (PDE) 7
BRISTOL MYERS SQUIBB CO79 citations97
US7683171B2Mar 23, 2010
1H-imidazo[4,5-d]thieno[3,2-b]pyridine based tricyclic compounds and pharmaceutical compositions comprising same
BRISTOL MYERS SQUIBB CO46 citations92
US7105667B2Sep 12, 2006
Fused heterocyclic compounds and use thereof
BRISTOL MYERS SQUIBB CO25 citations92
US7022849B2Apr 4, 2006
Quinazoline and pyrido[2,3-d]pyrimidine inhibitors of phosphodiesterase (PDE) 7
BRISTOL MYERS SQUIBB CO36 citations92
US8354398B2Jan 15, 2013
Substituted isoxazole compounds
BRISTOL MYERS SQUIBB CO13 citations84
US6596747B2Jul 22, 2003
Compounds derived from an amine nucleus and pharmaceutical compositions comprising same
BRISTOL MYERS SQUIBB CO20 citations84
US10913738B2Feb 9, 2021
Aminotriazolopyridines as kinase inhibitors
BRISTOL MYERS SQUIBB CO7 citations83
US9862715B2Jan 9, 2018
Thiazolyl- or thiadiazolyl-substituted pyridyl compounds useful as kinase inhibitors
BRISTOL MYERS SQUIBB CO5 citations83
US8987311B2Mar 24, 2015
Triazolyl-substituted pyridyl compounds useful as kinase inhibitors
BRISTOL MYERS SQUIBB CO14 citations83
US7601836B2Oct 13, 2009
Pyrido[2,3-D]pyrimidine inhibitors of phosphodiesterase (PDE) 7
BRISTOL MYERS SQUIBB CO11 citations83
US6919335B2Jul 19, 2005
Heterocycles that are inhibitors of IMPDH enzyme
BRISTOL MYERS SQUIBB CO16 citations83
US7109224B2Sep 19, 2006
Acyl guanidine compounds and use thereof
BRISTOL MYERS SQUIBB CO15 citations82
US7595317B2Sep 29, 2009
Barbituric acid derivatives as inhibitors of TNF-α converting enzyme (TACE) and/or matrix metalloproteinases
BRISTOL MYERS SQUIBB CO7 citations73
US9242975B2Jan 26, 2016
Heterocyclic-substituted pyridyl compounds useful as kinase inhibitors
BRISTOL MYERS SQUIBB CO4 citations72
US9657009B2May 23, 2017
Heteroaryl substituted pyridyl compounds useful as kinase modulators
BRISTOL MYERS SQUIBB CO4 citations71
US9546153B2Jan 17, 2017
Bicyclic heterocycle substituted pyridyl compounds useful as kinase modulators
BRISTOL MYERS SQUIBB CO5 citations71
US12157733B2Dec 3, 2024
Aminotriazolopyridines as kinase inhibitors
BRISTOL MYERS SQUIBB CO0 citations62
US11440913B2Sep 13, 2022
Aminoimidazopyridazines as kinase inhibitors
BRISTOL MYERS SQUIBB CO2 citations62
US10865191B2Dec 15, 2020
Heterocyclic compounds useful as modulators of TNF alpha
BRISTOL MYERS SQUIBB CO1 citations62
US9242976B2Jan 26, 2016
Thiazolyl- or thiadiazolyl-substituted pyridyl compounds useful as kinase inhibitors
BRISTOL MYERS SQUIBB CO1 citations62
US7737279B2Jun 15, 2010
1,6-dihydro-1,3,5,6-tetraaza-as-indacene based tricyclic compounds and pharmaceutical compositions comprising same
BRISTOL MYERS SQUIBB CO4 citations62
US7557211B2Jul 7, 2009
8H-imidazo[4,5-D]thiazolo[4,5-B]pyridine based tricyclic compounds and pharmaceutical compositions comprising same
BRISTOL MYERS SQUIBB CO2 citations62
US7176214B2Feb 13, 2007
Imidazo-fused oxazolo[4,5-β]pyridine and imidazo-fused thiazolo[4,5-β]pyridine based tricyclic compounds and pharmaceutical compositions comprising same
BRISTOL MYERS SQUIBB CO3 citations62
US7456194B2Nov 25, 2008
Imidazo-fused oxazolo [4,5-b]pyridine and imidazo-fused thiazolo[4,5-b]pyridine based tricyclic compounds and pharmaceutical compositions comprising same
BRISTOL MYERS SQUIBB CO5 citations60
US12275721B2Apr 15, 2025
Indazole carboxamides as kinase inhibitors
BRISTOL MYERS SQUIBB CO0 citations52
US12172975B2Dec 24, 2024
1H-indazole carboxamides as receptor-interacting protein kinase 1 inhibitors (RIPK1)
BRISTOL MYERS SQUIBB CO0 citations52
US10544133B2Jan 28, 2020
Heteroaryl substituted pyridyl compounds useful as kinase modulators
BRISTOL MYERS SQUIBB CO0 citations52
US12240840B2Mar 4, 2025
Amide-substituted heterocyclic compounds for the treatment of conditions related to the modulation of IL-12, IL-23 and/or IFN-alpha
BRISTOL MYERS SQUIBB CO0 citations51
US12084426B2Sep 10, 2024
Indazole carboxamides as kinase inhibitors
BRISTOL MYERS SQUIBB CO0 citations51
US11618753B2Apr 4, 2023
Aminopyrrolotriazines as kinase inhibitors
BRISTOL MYERS SQUIBB CO0 citations51
US10227340B2Mar 12, 2019
Thiazolyl- or thiadiazolyl-substituted pyridyl compounds useful as kinase inhibitors
BRISTOL MYERS SQUIBB CO0 citations51
US10023562B2Jul 17, 2018
Heteroaryl substituted pyridyl compounds useful as kinase modulators
BRISTOL MYERS SQUIBB CO0 citations51
US7981881B2Jul 19, 2011
Fused heterocyclic compounds and use thereof
BRISTOL MYERS SQUIBB CO0 citations51
US7384937B2Jun 10, 2008
Fused heterocyclic compounds and use thereof
BRISTOL MYERS SQUIBB CO0 citations51
US7329668B2Feb 12, 2008
Pyrazolopurine-based tricyclic compounds and pharmaceutical compositions comprising same
BRISTOL MYERS SQUIBB CO2 citations51
US10301306B2May 28, 2019
Substituted dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-ones as RIPK3 inhibitors
BRISTOL MYERS SQUIBB CO0 citations40
US9428511B2Aug 30, 2016
Imidazopyridazine JAK3 inhibitors and their use for the treatment of inflammatory and autoimmune diseases
BRISTOL MYERS SQUIBB CO0 citations40